Divergent and Regioselective Synthesis of Pyrazolo[1,5‑a]pyridines and Imidazo[1,5‑a]pyridines von Mennie, Katrina M, Reutershan, Michael H, White, Catherine, Adams, Bruce, Becker, Bridget, Deng, James, Katz, Jason D, LaBlue, Elisabeth, Margrey, Kaila, Saurí, Josep

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NMR Data‐Driven Docking of HDM2‐Inhibitor Complexes von Fradera, Xavier, Reutershan, Michael H., Machacek, Michelle R., Trotter, B. Wesley, McCoy, Mark A.

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Discovery of MK-4688: an Efficient Inhibitor of the HDM2–p53 Protein–Protein Interaction von Reutershan, Michael H, Machacek, Michelle R, Altman, Michael D, Bogen, Stephane, Cai, Mingmei, Cammarano, Carolyn, Chen, Dapeng, Christopher, Matthew, Cryan, John, Daublain, Pierre, Fradera, Xavier, Geda, Prasanthi, Goldenblatt, Peter, Hill, Armetta D, Kemper, Raymond A, Kutilek, Victoria, Li, Chaomin, Martinez, Michelle, McCoy, Mark, Nair, Latha, Pan, Weidong, Thompson, Christopher F, Scapin, Giovanna, Shizuka, Manami, Spatz, Marianne L, Steinhuebel, Dietrich, Sun, Binyuan, Voss, Matthew E, Wang, Xiao, Yang, Liping, Yeh, Tammie C, Dussault, Isabelle, Marshall, C. Gary, Trotter, B. Wesley

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Development of a Flexible and Robust Synthesis of Tetrahydrofuro[3,4‑b]furan Nucleoside Analogues von Candito, David A, Ye, Yingchun, Quiroz, Ryan V, Reutershan, Michael H, Witter, David, Gadamsetty, Surendra B, Li, Hongming, Saurí, Josep, Schneider, Sebastian E, Lam, Yu-hong, Palte, Rachel L

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The Discovery of Two Novel Classes of 5,5-Bicyclic Nucleoside-Derived PRMT5 Inhibitors for the Treatment of Cancer von Quiroz, Ryan V, Reutershan, Michael H, Schneider, Sebastian E, Sloman, David, Lacey, Brian M, Swalm, Brooke M, Yeung, Charles S, Gibeau, Craig, Spellman, Daniel S, Rankic, Danica A, Chen, Dapeng, Witter, David, Linn, Doug, Munsell, Erik, Feng, Guo, Xu, Haiyan, Hughes, Jonathan M. E, Lim, Jongwon, Saurí, Josep, Geddes, Kristin, Wan, Murray, Mansueto, My Sam, Follmer, Nicole E, Fier, Patrick S, Siliphaivanh, Phieng, Daublain, Pierre, Palte, Rachel L, Hayes, Robert P, Lee, Sandra, Kawamura, Shuhei, Silverman, Steven, Sanyal, Sulagna, Henderson, Timothy J, Ye, Yingchun, Gao, Yuanwei, Nicholson, Benjamin, Machacek, Michelle R

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Diminishing GSH-Adduct Formation of Tricyclic Diazepine-based Mutant IDH1 Inhibitors von Huang, Chunhui, Fischer, Christian, Machacek, Michelle R, Bogen, Stephane, Biftu, Tesfaye, Huang, Xianhai, Reutershan, Michael H, Otte, Ryan, Hong, Qingmei, Wu, Zhicai, Yu, Yang, Park, Min, Chen, Lei, Biju, Purakkattle, Knemeyer, Ian, Lu, Ping, Kochansky, Christopher J, Hicks, Michael Brendan, Liu, Yong, Helmy, Roy, Fradera, Xavier, Donofrio, Anthony, Close, Josh, Maddess, Matthew L, White, Catherine, Sloman, David L, Sciammetta, Nunzio, Lu, Jun, Gibeau, Craig, Simov, Vladimir, Zhang, Hongjun, Fuller, Peter, Witter, David

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Deuterium Exchange as an Indicator of Hydrogen Bond Donors and Acceptors von Steffel, Lauren R, Cashman, Timothy J, Reutershan, Michael H, Linton, Brian R

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Purine derivatives as potent γ-secretase modulators von Rivkin, Alexey, Ahearn, Sean P., Chichetti, Stephanie M., Hamblett, Christopher L., Garcia, Yudith, Martinez, Michelle, Hubbs, Jed L., Reutershan, Michael H., Daniels, Matthew H., Siliphaivanh, Phieng, Otte, Karin M., Li, Chaomin, Rosenau, Andrew, Surdi, Laura M., Jung, Joon, Hughes, Bethany L., Crispino, Jamie L., Nikov, George N., Middleton, Richard E., Moxham, Christopher M., Szewczak, Alexander A., Shah, Sanjiv, Moy, Lily Y., Kenific, Candia M., Tanga, Flobert, Cruz, Jonathan C., Andrade, Paula, Angagaw, Minilik H., Shomer, Nirah H., Miller, Thomas, Munoz, Benito, Shearman, Mark S.

