A Practical Stereoselective Synthesis and Novel Cocrystallizations of an Amphiphatic SGLT-2 Inhibitor von Deshpande, Prashant P, Singh, Janak, Pullockaran, Annie, Kissick, Thomas, Ellsworth, Bruce A, Gougoutas, Jack Z, Dimarco, John, Fakes, Michael, Reyes, Mayra, Lai, Chiajen, Lobinger, Hidegard, Denzel, Theo, Ermann, Peter, Crispino, Gerard, Randazzo, Michael, Gao, Zenrong, Randazzo, Renee, Lindrud, Mark, Rosso, Victor, Buono, Frederic, Doubleday, Wendel W, Leung, Simon, Richberg, Pricilla, Hughes, David, Washburn, William N, Meng, Wei, Volk, Kevin J, Mueller, Richard H

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Insights Into Palladium-Catalyzed Cyanation of Bromobenzene: Additive Effects on the Rate-Limiting Step von Buono, Frederic G, Chidambaram, Rama, Mueller, Richard H, Waltermire, Robert E

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Process Research and Development for an Efficient Synthesis of the HIV Protease Inhibitor BMS-232632 von Xu, Zhongmin, Singh, Janak, Schwinden, Mark D, Zheng, Bin, Kissick, Thomas P, Patel, Bharat, Humora, Michael J, Quiroz, Fernando, Dong, Lin, Hsieh, Dau-Ming, Heikes, James E, Pudipeddi, Madhusudhan, Lindrud, Mark D, Srivastava, Sushil K, Kronenthal, David R, Mueller, Richard H

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Efficient Asymmetric Synthesis of the Vasopeptidase Inhibitor BMS-189921 von Singh, Janak, Kronenthal, David R, Schwinden, Mark, Godfrey, Jollie D, Fox, Rita, Vawter, Edward J, Zhang, Bo, Kissick, Thomas P, Patel, Bharat, Mneimne, Omar, Humora, Michael, Papaioannou, Chris G, Szymanski, Walter, Wong, Michael K. Y, Chen, Chien K, Heikes, James E, DiMarco, John D, Qiu, Jun, Deshpande, Rajendra P, Gougoutas, Jack Z, Mueller, Richard H

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Remarkable β-Selectivity in the Synthesis of β-1-C-Arylglucosides:  Stereoselective Reduction of Acetyl-Protected Methyl 1-C-Arylglucosides without Acetoxy-Group Participation von Deshpande, Prashant P, Ellsworth, Bruce A, Buono, Frederic G, Pullockaran, Annie, Singh, Janak, Kissick, Thomas P, Huang, Ming-H, Lobinger, Hildegard, Denzel, Theodor, Mueller, Richard H

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Microbial hydroxylation of o-bromophenylacetic acid: synthesis of 4-substituted-2,3-dihydrobenzofurans von Deshpande, Prashant P, Nanduri, Venkata B, Pullockaran, Annie, Christie, Hamish, Mueller, Richard H, Patel, Ramesh N

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A Practical Asymmetric Synthesis of the Antiviral Agent Lobucavir, BMS-180194 von Singh, Janak, Bisacchi, Gregory S, Ahmad, Saleem, Godfrey, Jollie D, Kissick, Thomas P, Mitt, Toomas, Kocy, Octavian, Vu, Truc, Papaioannou, Chris G, Wong, Michael K, Heikes, James E, Zahler, Robert, Mueller, Richard H

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Conversion of L-pyroglutamic acid to 4-alkyl-substituted L-prolines. The synthesis of trans-4-cyclohexyl-L-proline von Thottathil, John K, Moniot, Jerome L, Mueller, Richard H, Wong, Michael K. Y, Kissick, Thomas P

