Mono-Oxidation of Bidentate Bis-phosphines in Catalyst Activation: Kinetic and Mechanistic Studies of a Pd/Xantphos-Catalyzed C–H Functionalization von Ji, Yining, Plata, R. Erik, Regens, Christopher S, Hay, Michael, Schmidt, Michael, Razler, Thomas, Qiu, Yuping, Geng, Peng, Hsiao, Yi, Rosner, Thorsten, Eastgate, Martin D, Blackmond, Donna G

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Highly Efficient Asymmetric Synthesis of Sitagliptin von Hansen, Karl B, Hsiao, Yi, Xu, Feng, Rivera, Nelo, Clausen, Andrew, Kubryk, Michele, Krska, Shane, Rosner, Thorsten, Simmons, Bryon, Balsells, Jaume, Ikemoto, Nori, Sun, Yongkui, Spindler, Felix, Malan, Christophe, Grabowski, Edward J. J, Armstrong, Joseph D

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Detection and Elimination of Product Inhibition from the Asymmetric Catalytic Hydrogenation of Enamines von Hansen, Karl B, Rosner, Thorsten, Kubryk, Michele, Dormer, Peter G, Armstrong, Joseph D

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Asymmetric synthesis of ENT-03, the predicted mammalian ortholog of the dog fish shark aminosterol trodusquemine (MSI-1436) von Kinney, William A., Phillip Cox, D., Jones, Stephen R., Hessler, Edward J., Karnes, Harold A., Fevig, Thomas L., Hewitt, Bradley D., Sullivan, Ryan, Tseng, Nai-Wen, Pasion, Edward, Beale, Thomas, Rosner, Thorsten, Crouch, Ian T., D’Ambrosio, Stephen, Wade, Peter, Chen, Hui, Gao, Qi, Thompson, Andrew S., Muzzio, Miguel, Barbut, Denise, Zasloff, Michael A.

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Adventures in Atropisomerism: Total Synthesis of a Complex Active Pharmaceutical Ingredient with Two Chirality Axes von Beutner, Gregory, Carrasquillo, Ronald, Geng, Peng, Hsiao, Yi, Huang, Eric C, Janey, Jacob, Katipally, Kishta, Kolotuchin, Sergei, La Porte, Thomas, Lee, Andrew, Lobben, Paul, Lora-Gonzalez, Federico, Mack, Brendan, Mudryk, Boguslaw, Qiu, Yuping, Qian, Xinhua, Ramirez, Antonio, Razler, Thomas M, Rosner, Thorsten, Shi, Zhongping, Simmons, Eric, Stevens, Jason, Wang, Jianji, Wei, Carolyn, Wisniewski, Steven R, Zhu, Ye

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An Efficient Asymmetric Synthesis of an Estrogen Receptor Modulator by Sulfoxide-Directed Borane Reduction von Song, Zhiguo J., King, Anthony O., Waters, Marjorie S., Lang, Fengrui, Zewge, Daniel, Bio, Matthew, Leazer, Johnnie L., Javadi, Gary, Kassim, Amude, Tschaen, David M., Reamer, Robert A., Rosner, Thorsten, Chilenski, Jennifer R., Mathre, David J., Volante, R. P., Tillyer, Richard, Trost, Barry M.

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Highly Efficient Asymmetric Synthesis of Sitagliptin (vol 131, pg 8798, 2009) von Hansen, Karl B., Hsiao, Yi, Xu, Feng, Rivera, Nelo, Clausen, Andrew, Kubryk, Michele, Krska, Shane, Rosner, Thorsten, Simmons, Bryon, Balsells, Jaume, Ikemoto, Nori, Sun, Yongkui, Spindler, Felix, Malan, Christophe, Grabowski, Edward J. J., Armstrong, Joseph D.

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C–H Arylation in the Formation of a Complex Pyrrolopyridine, the Commercial Synthesis of the Potent JAK2 Inhibitor, BMS-911543 von Fox, Richard J, Cuniere, Nicolas L, Bakrania, Lopa, Wei, Carolyn, Strotman, Neil A, Hay, Michael, Fanfair, Dayne, Regens, Christopher, Beutner, Gregory L, Lawler, Michael, Lobben, Paul, Soumeillant, Maxime C, Cohen, Benjamin, Zhu, Keming, Skliar, Dimitri, Rosner, Thorsten, Markwalter, Chester E, Hsiao, Yi, Tran, Kristy, Eastgate, Martin D

