Discovery of Selective Estrogen Receptor Covalent Antagonists for the Treatment of ERα WT and ERα MUT Breast Cancer von Puyang, Xiaoling, Furman, Craig, Zheng, Guo Zhu, Wu, Zhenhua J, Banka, Deepti, Aithal, Kiran, Agoulnik, Sergei, Bolduc, David M, Buonamici, Silvia, Caleb, Benjamin, Das, Subhasree, Eckley, Sean, Fekkes, Peter, Hao, Ming-Hong, Hart, Andrew, Houtman, René, Irwin, Sean, Joshi, Jaya J, Karr, Craig, Kim, Amy, Kumar, Namita, Kumar, Pavan, Kuznetsov, Galina, Lai, Weidong G, Larsen, Nicholas, Mackenzie, Crystal, Martin, Lesley-Ann, Melchers, Diana, Moriarty, Alyssa, Nguyen, Tuong-Vi, Norris, John, O'Shea, Morgan, Pancholi, Sunil, Prajapati, Sudeep, Rajagopalan, Sujatha, Reynolds, Dominic J, Rimkunas, Victoria, Rioux, Nathalie, Ribas, Ricardo, Siu, Amy, Sivakumar, Sasirekha, Subramanian, Vanitha, Thomas, Michael, Vaillancourt, Frédéric H, Wang, John, Wardell, Suzanne, Wick, Michael J, Yao, Shihua, Yu, Lihua, Warmuth, Markus, Smith, Peter G, Zhu, Ping, Korpal, Manav

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Abstract 4418: Pharmacological characterization of a preclinical candidate covalently inhibiting CDK12 von Poddutoori, Ramulu, Rajagopalan, Sujatha, Mukherjee, Subhendu, Marappan, Sivapriya, D. S., Samiulla, Sivakumar, Sasirekha, Nayak, Shilpa S, M V, Ravindra, TS, Devaraja, Kondela, Srinivas, Tgore, Suraj, Dhudashiya, Amit A, K. B, Charamanna, A B, Aravind, A, Amith, S, Pavithra, Pathange, Hema Sankar, Antony, Thomas, Jaleel, Mahaboobi, Giri, Sanjeev, Daginakatte, Girish, Nellore, Kavitha, Chelur, Shekar, Ramachandra, Murali, Samajdar, Susanta

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Abstract 1392: Preclinical In vivo evaluation of efficacy, pharmacokinetics and pharmacodynamics of novel PRMT5 inhibitors in multiple tumor models von Chikkanna, Dinesh, Panigrahi, Sunil Kumar, Rajagopalan, Sujatha, Sammeta, Srinivasa Raju, Chawla, Darshan, S, Pavithra, D.S, Samiulla, Prasanna, Angelene, Chand, Priyabrata, Aithal, Kiran, Marri, Sai Sudheer, Kumar, Naveen, Ganipisetty, Srinivasa Rao, Mutyala, Raju, Rao, Kasieswara, Antony, Thomas, Daginakatte, Girish, Lakshminarasimhan, Anirudha, R, Mohan, K, Narasihmarao, Chelur, Shekar, Pandit, Chetan, Samajdar, Susanta, Ramachandra, Murali

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Abstract 2384: Preclinical evaluation of PD and efficacy of novel potent selective and orally bioavailable CDK12 covalent inhibitors in TNBC model von Poddutoori, Ramulu, Rajagopalan, Sujatha, Mukherjee, Subhendu, Marappan, Sivapriya, S, Samiulla D, Sivakumar, Sasirekha, Nayak, Shilpa S., V, Ravindra M., Murtuza, Hadianawala, S, Devaraja T., Kondela, Srinivas, Tgore, Suraj, Dhudashiya, Amit A., B, Charamanna K., Antony, Thomas, Daginakatte, Girish, Giri, Sanjeev, Chelur, Shekar, Ramachandra, Murali, Pandit, Chetan, Samajdar, Susanta

