Long‐term monitoring shows hepatitis B virus resistance to entecavir in nucleoside‐naïve patients is rare through 5 years of therapy von Tenney, Daniel J., Rose, Ronald E., Baldick, Carl J., Pokornowski, Kevin A., Eggers, Betsy J., Fang, Jie, Wichroski, Michael J., Xu, Dong, Yang, Joanna, Wilber, Richard B., Colonno, Richard J.

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Preclinical Profile and Characterization of the Hepatitis C Virus NS3 Protease Inhibitor Asunaprevir (BMS-650032) von MCPHEE, Fiona, SHEAFFER, Amy K, CHAOQUN CHEN, LEE, Min S, MOSURE, Kathy, SUN, Li-Qiang, SINZ, Michael, MEANWELL, Nicholas A, COLONNO, Richard J, KNIPE, Jay, SCOLA, Paul, FRIBORG, Jacques, HERNANDEZ, Dennis, FALK, Paul, GUANGZHI ZHAI, LEVINE, Steven, CHANIEWSKI, Susan, FEI YU, BARRY, Diana

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Protection of macaques from vaginal SHIV challenge by vaginally delivered inhibitors of virus-cell fusion von Moore, John P, Klasse, Per Johan, Schader, Susan M, Marx, Preston A, Dufour, Jason, Colonno, Richard J, Ketas, Thomas J, Hu, Qinxue, Lu, Min, Shattock, Robin J, Springer, Martin S, Veazey, Ronald S

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Two-Year Assessment of Entecavir Resistance in Lamivudine-Refractory Hepatitis B Virus Patients Reveals Different Clinical Outcomes Depending on the Resistance Substitutions Presen... von TENNEY, Daniel J, ROSE, Ronald E, EGGERS, Betsy, HSU, Mayla, MARY JANE PLYM, POUNDSTONE, Patricia, YANG, Joanna, COLONNO, Richard J, BALDICK, Carl J, LEVINE, Steven M, POKORNOWSKI, Kevin A, WALSH, Ann W, JIE FANG, YU, Cheng-Fang, SHARON ZHANG, MAZZUCCO, Charles E

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A Dose-Ranging Study of the Efficacy and Tolerability of Entecavir in Lamivudine-Refractory Chronic Hepatitis B Patients von Chang, Ting–Tsung, Gish, Robert G., Hadziyannis, Stephanos J., Cianciara, Janusz, Rizzetto, Mario, Schiff, Eugene R., Pastore, Giuseppe, Bacon, Bruce R., Poynard, Thierry, Joshi, Shobha, Klesczewski, Kenneth S., Thiry, Alexandra, Rose, Ronald E., Colonno, Richard J., Hindes, Robert G.

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Inhibition of Hepatitis B Virus Polymerase by Entecavir von LANGLEY, David R, WALSH, Ann W, BALDICK, Carl J, EGGERS, Betsy J, ROSE, Ronald E, LEVINE, Steven M, JAYNE KAPUR, A, COLONNO, Richard J, TENNEY, Daniel J

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Mechanistic characterization and molecular modeling of hepatitis B virus polymerase resistance to entecavir von Walsh, Ann W, Langley, David R, Colonno, Richard J, Tenney, Daniel J

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Entecavir for Treatment of Hepatitis B Virus Displays No In Vitro Mitochondrial Toxicity or DNA Polymerase Gamma Inhibition von MAZZUCCO, Charles E, HAMATAKE, Robert K, COLONNO, Richard J, TENNEY, Daniel J

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Activities of Atazanavir (BMS-232632) against a Large Panel of Human Immunodeficiency Virus Type 1 Clinical Isolates Resistant to One or More Approved Protease Inhibitors von COLONNO, Richard J, THIRY, Alexandra, LIMOLI, Kay, PARKIN, Neil

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Long-Term Entecavir Treatment Results in Sustained Antiviral Efficacy and Prolonged Life Span in the Woodchuck Model of Chronic Hepatitis Infection von Colonno, Richard J., Genovesi, Eugene V., Medina, Ivette, Lamb, Lucinda, Durham, Stephen K., Huang, Meei-Li, Corey, Lawrence, Littlejohn, Margaret, Locarnini, Steven, Tennant, Bud C., Rose, Burt, Clark, Junius M.

