Fragment library design, synthesis and expansion: nurturing a synthesis and training platform von Ray, Peter C., Kiczun, Michael, Huggett, Margaret, Lim, Andrew, Prati, Federica, Gilbert, Ian H., Wyatt, Paul G.

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Inhibiting Mycobacterium tuberculosis CoaBC by targeting an allosteric site von Mendes, Vitor, Green, Simon R., Evans, Joanna C., Hess, Jeannine, Blaszczyk, Michal, Spry, Christina, Bryant, Owain, Cory-Wright, James, Chan, Daniel S-H., Torres, Pedro H. M., Wang, Zhe, Nahiyaan, Navid, O’Neill, Sandra, Damerow, Sebastian, Post, John, Bayliss, Tracy, Lynch, Sasha L., Coyne, Anthony G., Ray, Peter C., Abell, Chris, Rhee, Kyu Y., Boshoff, Helena I. M., Barry, Clifton E., Mizrahi, Valerie, Wyatt, Paul G., Blundell, Tom L.

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Nitro-Mannich/Lactamization Cascades for the Direct Stereoselective Synthesis of Pyrrolidin-2-ones von Pelletier, Sophie M.-C, Ray, Peter C, Dixon, Darren J

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PE/PPE proteins mediate nutrient transport across the outer membrane of Mycobacterium tuberculosis von Wang, Qinglan, Boshoff, Helena I. M., Harrison, Justin R., Ray, Peter C., Green, Simon R., Wyatt, Paul G., Barry, Clifton E.

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Structure–Activity Relationships of Pyrazolo[1,5‑a]pyrimidin-7(4H)‑ones as Antitubercular Agents von Oh, Sangmi, Libardo, M. Daben J, Azeeza, Shaik, Pauly, Gary T, Roma, Jose Santinni O, Sajid, Andaleeb, Tateishi, Yoshitaka, Duncombe, Caroline, Goodwin, Michael, Ioerger, Thomas R, Wyatt, Paul G, Ray, Peter C, Gray, David W, Boshoff, Helena I. M, Barry, Clifton E

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Respiratory flexibility in response to inhibition of cytochrome C oxidase in Mycobacterium tuberculosis von Arora, Kriti, Ochoa-Montaño, Bernardo, Tsang, Patricia S, Blundell, Tom L, Dawes, Stephanie S, Mizrahi, Valerie, Bayliss, Tracy, Mackenzie, Claire J, Cleghorn, Laura A T, Ray, Peter C, Wyatt, Paul G, Uh, Eugene, Lee, Jinwoo, Barry, 3rd, Clifton E, Boshoff, Helena I

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Identification of Morpholino Thiophenes as Novel Mycobacterium tuberculosis Inhibitors, Targeting QcrB von Cleghorn, Laura A. T, Ray, Peter C, Odingo, Joshua, Kumar, Anuradha, Wescott, Heather, Korkegian, Aaron, Masquelin, Thierry, Lopez Moure, Abraham, Wilson, Caroline, Davis, Susan, Huggett, Margaret, Turner, Penelope, Smith, Alasdair, Epemolu, Ola, Zuccotto, Fabio, Riley, Jennifer, Scullion, Paul, Shishikura, Yoko, Ferguson, Liam, Rullas, Joaquin, Guijarro, Laura, Read, Kevin D, Green, Simon R, Hipskind, Phil, Parish, Tanya, Wyatt, Paul G

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Resistance of Mycobacterium tuberculosis to indole 4-carboxamides occurs through alterations in drug metabolism and tryptophan biosynthesis von Libardo, M. Daben J., Duncombe, Caroline J., Green, Simon R., Wyatt, Paul G., Thompson, Stephen, Ray, Peter C., Ioerger, Thomas R., Oh, Sangmi, Goodwin, Michael B., Boshoff, Helena I.M., Barry, Clifton E.

