Current status of the research and development of diacylglycerol O-acyltransferase 1 (DGAT1) inhibitors von DeVita, Robert J, Pinto, Shirly

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Current Status of the Research and Development of Diacylglycerol O‑Acyltransferase 1 (DGAT1) Inhibitors: Miniperspective von DeVita, Robert J, Pinto, Shirly

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Monoubiquitination empowers ubiquitin chain elongation von Wu, Kenneth, DeVita, Robert J., Pan, Zhen-Qiang

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Modulation of Cullin-RING E3 ubiquitin ligase-dependent ubiquitination by small molecule compounds von Wu, Kenneth, DeVita, Robert J., Pan, Zhen-Qiang

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DYRK1A Inhibitors as Potential Therapeutics for β‑Cell Regeneration for Diabetes von Kumar, Kunal, Suebsuwong, Chalada, Wang, Peng, Garcia-Ocana, Adolfo, Stewart, Andrew F, DeVita, Robert J

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Development of Kinase-Selective, Harmine-Based DYRK1A Inhibitors that Induce Pancreatic Human β‑Cell Proliferation von Kumar, Kunal, Wang, Peng, Sanchez, Roberto, Swartz, Ethan A, Stewart, Andrew F, DeVita, Robert J

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Small-molecule activation of SERCA2a SUMOylation for the treatment of heart failure von Kho, Changwon, Lee, Ahyoung, Jeong, Dongtak, Oh, Jae Gyun, Gorski, Przemek A., Fish, Kenneth, Sanchez, Roberto, DeVita, Robert J., Christensen, Geir, Dahl, Russell, Hajjar, Roger J.

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IUPAC-Richter Prize Call for Nominations von Fischer, János, Ali, Amjad, DeVita, Robert J

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Food colorants metabolized by commensal bacteria promote colitis in mice with dysregulated expression of interleukin-23 von He, Zhengxiang, Chen, Lili, Catalan-Dibene, Jovani, Bongers, Gerold, Faith, Jeremiah J., Suebsuwong, Chalada, DeVita, Robert J., Shen, Zeli, Fox, James G., Lafaille, Juan J., Furtado, Glaucia C., Lira, Sergio A.

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Small Molecule Inhibition of Ligand-Stimulated RAGE-DIAPH1 Signal Transduction von Manigrasso, Michaele B., Pan, Jinhong, Rai, Vivek, Zhang, Jinghua, Reverdatto, Sergey, Quadri, Nosirudeen, DeVita, Robert J., Ramasamy, Ravichandran, Shekhtman, Alexander, Schmidt, Ann Marie

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Synthesis and Biological Validation of a Harmine-Based, Central Nervous System (CNS)-Avoidant, Selective, Human β‑Cell Regenerative Dual-Specificity Tyrosine Phosphorylation-Regula... von Kumar, Kunal, Wang, Peng, Wilson, Jessica, Zlatanic, Viktor, Berrouet, Cecilia, Khamrui, Susmita, Secor, Cody, Swartz, Ethan A, Lazarus, Michael, Sanchez, Roberto, Stewart, Andrew F, Garcia-Ocana, Adolfo, DeVita, Robert J

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Acyl-CoA dehydrogenase substrate promiscuity: Challenges and opportunities for development of substrate reduction therapy in disorders of valine and isoleucine metabolism von Houten, Sander M, Dodatko, Tetyana, Dwyer, William, Violante, Sara, Chen, Hongjie, Stauffer, Brandon, DeVita, Robert J, Vaz, Frédéric M, Cross, Justin R, Yu, Chunli, Leandro, João

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CRL4b Inhibition Ameliorates Experimental Autoimmune Encephalomyelitis Progression von Dar, Asif A, Ortega, Yohaniz, Aktas, Sera, Wu, Kenneth, Guha, Ipsita, Porter, Nadia, Rosen, Siera, DeVita, Robert J, Pan, Zhen-Qiang, Oliver, Paula M

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Human Beta Cell Regenerative Drug Therapy for Diabetes: Past Achievements and Future Challenges von Wang, Peng, Karakose, Esra, Choleva, Lauryn, Kumar, Kunal, DeVita, Robert J, Garcia-Ocaña, Adolfo, Stewart, Andrew F

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349-OR: Selected DYRK1A Inhibitors Simultaneously Drive Both Human Beta-Cell Proliferation and Differentiation von WANG, PENG, KUMAR, KUNAL, LIU, HONGTAO, WOOD, OLIVIA, KARAKOSE, ESRA, CHOLEVA, LAURYN, LAMBERTINI, LUCA, GARCIA-OCANA, ADOLFO, DEVITA, ROBERT J., STEWART, ANDREW F.

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Encounter and React: Computer-Guided Design of Covalent Inhibitors von Ung, Peter Man-Un, DeVita, Robert J., Schlessinger, Avner

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DHTKD1 and OGDH display substrate overlap in cultured cells and form a hybrid 2-oxo acid dehydrogenase complex in vivo von Leandro, João, Dodatko, Tetyana, Aten, Jan, Nemeria, Natalia S, Zhang, Xu, Jordan, Frank, Hendrickson, Ronald C, Sanchez, Roberto, Yu, Chunli, DeVita, Robert J, Houten, Sander M

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Novel selective thiadiazine DYRK1A inhibitor lead scaffold with human pancreatic β-cell proliferation activity von Kumar, Kunal, Man-Un Ung, Peter, Wang, Peng, Wang, Hui, Li, Hailing, Andrews, Mary K., Stewart, Andrew F., Schlessinger, Avner, DeVita, Robert J.

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Deletion of 2‐aminoadipic semialdehyde synthase limits metabolite accumulation in cell and mouse models for glutaric aciduria type 1 von Leandro, João, Dodatko, Tetyana, DeVita, Robert J., Chen, Hongjie, Stauffer, Brandon, Yu, Chunli, Houten, Sander M.

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Structure-Activity Relationships and Biological Evaluation of 7-Substituted Harmine Analogs for Human β-Cell Proliferation von Kumar, Kunal, Wang, Peng, A Swartz, Ethan, Khamrui, Susmita, Secor, Cody, B Lazarus, Michael, Sanchez, Roberto, F Stewart, Andrew, DeVita, Robert J

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