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Hepatitis B virus quasispecies susceptibility to entecavir confirms the relationship between genotypic resistance and patient virologic response von Baldick, Carl J, Eggers, Betsy J, Fang, Jie, Levine, Steven M, Pokornowski, Kevin A, Rose, Ronald E, Yu, Cheng-Fang, Tenney, Daniel J, Colonno, Richard J

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Biochemical and Genetic Characterizations of a Novel Human Immunodeficiency Virus Type 1 Inhibitor That Blocks gp120-CD4 Interactions von Guo, Qi, Ho, Hsu-Tso, Dicker, Ira, Fan, Li, Zhou, Nannan, Friborg, Jacques, Wang, Tao, McAuliffe, Brian V, Wang, Hwei-Gene Heidi, Rose, Ronald E, Fang, Hua, Scarnati, Helen T, Langley, David R, Meanwell, Nicholas A, Abraham, Ralph, Colonno, Richard J, Lin, Pin-Fang

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Chemical genetics strategy identifies an HCV NS5A inhibitor with a potent clinical effect von Meanwell, Nicholas A, Gao, Min, Nettles, Richard E, Belema, Makonen, Snyder, Lawrence B, Nguyen, Van N, Fridell, Robert A, Serrano-Wu, Michael H, Langley, David R, Sun, Jin-Hua, O’Boyle II, Donald R, Lemm, Julie A, Wang, Chunfu, Knipe, Jay O, Chien, Caly, Colonno, Richard J, Grasela, Dennis M, Hamann, Lawrence G

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In Vitro Inhibition of Hepadnavirus Polymerases by the Triphosphates of BMS-200475 and Lobucavir von SEIFER, M, HAMATAKE, R. K, COLONNO, R. J, STANDRING, D. N

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BMS-232632, a Highly Potent Human Immunodeficiency Virus Protease Inhibitor That Can Be Used in Combination with Other Available Antiretroviral Agents von ROBINSON, B. S, RICCARDI, K. A, LIN, P.-F, GONG, Y.-F, QI GUO, STOCK, D. A, BLAIR, W. S, TERRY, B. J, DEMINIE, C. A, DJANG, F, COLONNO, R. J

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Inhibitors of HIV-1 attachment. Part 2: An initial survey of indole substitution patterns von MEANWELL, Nicholas A, WALLACE, Owen B, YEUNG, Kap-Sun, ZHILEI QIU, WRIGHT, J. J. Kim, ZHENG YANG, ZADJURA, Lisa, TWEEDIE, Donald L, YEOLA, Suresh, FANG ZHAO, RANADIVE, Sunanda, ROBINSON, Brett A, HAIQUAN FANG, GONG, Yi-Fei, WANG, Hwei-Gene Heidi, BLAIR, Wade S, SHI, Pei-Yong, COLONNO, Richard J, LIN, Pin-Fang, WANG, Henry, DESHPANDE, Milind, TAO WANG, ZHIWEI YIN, ZHONGXING ZHANG, PEARCE, Bradley C, JAMES, Jennifer

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Discovery of the Human Immunodeficiency Virus Type 1 (HIV-1) Attachment Inhibitor Temsavir and Its Phosphonooxymethyl Prodrug Fostemsavir von Wang, Tao, Ueda, Yasu, Zhang, Zhongxing, Yin, Zhiwei, Matiskella, John, Pearce, Bradley C, Yang, Zheng, Zheng, Ming, Parker, Dawn D, Yamanaka, Gregory A, Gong, Yi-Fei, Ho, Hsu-Tso, Colonno, Richard J, Langley, David R, Lin, Pin-Fang, Meanwell, Nicholas A, Kadow, John F

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In Vitro Resistance Profile of the Human Immunodeficiency Virus Type 1 Protease Inhibitor BMS-232632 von GONG, Y.-F, ROBINSON, B. S, ROSE, R. E, DEMINIE, C, SPICER, T. P, STOCK, D, COLONNO, R. J, LIN, P.-F

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Entecavir resistance is rare in nucleoside naïve patients with hepatitis B von Colonno, Richard J., Rose, Ronald, Baldick, Carl J., Levine, Steven, Pokornowski, Kevin, Yu, Cheng F., Walsh, Ann, Fang, Jie, Hsu, Mayla, Mazzucco, Charles, Eggers, Betsy, Zhang, Sharon, Plym, Mary, Klesczewski, Kenneth, Tenney, Daniel J.

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Molecular Basis for Increased Susceptibility of Isolates with Atazanavir Resistance-Conferring Substitution I50L to Other Protease Inhibitors von Yanchunas, Jr, Joseph, Langley, David R, Tao, Li, Rose, Ronald E, Friborg, Jacques, Colonno, Richard J, Doyle, Michael L

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