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Antitubercular 2-Pyrazolylpyrimidinones: Structure-Activity Relationship and Mode-of-Action Studies von de Melo, Candice Soares, Singh, Vinayak, Myrick, Alissa, Simelane, Sandile B., Taylor, Dale, Brunschwig, Christel, Lawrence, Nina, Schnappinger, Dirk, Engelhart, Curtis A., Kumar, Anuradha, Parish, Tanya, Su, Qin, Myers, Timothy G., Boshoff, Helena I. M., Barry, Clifton E., Sirgel, Frederick A., van Helden, Paul D., Buchanan, Kirsteen, Bayliss, Tracy, Green, Simon R., Ray, Peter C., Wyatt, Paul G., Basarab, Gregory S., Eyermann, Charles J., Chibale, Kelly, Ghorpade, Sandeep R.

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Inhibition of CorA-Dependent Magnesium Homeostasis Is Cidal in Mycobacterium tuberculosis von Park, Yumi, Ahn, Yong-Mo, Jonnala, Surendranadha, Oh, Sangmi, Fisher, Julia M, Goodwin, Michael B, Ioerger, Thomas R, Via, Laura E, Bayliss, Tracy, Green, Simon R, Ray, Peter C, Wyatt, Paul G, Barry, 3rd, Clifton E, Boshoff, Helena I

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2‑Mercapto-Quinazolinones as Inhibitors of Type II NADH Dehydrogenase and Mycobacterium tuberculosis: Structure–Activity Relationships, Mechanism of Action and Absorption, Distribu... von Murugesan, Dinakaran, Ray, Peter C., Bayliss, Tracy, Prosser, Gareth A., Harrison, Justin R., Green, Kirsteen, Soares de Melo, Candice, Feng, Tzu-Shean, Street, Leslie J., Chibale, Kelly, Warner, Digby F., Mizrahi, Valerie, Epemolu, Ola, Scullion, Paul, Ellis, Lucy, Riley, Jennifer, Shishikura, Yoko, Ferguson, Liam, Osuna-Cabello, Maria, Read, Kevin D., Green, Simon R., Lamprecht, Dirk A., Finin, Peter M., Steyn, Adrie J. C., Ioerger, Thomas R., Sacchettini, Jim, Rhee, Kyu Y., Arora, Kriti, Barry, Clifton E., Wyatt, Paul G., Boshoff, Helena I. M.

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Correction for Arora et al., "Respiratory Flexibility in Response to Inhibition of Cytochrome c Oxidase in Mycobacterium tuberculosis " von Arora, Kriti, Ochoa-Montaño, Bernardo, Tsang, Patricia S, Blundell, Tom L, Dawes, Stephanie S, Mizrahi, Valerie, Bayliss, Tracy, Mackenzie, Claire J, Cleghorn, Laura A T, Ray, Peter C, Wyatt, Paul G, Uh, Eugene, Lee, Jinwoo, Barry, 3rd, Clifton E, Boshoff, Helena I

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Screening of a Novel Fragment Library with Functional Complexity against Mycobacterium tuberculosis InhA von Prati, Federica, Zuccotto, Fabio, Fletcher, Daniel, Convery, Maire A., Fernandez‐Menendez, Raquel, Bates, Robert, Encinas, Lourdes, Zeng, Jingkun, Chung, Chun‐wa, De Dios Anton, Paco, Mendoza‐Losana, Alfonso, Mackenzie, Claire, Green, Simon R., Huggett, Margaret, Barros, David, Wyatt, Paul G., Ray, Peter C.

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Diastereoselective Synthesis of 1,3,5-Trisubstituted 4-Nitropyrrolidin-2-ones via a Nitro-Mannich/Lactamization Cascade von Pelletier, Sophie M.-C, Ray, Peter C, Dixon, Darren J

