Spiroindolines identify the vesicular acetylcholine transporter as a novel target for insecticide action von Sluder, Ann, Shah, Sheetal, Cassayre, Jérôme, Clover, Ralph, Maienfisch, Peter, Molleyres, Louis-Pierre, Hirst, Elizabeth A, Flemming, Anthony J, Shi, Min, Cutler, Penny, Stanger, Carole, Roberts, Richard S, Hughes, David J, Flury, Thomas, Robinson, Michael P, Hillesheim, Elke, Pitterna, Thomas, Cederbaum, Fredrik, Worthington, Paul A, Crossthwaite, Andrew J, Windass, John D, Currie, Richard A, Earley, Fergus G P

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Structure–activity relationships (SAR) and structure–kinetic relationships (SKR) of bicyclic heteroaromatic acetic acids as potent CRTh2 antagonists III: The role of a hydrogen-bon... von Alonso, Juan Antonio, Andrés, Miriam, Bravo, Mónica, Buil, Maria Antonia, Calbet, Marta, Castro, Jordi, Eastwood, Paul R., Esteve, Cristina, Ferrer, Manel, Forns, Pilar, Gómez, Elena, González, Jacob, Lozoya, Estrella, Mir, Marta, Moreno, Imma, Petit, Silvia, Roberts, Richard S., Sevilla, Sara, Vidal, Bernat, Vidal, Laura, Vilaseca, Pere

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2‑(Fluoromethoxy)-4′‑(S‑methanesulfonimidoyl)-1,1′-biphenyl (UCM-1306), an Orally Bioavailable Positive Allosteric Modulator of the Human Dopamine D1 Receptor for Parkinson’s Disea... von García-Cárceles, Javier, Vázquez-Villa, Henar, Brea, José, Ladron de Guevara-Miranda, David, Cincilla, Giovanni, Sánchez-Martínez, Melchor, Sánchez-Merino, Anabel, Algar, Sergio, Teresa de los Frailes, María, Roberts, Richard S., Ballesteros, Juan A., Rodríguez de Fonseca, Fernando, Benhamú, Bellinda, Loza, María I., López-Rodríguez, María L.

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4‑Amino-7,8-dihydro-1,6-naphthyridin-5(6H)‑ones as Inhaled Phosphodiesterase Type 4 (PDE4) Inhibitors: Structural Biology and Structure–Activity Relationships von Roberts, Richard S, Sevilla, Sara, Ferrer, Manel, Taltavull, Joan, Hernández, Begoña, Segarra, Victor, Gràcia, Jordi, Lehner, Martin D, Gavaldà, Amadeu, Andrés, Miriam, Cabedo, Judit, Vilella, Dolors, Eichhorn, Peter, Calama, Elena, Carcasona, Carla, Miralpeix, Montserrat

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Impurity Annihilation:  Chromatography-Free Parallel Mitsunobu Reactions von Barrett, Anthony G. M, Roberts, Richard S, Schröder, Jürgen

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Biphenyl Pyridazinone Derivatives as Inhaled PDE4 Inhibitors: Structural Biology and Structure–Activity Relationships von Gràcia, Jordi, Buil, Maria Antonia, Castro, Jordi, Eichhorn, Peter, Ferrer, Manel, Gavaldà, Amadeu, Hernández, Begoña, Segarra, Victor, Lehner, Martin D, Moreno, Imma, Pagès, Lluís, Roberts, Richard S, Serrat, Jordi, Sevilla, Sara, Taltavull, Joan, Andrés, Miriam, Cabedo, Judit, Vilella, Dolors, Calama, Elena, Carcasona, Carla, Miralpeix, Montserrat

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Structure–activity relationships (SAR) and structure–kinetic relationships (SKR) of pyrrolopiperidinone acetic acids as CRTh2 antagonists von Andrés, Miriam, Buil, Maria Antonia, Calbet, Marta, Casado, Oscar, Castro, Jordi, Eastwood, Paul R., Eichhorn, Peter, Ferrer, Manel, Forns, Pilar, Moreno, Imma, Petit, Silvia, Roberts, Richard S.

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Structure-activity relationships (SAR) and structure-kinetic relationships (SKR) of sulphone-based CRTh2 antagonists von Buil, Maria Antonia, Calbet, Marta, Castillo, Marcos, Castro, Jordi, Esteve, Cristina, Ferrer, Manel, Forns, Pilar, González, Jacob, López, Sara, Roberts, Richard S., Sevilla, Sara, Vidal, Bernat, Vidal, Laura, Vilaseca, Pere

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2-(1H-Pyrazol-1-yl)acetic acids as chemoattractant receptor-homologous molecule expressed on Th2 lymphocytes (CRTh2) antagonists von Andrés, Miriam, Bravo, Mónica, Buil, Maria Antonia, Calbet, Marta, Castillo, Marcos, Castro, Jordi, Eichhorn, Peter, Ferrer, Manel, Lehner, Martin D., Moreno, Imma, Roberts, Richard S., Sevilla, Sara

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Structure–activity relationships (SAR) and structure–kinetic relationships (SKR) of bicyclic heteroaromatic acetic acids as potent CRTh2 antagonists I von Alonso, Juan Antonio, Andrés, Miriam, Bravo, Mónica, Buil, Maria Antonia, Calbet, Marta, Castro, Jordi, Eastwood, Paul R., Eichhorn, Peter, Esteve, Cristina, Gómez, Elena, González, Jacob, Mir, Marta, Petit, Silvia, Roberts, Richard S., Vidal, Bernat, Vidal, Laura, Vilaseca, Pere, Zanuy, Miriam