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3‑Alkoxy-pyrrolo[1,2‑b]pyrazolines as Selective Androgen Receptor Modulators with Ideal Physicochemical Properties for Transdermal Administration von Ullrich, Thomas, Sasmal, Sanjita, Boorgu, Venkatesham, Pasagadi, Srinivasu, Cheera, Srisailam, Rajagopalan, Sujatha, Bhumireddy, Archana, Shashikumar, Dhanya, Chelur, Shekar, Belliappa, Charamanna, Pandit, Chetan, Krishnamurthy, Narasimharao, Mukherjee, Subhendu, Ramanathan, Anuradha, Ghadiyaram, Chakshusmathi, Ramachandra, Murali, Santos, Paulo G, Lagu, Bharat, Bock, Mark G, Perrone, Mark H, Weiler, Sven, Keller, Hansjoerg

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Abstract B165: Potent selective and orally bioavailable inhibition of CDK12 by novel covalent inhibitors von Poddutoori, Ramulu, Rajagopalan, Sujatha, Mukherjee, Subhendu, Marappan, Sivapriya, D S, Samiulla, Kasturi, Venkateswarlu, Sivakumar, Sasirekha, Nayak, Shilpa, M V, Ravindra, Tgore, Suraj, Dhudashiya, Amit, K B, Charamanna, Antony, Thomas, M, Mahaboobi, Giri, Sanjeev, Daginakatte, Girish C., Chelur, Shekar, Ramachandra, Murali, Pandit, Chetan, Samajdar, Susanta

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Abstract A174: Novel inhibitors of protein arginine methyltransferase 5 (PRMT5) for the treatment of solid tumors von Chikkanna, Dinesh, Panigrahi, Sunil Kumar, Rajagopalan, Sujatha, Sammeta, Srinivasa Raju, Lakshminarasimhan, Anirudha, R, Mohan, K, Narasihmarao, Chawla, Darshan, Bhat, Harsha, Kasturi, Venkateswarlu, D.S, Samiulla, Prasanna, Angelene, Aithal, Kiran, Chand, Priyabrata Chand, Kumar, Naveen, Marri, Sai Sudheer, Ganipisetty, Srinivasa Rao, N, Kasieswara Rao, Mutyala, Raju, Neerukattu, Nageswara Rao, K, Nithesh, Amin, Ramya, Gorade, Priyanka Machhindra, Antony, Thomas, Daginakatte, Girish, Chelur, Shekar, Pandit, Chetan, Samajdar, Susanta, Ramachandra, Murali

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Abstract B164: Identification of a novel highly selective and orally bioavailable preclinical candidate for CDK7 covalent inhibition von Poddutoori, Ramulu, Khare Satyam, Leena, Mukherjee, Subhendu, Marappan, Sivapriya, Gopinath, Sreevalsam, KB, Charamanna, Kaza, Lakshmi Narayana, Pothuganti, Manoj Kumar, Rajagopalan, Sujatha, Sivakumar, Sasirekha, E N, Bharath, A B, Aravind, A, Amith, M V, Ravindra, Tgore, Suraj, Antony, Thomas, Pandit, Chetan, Chelur, Shekar, Daginakatte, Girish, Ramachandra, Murali, Samajdar, Susanta

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Discovery of 7-azaindole based anaplastic lymphoma kinase (ALK) inhibitors: Wild type and mutant (L1196M) active compounds with unique binding mode von Gummadi, Venkateshwar Rao, Rajagopalan, Sujatha, Looi, Chung-Yeng, Paydar, Mohammadjavad, Renukappa, Girish Aggunda, Ainan, Bharathi Raja, Krishnamurthy, Narasimha Rao, Panigrahi, Sunil Kumar, Mahasweta, Kumari, Raghuramachandran, Sangeetha, Rajappa, Manoj, Ramanathan, Anuradha, Lakshminarasimhan, Anirudha, Ramachandra, Murali, Wong, Pooi-Fong, Mustafa, Mohammad Rais, Nanduri, Srinivas, Hosahalli, Subramanya

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An Assessment of Ingestion Dose due to the Intake of ^210Po and ^210Pb through Drinking Water of Eloor, Ernakulam District, Kerala, India von A. G. Umadev Dhanya Balakrishnan Jose P. Abraham M. Rajagopalan M. George P. Dharmalingam Sujatha Radhakrishnan M. Harikumar

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VISUAL CHANGES IN GAIT IN INDIVIDUALS WITH PARKINSON DISEASE von Sujatha, J

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