On-demand male contraception via acute inhibition of soluble adenylyl cyclase von Balbach, Melanie, Rossetti, Thomas, Ferreira, Jacob, Ghanem, Lubna, Ritagliati, Carla, Myers, Robert W., Huggins, David J., Steegborn, Clemens, Miranda, Ileana C., Meinke, Peter T., Buck, Jochen, Levin, Lonny R.

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Development of an improved inhibitor of Lats kinases to promote regeneration of mammalian organs von Kastan, Nathaniel R., Oak, Sanyukta, Liang, Rui, Baxt, Leigh, Myers, Robert W., Ginn, John, Liverton, Nigel, Huggins, David J., Pichardo, John, Paul, Matthew, Carroll, Thomas S., Nagiel, Aaron, Gnedeva, Ksenia, Hudspeth, A. J.

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Acceptability, Feasibility, and Effectiveness of Internet-Based Cognitive-Behavioral Therapy for Obsessive-Compulsive Disorder in New York von Patel, Sapana R., Wheaton, Michael G., Andersson, Erik, Rück, Christian, Schmidt, Andrew B., La Lima, Christopher N., Galfavy, Hanga, Pascucci, Olivia, Myers, Robert W., Dixon, Lisa B., Simpson, Helen Blair

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Pharmacological AMPK activation induces transcriptional responses congruent to exercise in skeletal and cardiac muscle, adipose tissues and liver von Muise, Eric S, Guan, Hong-Ping, Liu, Jinqi, Nawrocki, Andrea R, Yang, Xiaodong, Wang, Chuanlin, Rodríguez, Carlos G, Zhou, Dan, Gorski, Judith N, Kurtz, Marc M, Feng, Danqing, Leavitt, Kenneth J, Wei, Lan, Wilkening, Robert R, Apgar, James M, Xu, Shiyao, Lu, Ku, Feng, Wen, Li, Ying, He, Huaibing, Previs, Stephen F, Shen, Xiaolan, van Heek, Margaret, Souza, Sandra C, Rosenbach, Mark J, Biftu, Tesfaye, Erion, Mark D, Kelley, David E, Kemp, Daniel M, Myers, Robert W, Sebhat, Iyassu K

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Assessing potency and binding kinetics of soluble adenylyl cyclase (sAC) inhibitors to maximize therapeutic potential von Rossetti, Thomas, Ferreira, Jacob, Ghanem, Lubna, Buck, Hannes, Steegborn, Clemens, Myers, Robert W, Meinke, Peter T, Levin, Lonny R, Buck, Jochen

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Antidiabetic and antisteatotic effects of the selective fatty acid synthase (FAS) inhibitor platensimycin in mouse models of diabetes von Wu, Margaret, Singh, Sheo B, Wang, Jun, Chung, Christine C, Salituro, Gino, Karanam, Bindhu V, Lee, Sang Ho, Powles, Maryann, Ellsworth, Kenneth P, Lassman, Michael E, Miller, Corey, Myers, Robert W, Tota, Michael R, Zhang, Bei B, Li, Cai

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GPR40 partial agonist MK-2305 lower fasting glucose in the Goto Kakizaki rat via suppression of endogenous glucose production von Miller, Corin, Pachanski, Michele J, Kirkland, Melissa E, Kosinski, Daniel T, Mane, Joel, Bunzel, Michelle, Cao, Jin, Souza, Sarah, Thomas-Fowlkes, Brande, Di Salvo, Jerry, Weinglass, Adam B, Li, Xiaoyan, Myers, Robert W, Knagge, Kevin, Carrington, Paul E, Hagmann, William K, Trujillo, Maria E

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Corrigendum: Assessing potency and binding kinetics of soluble adenylyl cyclase (sAC) inhibitors to maximize therapeutic potential von Rossetti, Thomas, Ferreira, Jacob, Ghanem, Lubna, Buck, Hannes, Steegborn, Clemens, Myers, Robert W, Meinke, Peter T, Levin, Lonny R, Buck, Jochen

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Discovery of MK-8722: A Systemic, Direct Pan-Activator of AMP-Activated Protein Kinase von Feng, Danqing, Biftu, Tesfaye, Romero, F. Anthony, Kekec, Ahmet, Dropinski, James, Kassick, Andrew, Xu, Shiyao, Kurtz, Marc M, Gollapudi, Anantha, Shao, Qing, Yang, Xiaodong, Lu, Ku, Zhou, Gaochao, Kemp, Daniel, Myers, Robert W, Guan, Hong-Ping, Trujillo, Maria E, Li, Cai, Weber, Ann, Sebhat, Iyassu K

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Apicidin: A Novel Antiprotozoal Agent that Inhibits Parasite Histone Deacetylase von Darkin-Rattray, Sandra J., Gurnett, Anne M., Myers, Robert W., Dulski, Paula M., Crumley, Tami M., Allocco, John J., Cannova, Christine, Meinke, Peter T., Colletti, Steven L., Bednarek, Maria A., Singh, Sheo B., Goetz, Michael A., Dombrowski, Anne W., Polishook, Jon D., Schmatz, Dennis M.