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Spirocycle MmpL3 Inhibitors with Improved hERG and Cytotoxicity Profiles as Inhibitors of Mycobacterium tuberculosis Growth von Ray, Peter C, Huggett, Margaret, Turner, Penelope A, Taylor, Malcolm, Cleghorn, Laura A. T, Early, Julie, Kumar, Anuradha, Bonnett, Shilah A, Flint, Lindsay, Joerss, Douglas, Johnson, James, Korkegian, Aaron, Mullen, Steven, Moure, Abraham L, Davis, Susan H, Murugesan, Dinakaran, Mathieson, Michael, Caldwell, Nicola, Engelhart, Curtis A, Schnappinger, Dirk, Epemolu, Ola, Zuccotto, Fabio, Riley, Jennifer, Scullion, Paul, Stojanovski, Laste, Massoudi, Lisa, Robertson, Gregory T, Lenaerts, Anne J, Freiberg, Gail, Kempf, Dale J, Masquelin, Thierry, Hipskind, Philip A, Odingo, Joshua, Read, Kevin D, Green, Simon R, Wyatt, Paul G, Parish, Tanya

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Targeting Mycobacterium tuberculosis CoaBC through Chemical Inhibition of 4′-Phosphopantothenoyl‑l‑cysteine Synthetase (CoaB) Activity von Evans, Joanna C, Murugesan, Dinakaran, Post, John M, Mendes, Vitor, Wang, Zhe, Nahiyaan, Navid, Lynch, Sasha L, Thompson, Stephen, Green, Simon R, Ray, Peter C, Hess, Jeannine, Spry, Christina, Coyne, Anthony G, Abell, Chris, Boshoff, Helena I. M, Wyatt, Paul G, Rhee, Kyu Y, Blundell, Tom L, Barry, Clifton E, Mizrahi, Valerie

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Triazine and pyrimidine based ROCK inhibitors with efficacy in spontaneous hypertensive rat model von Ho, Koc-Kan, Beasley, James R., Belanger, Laura, Black, Darcey, Chan, Jui-Hsiang, Dunn, David, Hu, Bing, Klon, Anthony, Kultgen, Steven G., Ohlmeyer, Michael, Parlato, Susan M., Ray, Peter C., Pham, Quynhchi, Rong, Yajing, Roughton, Andrew L., Walker, Tiffany L., Wright, Jane, Xu, Kai, Xu, Yan, Zhang, Limei, Webb, Maria

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The role of phthiocerol dimycoserosate and the PE/PPE protein family in outer cell wall permeability in Mycobacterium tuberculosis von Wang, Qinglan, Boshoff, Helena I. M., Harrison, Justin R., Ray, Peter C., Green, Simon R., Wyatt, Paul G., Barry, Clifton E.

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Essential but Not Vulnerable: Indazole Sulfonamides Targeting Inosine Monophosphate Dehydrogenase as Potential Leads against Mycobacterium tuberculosis von Park, Yumi, Pacitto, Angela, Bayliss, Tracy, Cleghorn, Laura A. T, Wang, Zhe, Hartman, Travis, Arora, Kriti, Ioerger, Thomas R, Sacchettini, Jim, Rizzi, Menico, Donini, Stefano, Blundell, Tom L, Ascher, David B, Rhee, Kyu, Breda, Ardala, Zhou, Nian, Dartois, Veronique, Jonnala, Surendranadha Reddy, Via, Laura E, Mizrahi, Valerie, Epemolu, Ola, Stojanovski, Laste, Simeons, Fred, Osuna-Cabello, Maria, Ellis, Lucy, MacKenzie, Claire J, Smith, Alasdair R. C, Davis, Susan H, Murugesan, Dinakaran, Buchanan, Kirsteen I, Turner, Penelope A, Huggett, Margaret, Zuccotto, Fabio, Rebollo-Lopez, Maria Jose, Lafuente-Monasterio, Maria Jose, Sanz, Olalla, Diaz, Gracia Santos, Lelièvre, Joël, Ballell, Lluis, Selenski, Carolyn, Axtman, Matthew, Ghidelli-Disse, Sonja, Pflaumer, Hannah, Bösche, Markus, Drewes, Gerard, Freiberg, Gail M, Kurnick, Matthew D, Srikumaran, Myron, Kempf, Dale J, Green, Simon R, Ray, Peter C, Read, Kevin, Wyatt, Paul, Barry, Clifton E, Boshoff, Helena I

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Liver X receptor agonists as a treatment for atherosclerosis von Bennett, D Jonathan, Cooke, Andrew J, Edwards, Andrew S, Moir, Elizabeth, Ray, Peter C

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