Pd-Catalyzed Cross-Coupling Reactions Promoted by Biaryl Phosphorinane Ligands von Laffoon, Summer D, Chan, Vincent S, Fickes, Michael G, Kotecki, Brian, Ickes, Andrew R, Henle, Jeremy, Napolitano, José G, Franczyk, Thaddeus S, Dunn, Travis B, Barnes, David M, Haight, Anthony R, Henry, Rodger F, Shekhar, Shashank

Volltext

Efficient Co-crystal Screening Using Solution-Mediated Phase Transformation von Zhang, Geoff G.Z., Henry, Rodger F., Borchardt, Thomas B., Lou, Xiaochun

Volltext

Synthon Hierarchies in Crystal Forms Composed of Theophylline and Hydroxybenzoic Acids: Cocrystal Screening via Solution-Mediated Phase Transformation von Bučar, Dejan-Krešimir, Henry, Rodger F, Zhang, Geoff G. Z, MacGillivray, Leonard R

Volltext

Cocrystals of Caffeine and Hydroxybenzoic Acids Composed of Multiple Supramolecular Heterosynthons: Screening via Solution-Mediated Phase Transformation and Structural Characteriza... von Bučar, Dejan-Krešimir, Henry, Rodger F, Lou, Xiaochun, Duerst, Richard W, MacGillivray, Leonard R, Zhang, Geoff G. Z

Volltext

Pharmaceutical Nano-Cocrystals: Sonochemical Synthesis by Solvent Selection and Use of a Surfactant von Sander, John R.G, Bučar, Dejan-Krešimir, Henry, Rodger F, Zhang, Geoff G.Z, MacGillivray, Leonard R

Volltext

Ritonavir Form III: A New Polymorph After 24 Years von Yao, Xin, Henry, Rodger F., Zhang, Geoff G.Z.

Volltext

Cocrystal screening in minutes by solution-mediated phase transformation (SMPT): Preparation and characterization of ketoconazole cocrystals with nine aliphatic dicarboxylic acids von Yu, Junguang, Henry, Rodger F., Zhang, Geoff G.Z.

Volltext

Inhibiting Sublimation of Thymol by Cocrystallization von Zu, Hui, Henry, Rodger F., Zhang, Geoff G.Z., MacGillivray, Leonard R.

Volltext

Co-Crystals of Caffeine and Hydroxy-2-naphthoic Acids:  Unusual Formation of the Carboxylic Acid Dimer in the Presence of a Heterosynthon von Bučar, Dejan-Krešimir, Henry, Rodger F., Lou, Xiaochun, Duerst, Richard W., Borchardt, Thomas B., MacGillivray, Leonard R., Zhang, Geoff G. Z.

Volltext

Implications of the Conformationally Flexible, Macrocyclic Structure of the First-Generation, Direct-Acting Anti-Viral Paritaprevir on Its Solid Form Complexity and Chameleonic Beh... von Sheikh, Ahmad Y., Mattei, Alessandra, Miglani Bhardwaj, Rajni, Hong, Richard S., Abraham, Nathan S., Schneider-Rauber, Gabriela, Engstrom, Kenneth M., Diwan, Moiz, Henry, Rodger F., Gao, Yi, Juarez, Vivian, Jordan, Erin, DeGoey, David A., Hutchins, Charles W.

Volltext

Pd-Catalyzed Cross-Coupling of Hindered, Electron-Deficient Anilines with Bulky (Hetero)aryl Halides Using Biaryl Phosphorinane Ligands von Wilders, Alison M, Henle, Jeremy, Haibach, Michael C, Swiatowiec, Rafal, Bien, Jeffrey, Henry, Rodger F, Asare, Shardrack O, Wall, Amanda L, Shekhar, Shashank

Volltext

Small Molecule IL-36γ Antagonist as a Novel Therapeutic Approach for Plaque Psoriasis von Todorović, Viktor, Su, Zhi, Putman, C. Brent, Kakavas, Stevan J., Salte, Katherine M., McDonald, Heath A., Wetter, Joseph B., Paulsboe, Stephanie E., Sun, Qi, Gerstein, Clare E., Medina, Limary, Sielaff, Bernhard, Sadhukhan, Ramkrishna, Stockmann, Henning, Richardson, Paul L., Qiu, Wei, Argiriadi, Maria A., Henry, Rodger F., Herold, J. Martin, Shotwell, J. Brad, McGaraughty, Steve P., Honore, Prisca, Gopalakrishnan, Sujatha M., Sun, Chaohong C., Scott, Victoria E.