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Enantioselective Synthesis of a γ‑Secretase Modulator via Vinylogous Dynamic Kinetic Resolution von Strotman, Neil A, Ramirez, Antonio, Simmons, Eric M, Soltani, Omid, Parsons, Andrew T, Fan, Yu, Sawyer, James R, Rosner, Thorsten, Janey, Jacob M, Tran, Kristy, Li, Jun, La Cruz, Thomas E, Pathirana, Charles, Ng, Alicia T, Deerberg, Joerg

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Correction to “Highly Efficient Asymmetric Synthesis of Sitagliptin” von Hansen, Karl B, Hsiao, Yi, Xu, Feng, Rivera, Nelo, Clausen, Andrew, Kubryk, Michele, Krska, Shane, Rosner, Thorsten, Simmons, Bryon, Balsells, Jaume, Ikemoto, Nori, Sun, Yongkui, Spindler, Felix, Malan, Christophe, Grabowski, Edward J. J

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Combining Solid-State and Solution Calorimetry for the Gibbs Free Energy Calculation of Polymorphs To Determine the Relative Stability and Solubility von Hsieh, Daniel S, Roberts, Daniel, Rosner, Thorsten, Rosenbaum, Tamar, Lai, Chiajen, Gao, Qi

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Mild and General Method for the α-Arylation of Heteroaromatic Ketones von Desai, Lopa V, Ren, Danan T, Rosner, Thorsten

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Highly Efficient Synthesis of β-Amino Acid Derivatives via Asymmetric Hydrogenation of Unprotected Enamines von Hsiao, Yi, Rivera, Nelo R, Rosner, Thorsten, Krska, Shane W, Njolito, Eugenia, Wang, Fang, Sun, Yongkui, Armstrong, Joseph D, Grabowski, Edward J. J, Tillyer, Richard D, Spindler, Felix, Malan, Christophe

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Kinetic Studies of Heck Coupling Reactions Using Palladacycle Catalysts: Experimental and Kinetic Modeling of the Role of Dimer Species von Rosner, Thorsten, Le Bars, Joel, Pfaltz, Andreas, Blackmond, Donna G

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Development of a scalable palladium-catalyzed α-arylation process for the synthesis of a CGRP antagonist von Desai, Lopa V., Hay, Michael B., Leahy, David K., Wei, Carolyn, Fanfair, Dayne, Rosner, Thorsten, Hsiao, Yi

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Efficient and Scalable Enantioselective Synthesis of a CGRP Antagonist von Leahy, David K, Fan, Yu, Desai, Lopa V, Chan, Collin, Zhu, Jason, Luo, Guanglin, Chen, Ling, Hanson, Ronald L, Sugiyama, Masano, Rosner, Thorsten, Cuniere, Nicolas, Guo, Zhiwei, Hsiao, Yi, Gao, Qi

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Multiparallel microfluidic high-performance liquid chromatography for high-throughput normal-phase chiral analysis von Sajonz, Peter, Schafer, Wes, Gong, Xiaoyi, Shultz, Scott, Rosner, Thorsten, Welch, Christopher J.

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Observation of Unusual Kinetics in Heck Reactions of Aryl Halides:  The Role of Non-Steady-State Catalyst Concentration von Rosner, Thorsten, Pfaltz, Andreas, Blackmond, Donna G

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Discovery of Indazoles as Potent, Orally Active Dual Neurokinin 1 Receptor Antagonists and Serotonin Transporter Inhibitors for the Treatment of Depression von Degnan, Andrew P, Tora, George O, Huang, Hong, Conlon, David A, Davis, Carl D, Hanumegowda, Umesh M, Hou, Xiaoping, Hsiao, Yi, Hu, Joanna, Krause, Rudolph, Li, Yu-Wen, Newton, Amy E, Pieschl, Rick L, Raybon, Joseph, Rosner, Thorsten, Sun, Jung-Hui, Taber, Matthew T, Taylor, Sarah J, Wong, Michael K, Zhang, Huiping, Lodge, Nicholas J, Bronson, Joanne J, Macor, John E, Gillman, Kevin W

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On the Mechanism of an Asymmetric α,β-Unsaturated Carboxylic Acid Hydrogenation:  Application to the Synthesis of a PGD2 Receptor Antagonist von Tellers, David M, McWilliams, J. Christopher, Humphrey, Guy, Journet, Michel, DiMichele, Lisa, Hinksmon, Joseph, McKeown, Arlene E, Rosner, Thorsten, Sun, Yongkui, Tillyer, Richard D

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