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Structure–activity relationships (SAR) and structure–kinetic relationships (SKR) of bicyclic heteroaromatic acetic acids as potent CRTh2 antagonists II: Lead optimization von Alonso, Juan Antonio, Andrés, Miriam, Bravo, Mónica, Calbet, Marta, Eastwood, Paul R., Eichhorn, Peter, Esteve, Cristina, Ferrer, Manel, Gómez, Elena, González, Jacob, Mir, Marta, Moreno, Imma, Petit, Silvia, Roberts, Richard S., Sevilla, Sara, Vidal, Bernat, Vidal, Laura, Vilaseca, Pere, Zanuy, Miriam

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2-(1H-Pyrazol-4-yl)acetic acids as CRTh2 antagonists von Andrés, Miriam, Bravo, Mónica, Buil, Maria Antonia, Calbet, Marta, Castro, Jordi, Domènech, Teresa, Eichhorn, Peter, Ferrer, Manel, Gómez, Elena, Lehner, Martin D., Moreno, Imma, Roberts, Richard S., Sevilla, Sara

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ROMP-Spheres:  A Novel High-Loading Polymer Support Using Cross Metathesis between Vinyl Polystyrene and Norbornene Derivatives von Barrett, Anthony G. M, Cramp, Susan M, Roberts, Richard S

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Multi-platform next-generation sequencing of the domestic turkey (Meleagris gallopavo): genome assembly and analysis von Dalloul, Rami A, Long, Julie A, Zimin, Aleksey V, Aslam, Luqman, Beal, Kathryn, Blomberg, Le Ann, Bouffard, Pascal, Burt, David W, Crasta, Oswald, Crooijmans, Richard P M A, Cooper, Kristal, Coulombe, Roger A, De, Supriyo, Delany, Mary E, Dodgson, Jerry B, Dong, Jennifer J, Evans, Clive, Frederickson, Karin M, Flicek, Paul, Florea, Liliana, Folkerts, Otto, Groenen, Martien A M, Harkins, Tim T, Herrero, Javier, Hoffmann, Steve, Megens, Hendrik-Jan, Jiang, Andrew, de Jong, Pieter, Kaiser, Pete, Kim, Heebal, Kim, Kyu-Won, Kim, Sungwon, Langenberger, David, Lee, Mi-Kyung, Lee, Taeheon, Mane, Shrinivasrao, Marcais, Guillaume, Marz, Manja, McElroy, Audrey P, Modise, Thero, Nefedov, Mikhail, Notredame, Cédric, Paton, Ian R, Payne, William S, Pertea, Geo, Prickett, Dennis, Puiu, Daniela, Qioa, Dan, Raineri, Emanuele, Ruffier, Magali, Salzberg, Steven L, Schatz, Michael C, Scheuring, Chantel, Schmidt, Carl J, Schroeder, Steven, Searle, Stephen M J, Smith, Edward J, Smith, Jacqueline, Sonstegard, Tad S, Stadler, Peter F, Tafer, Hakim, Tu, Zhijian Jake, Van Tassell, Curtis P, Vilella, Albert J, Williams, Kelly P, Yorke, James A, Zhang, Liqing, Zhang, Hong-Bin, Zhang, Xiaojun, Zhang, Yang, Reed, Kent M

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Lineage-specific biology revealed by a finished genome assembly of the mouse von Church, Deanna M, Goodstadt, Leo, Hillier, Ladeana W, Zody, Michael C, Goldstein, Steve, She, Xinwe, Bult, Carol J, Agarwala, Richa, Cherry, Joshua L, DiCuccio, Michael, Hlavina, Wratko, Kapustin, Yuri, Meric, Peter, Maglott, Donna, Birtle, Zoë, Marques, Ana C, Graves, Tina, Zhou, Shiguo, Teague, Brian, Potamousis, Konstantinos, Churas, Christopher, Place, Michael, Herschleb, Jill, Runnheim, Ron, Forrest, Daniel, Amos-Landgraf, James, Schwartz, David C, Cheng, Ze, Lindblad-Toh, Kerstin, Eichler, Evan E, Ponting, Chris P

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Oxazole Synthesis with Minimal Purification:  Synthesis and Application of a ROMPgel Tosmic Reagent von Barrett, Anthony G. M, Cramp, Susan M, Hennessy, Alan J, Procopiou, Panayiotis A, Roberts, Richard S

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Horner−Emmons Synthesis with Minimal Purification Using ROMPGEL:  A Novel High-Loading Matrix for Supported Reagents von Barrett, Anthony G. M, Cramp, Susan M, Roberts, Richard S, Zecri, Frederic J

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A ROMPGEL-Supported N-Hydroxysuccinimide:  A Host of Acylations with Minimal Purification von Barrett, Anthony G. M, Cramp, Susan M, Roberts, Richard S, Zecri, Frederic J

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Enhanced transformation efficiency in Treponema denticola enabled by SyngenicDNA-based plasmids lacking restriction-modification target motifs von Johnston, Christopher D, Goetting-Minesky, M Paula, Kennedy, Kelly, Godovikova, Valentina, Zayed, Sara M, Roberts, Richard J, Fenno, J Christopher

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A modular synthesis of novel 4-amino-7,8-dihydro-1,6-naphthyridin-5(6H)-ones as PDE4 inhibitors von Ferrer, Manel, Roberts, Richard S., Sevilla, Sara

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