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Systemic pan-AMPK activator MK-8722 improves glucose homeostasis but induces cardiac hypertrophy von Myers, Robert W., Guan, Hong-Ping, Ehrhart, Juliann, Petrov, Aleksandr, Prahalada, Srinivasa, Tozzo, Effie, Yang, Xiaodong, Kurtz, Marc M., Trujillo, Maria, Trotter, Dinko Gonzalez, Feng, Danqing, Xu, Shiyao, Eiermann, George, Holahan, Marie A., Rubins, Daniel, Conarello, Stacey, Niu, Xiaoda, Souza, Sandra C., Miller, Corin, Liu, Jinqi, Lu, Ku, Feng, Wen, Li, Ying, Painter, Ronald E., Milligan, James A., He, Huaibing, Liu, Franklin, Ogawa, Aimie, Wisniewski, Douglas, Rohm, Rory J., Wang, Liyang, Bunzel, Michelle, Qian, Ying, Zhu, Wei, Wang, Hongwu, Bennet, Bindu, Scheuch, Lisa LaFranco, Fernandez, Guillermo E., Li, Cai, Klimas, Michael, Zhou, Gaochao, van Heek, Margaret, Biftu, Tesfaye, Weber, Ann, Kelley, David E., Thornberry, Nancy, Erion, Mark D., Kemp, Daniel M., Sebhat, Iyassu K.

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Defining and Addressing Gaps in Care for Obsessive-Compulsive Disorder in the United States von Senter, Meredith S, Patel, Sapana R, Dixon, Lisa B, Myers, Robert W, Simpson, H. Blair

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Retrospective State Medicaid Claims Analysis of Children and Adults With Obsessive-Compulsive Disorder von Patel, Sapana R, Messner, Gabrielle R, Radigan, Marleen, Sang, Yi, Wang, Rui, Gu, Gyojeong, Myers, Robert W, Dixon, Lisa B, Simpson, H Blair

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Design, Synthesis, and Pharmacological Evaluation of Second-Generation Soluble Adenylyl Cyclase (sAC, ADCY10) Inhibitors with Slow Dissociation Rates von Miller, Michael, Rossetti, Thomas, Ferreira, Jacob, Ghanem, Lubna, Balbach, Melanie, Kaur, Navpreet, Levin, Lonny R., Buck, Jochen, Kehr, Maria, Coquille, Sandrine, van den Heuvel, Joop, Steegborn, Clemens, Fushimi, Makoto, Finkin-Groner, Efrat, Myers, Robert W., Kargman, Stacia, Liverton, Nigel J., Huggins, David J., Meinke, Peter T.

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Scaffold Hopping and Optimization of Small Molecule Soluble Adenyl Cyclase Inhibitors Led by Free Energy Perturbation von Sun, Shan, Fushimi, Makoto, Rossetti, Thomas, Kaur, Navpreet, Ferreira, Jacob, Miller, Michael, Quast, Jonathan, van den Heuvel, Joop, Steegborn, Clemens, Levin, Lonny R., Buck, Jochen, Myers, Robert W., Kargman, Stacia, Liverton, Nigel, Meinke, Peter T., Huggins, David J.

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Addition to “Scaffold Hopping and Optimization of Small Molecule Soluble Adenyl Cyclase Inhibitors Led by Free Energy Perturbation” von Sun, Shan, Fushimi, Makoto, Rossetti, Thomas, Kaur, Navpreet, Ferreira, Jacob, Miller, Michael, Quast, Jonathan, van den Heuvel, Joop, Steegborn, Clemens, Levin, Lonny R., Buck, Jochen, Myers, Robert W., Kargman, Stacia, Liverton, Nigel, Meinke, Peter T., Huggins, David J.

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Small-molecule inhibition of SARS-CoV-2 NSP14 RNA cap methyltransferase von Meyer, Cindy, Garzia, Aitor, Miller, Michael W, Huggins, David J, Myers, Robert W, Hoffmann, Hans-Heinrich, Ashbrook, Alison W, Jannath, Syeda Y, Liverton, Nigel, Kargman, Stacia, Zimmerman, Matthew, Nelson, Andrew M, Sharma, Vijeta, Dolgov, Enriko, Cangialosi, Julianna, Penalva-Lopez, Suyapa, Alvarez, Nadine, Chang, Ching-Wen, Oswal, Neelam, Gonzalez, Irene, Rasheed, Risha, Goldgirsh, Kira, Davis, Jada A, Ramos-Espiritu, Lavoisier, Menezes, Miriam-Rose, Larson, Chloe, Nitsche, Julius, Ganichkin, Oleg, Alwaseem, Hanan, Molina, Henrik, Steinbacher, Stefan, Glickman, J Fraser, Perlin, David S, Rice, Charles M, Meinke, Peter T, Tuschl, Thomas

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Using a Function-First “Scout Fragment”-Based Approach to Develop Allosteric Covalent Inhibitors of Conformationally Dynamic Helicase Mechanoenzymes von Ramsey, Jared R., Shelton, Patrick M. M., Heiss, Tyler K., Olinares, Paul Dominic B., Vostal, Lauren E., Soileau, Heather, Grasso, Michael, Casebeer, Sara W., Adaniya, Stephanie, Miller, Michael, Sun, Shan, Huggins, David J., Myers, Robert W., Chait, Brian T., Vinogradova, Ekaterina V., Kapoor, Tarun M.

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Discovery of ethyl ketone-based HDACs 1, 2, and 3 selective inhibitors for HIV latency reactivation von Yu, Wensheng, Liu, Jian, Yu, Younong, Zhang, Vivian, Clausen, Dane, Kelly, Joseph, Wolkenberg, Scott, Beshore, Douglas, Duffy, Joseph L., Chung, Christine C., Myers, Robert W., Klein, Daniel J., Fells, James, Holloway, Kate, Wu, Jin, Wu, Guoxin, Howell, Bonnie J., Barnard, Richard J.O., Kozlowski, Joseph

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Statewide Workforce Development Program to Improve Care for Individuals With Obsessive-Compulsive Disorder von Patel, Sapana R, Gershkovich, Marina, Hinds, Melissa, Jankowski, Samantha E, Dixon, Lisa B, Myers, Robert W, Simpson, H. Blair

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