Volltext

Overcoming Bioavailability Challenges of Dasabuvir and Enabling a Triple-Combination Direct-Acting Antiviral HCV Regimen through a Salt of Very Weak Acid for Oral Delivery von Chen, Shuang, Gao, Yi, Lou, Xiaochun, Henry, Rodger F., Stolarik, DeAnne F., Lipert, Maya P., Sheikh, Ahmad Y., Zhang, Geoff G. Z.

Volltext

Pharmaceutical Development Challenges in a Beyond Rule of Five Prodrug: Case Study of ABBV-167, Phosphate Prodrug of Venetoclax von Hong, Richard, Nie, Haichen, Henry, Rodger F., Garner, Sean M., Catron, Nathaniel D., Hertzler, Russell L., Souers, Andrew J., Sheikh, Ahmad Y., Chen, Shuang

Volltext

Discovery of ABBV-3373, an Anti-TNF Glucocorticoid Receptor Modulator Immunology Antibody Drug Conjugate von Hobson, Adrian D., McPherson, Michael J., Hayes, Martin E., Goess, Christian, Li, Xiang, Zhou, Jian, Wang, Zhongyuan, Yu, Yajie, Yang, Jindong, Sun, Liang, Zhang, Qiang, Qu, Pei, Yang, Shi, Hernandez, Axel, Bryant, Shaughn H., Mathieu, Suzanne L., Bischoff, Agnieszka K., Fitzgibbons, Julia, Santora, Ling C., Wang, Lu, Wang, Lu, Fettis, Margaret M., Li, Xiaofeng, Marvin, Christopher C., Wang, Zhi, Patel, Meena V., Schmidt, Diana L., Li, Tongmei, Randolph, John T., Henry, Rodger F., Graff, Candace, Tian, Yu, Aguirre, Ana L., Shrestha, Anurupa

Volltext

Enabling Suzuki-Miyaura coupling of Lewis-basic arylboronic esters with a nonprecious metal catalyst von Haibach, Michael C, Ickes, Andrew R, Tcyrulnikov, Sergei, Shekhar, Shashank, Monfette, Sebastien, Swiatowiec, Rafal, Kotecki, Brian J, Wang, Jason, Wall, Amanda L, Henry, Rodger F, Hansen, Eric C

Volltext

Enabling, Decagram-Scale Synthesis of Macrocyclic MCL‑1 Inhibitor ABBV-467 von Brady, Patrick B., Sorensen, Bryan K., Risi, Roberto M., Curtin, Michael L., Mantei, Robert A., Florjancic, Alan S., Mastracchio, Anthony, Ji, Cheng, Kunzer, Aaron R., Lai, Chunqiu, Storer, Gregory E., Chan, Vincent S., Henry, Rodger F., Souers, Andrew J., Michaelides, Michael R., Judd, Andrew S., Hansen, T. Matthew

Volltext

Scalable Synthesis and Isolation of the Four Stereoisomers of Methyl 1-Amino-3-(4-bromophenyl)cyclopentanecarboxylate, Useful Intermediates for the Synthesis of S1P1 Receptor Agoni... von Wallace, Grier A, Gordon, Thomas D, Hayes, Martin E, Konopacki, Donald B, Fix-Stenzel, Shannon R, Zhang, Xiaolei, Grongsaard, Pintipa, Cusack, Kevin P, Schaffter, Lisa M, Henry, Rodger F, Stoffel, Robert H

Volltext

Correction to “Discovery of ABBV-3373, an Anti-TNF Glucocorticoid Receptor Modulator Immunology Antibody Drug Conjugate” von Hobson, Adrian D., McPherson, Michael J., Hayes, Martin E., Goess, Christian, Li, Xiang, Zhou, Jian, Wang, Zhongyuan, Yu, Yajie, Yang, Jindong, Sun, Liang, Zhang, Qiang, Qu, Pei, Yang, Shi, Hernandez, Axel, Bryant, Shaughn H., Mathieu, Suzanne L., Bischoff, Agnieszka K., Fitzgibbons, Julia, Santora, Ling C., Wang, Lu, Wang, Lu, Fettis, Margaret M., Li, Xiaofeng, Marvin, Christopher C., Wang, Zhi, Patel, Meena V., Schmidt, Diana L., Li, Tongmei, Randolph, John T., Henry, Rodger F., Graff, Candace, Tian, Yu, Aguirre, Ana L., Shrestha, Anurupa

Volltext

Targeting lysine specific demethylase 4A (KDM4A) tandem TUDOR domain – A fragment based approach von Upadhyay, Anup K., Judge, Russell A., Li, Leiming, Pithawalla, Ron, Simanis, Justin, Bodelle, Pierre M., Marin, Violeta L., Henry, Rodger F., Petros, Andrew M., Sun, Chaohong

Volltext