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Regioselective enzymatic aminoacylation of lobucavir to give an intermediate for lobucavir prodrug von Hanson, Ronald L, Shi, Zhongping, Brzozowski, David B, Banerjee, Amit, Kissick, Thomas P, Singh, Janak, Pullockaran, Annie J, North, Jeffrey T, Fan, Junying, Howell, Jeffrey, Durand, Susan C, Montana, Michael A, Kronenthal, David R, Mueller, Richard H, Patel, Ramesh N

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Cupric bromide mediated oxidation of 4-carboxyoxazolines to the corresponding oxazoles von Barrish, Joel C, Singh, Janak, Spergel, Steven H, Han, Wen Ching, Kissick, Thomas P, Kronenthal, David R, Mueller, Richard H

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Regioselective Activation of Aminothiazole(iminoxyacetic acid)acetic Acid:  An Efficient Synthesis of the Monobactam Aztreonam von Singh, Janak, Denzel, Theodor W, Fox, Rita, Kissick, Thomas P, Herter, Rolf, Wurdinger, Joseph, Schierling, Peter, Papaioannou, Chris G, Moniot, Jerome L, Mueller, Richard H, Cimarusti, Christopher M

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A Practical Synthesis of an Anti-Methicillin Resistant Staphylococcus aureus Cephalosporin BMS-247243 von Singh, Janak, Kim, Oak K, Kissick, Thomas P, Natalie, Kenneth J, Zhang, Bo, Crispino, Gerard A, Springer, Dane M, Wichtowski, John A, Zhang, Yunhui, Goodrich, Jason, Ueda, Yasutsugu, Luh, Bing Y, Burke, Brian D, Brown, Matthew, Dutka, Anthony P, Zheng, Bin, Hsieh, Dau-Ming, Humora, Michael J, North, Jeffrey T, Pullockaran, Anne J, Livshits, Juliya, Swaminathan, Shankar, Gao, Zhinong, Schierling, Peter, Ermann, Peter, Perrone, Robert K, Lai, Mei C, Gougoutas, Jack Z, DiMarco, John D, Bronson, Joanne J, Heikes, James E, Grosso, John A, Kronenthal, David R, Denzel, Theodor W, Mueller, Richard H

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The ester enolate Claisen rearrangement. Stereochemical control through stereoselective enolate formation von Ireland, Robert E, Mueller, Richard H, Willard, Alvin K

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Diastereoselective Reaction of a Grignard Reagent with Chiral Imides:  A Practical Preparation of a Key Intermediate in the Synthesis of Ifetroban Sodium von Mueller, Richard H, Wang, Shaopeng, Pansegrau, Paul D, Jannotti, Joy Q, Poss, Michael A, Thottathil, John K, Singh, Janak, Humora, Michael J, Kissick, Thomas P, Boyhan, Brenda

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Ester enolate Claisen rearrangement. Construction of the prostanoid skeleton von Ireland, Robert E, Mueller, Richard H, Willard, Alvin K

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A Practical Asymmetric Synthesis of the Antiviral Agent Lobucavir, BMS-180194 von Singh, Janak, Bisacchi, Gregory S, Ahmad, Saleem, Godfrey, Jollie D, Kissick, Thomas P, Mitt, Toomas, Kocy, Octavian, Vu, Truc, Papaioannou, Chris G, Wong, Michael K, Heikes, James E, Zahler, Robert, Mueller, Richard H

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Claisen rearrangement of allyl esters von Ireland, Robert E, Mueller, Richard H

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Stereo- and regioselective total synthesis of the hydropyrido[2,1,6-de]quinolizine ladybug defensive alkaloids von Mueller, Richard H, Thompson, Mark E, DiPardo, Robert M

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Improved synthesis of aryl 1,1-dimethylpropargyl ethers von Godfrey, Jollie D., Mueller, Richard H., Sedergran, Thomas C., Soundararajan, Nachimuthu, Colandrea, Vincent J.

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β-Lactam synthesis: Cyclization versus 1,2-acyl migration-cyclization. The mechanism of the 1,2-acyl migration-cyclization von Godfrey, Jollie D, Mueller, Richard H, Von Langen, Derek J

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