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Allosteric Modulation of Protein Arginine Methyltransferase 5 (PRMT5) von Palte, Rachel L, Schneider, Sebastian E, Altman, Michael D, Hayes, Robert P, Kawamura, Shuhei, Lacey, Brian M, Mansueto, My Sam, Reutershan, Michael, Siliphaivanh, Phieng, Sondey, Christopher, Xu, Haiyan, Xu, Zangwei, Ye, Yingchun, Machacek, Michelle R

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Discovery of 1‑[3-(1-Methyl‑1H‑pyrazol-4-yl)-5-oxo‑5H‑benzo[4,5]cyclohepta[1,2‑b]pyridin-7-yl]‑N‑(pyridin-2-ylmethyl)methanesulfonamide (MK-8033): A Specific c‑Met/Ron Dual Kinase... von Northrup, Alan B, Katcher, Matthew H, Altman, Michael D, Chenard, Melissa, Daniels, Matthew H, Deshmukh, Sujal V, Falcone, Danielle, Guerin, David J, Hatch, Harold, Li, Chaomin, Lu, Wei, Lutterbach, Bart, Allison, Timothy J, Patel, Sangita B, Reilly, John F, Reutershan, Michael, Rickert, Keith W, Rosenstein, Craig, Soisson, Stephen M, Szewczak, Alexander A, Walker, Deborah, Wilson, Kevin, Young, Jonathan R, Pan, Bo-Sheng, Dinsmore, Christopher J

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Asymmetric Michael addition of α-nitro-ketones using catalytic peptides von Linton, Brian R., Reutershan, Michael H., Aderman, Christopher M., Richardson, Elizabeth A., Brownell, Kristen R., Ashley, Charles W., Evans, Catherine A., Miller, Scott J.

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PRMT5 inhibitors von Reutershan, Michael H, Lim, Jongwon, Machacek, Michelle, Schneider, Sebastian

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PRMT5 INHIBITORS von LIM, Jongwon, REUTERSHAN, Michael, H, MACHACEK, Michelle, SCHNEIDER, Sebastian

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Purine derivatives as potent g-secretase modulators von Rivkin, Alexey, Ahearn, Sean P, Chichetti, Stephanie M, Hamblett, Christopher L, Garcia, Yudith, Martinez, Michelle, Hubbs, Jed L, Reutershan, Michael H, Daniels, Matthew H, Siliphaivanh, Phieng, Otte, Karin M, Li, Chaomin, Rosenau, Andrew, Surdi, Laura M, Jung, Joon, Hughes, Bethany L, Crispino, Jamie L, Nikov, George N, Middleton, Richard E, Moxham, Christopher M, Szewczak, Alexander A, Shah, Sanjiv, Moy, Lily Y, Kenific, Candia M, Tanga, Flobert, Cruz, Jonathan C, Andrade, Paula, Angagaw, Minilik H, Shomer, Nirah H, Miller, Thomas, Munoz, Benito, Shearman, Mark S

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Prmt5 inhibitors von Sloman, David, Machacek, Michelle, Reutershan, Michael, Gibeau, Craig, Huang, Chunhui, Witter, David, Altman, Michael

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PRMT5 INHIBITORS von WITTER, David J, HUANG, Chunhui, REUTERSHAN, Michael H, MACHACEK, Michelle, GIBEAU, Craig R, SLOMAN, David L, ALTMAN, Michael D

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PRMT5 INHIBITORS von LIM, Jongwon, REUTERSHAN, Michael, H, MACHACEK, Michelle, SCHNEIDER, Sebastian

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PRMT5 inhibitors von Reutershan, Michael H, Machacek, Michelle, Quiroz, Ryan, Schneider, Sebastian, Kawamura, Shuhei, Yeung, Charles S, Siliphaivanh, Phieng, Witter, David, Ye, Yingchun

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PRMT5 INHIBITORS von Reutershan, Michael H, Lim, Jongwon, Machacek, Michelle, Schneider, Sebastian

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PRMT5 INHIBITORS von MACHACEK, Michelle, R, STUPPLE, Paul Anthony, WITTER, David, J, REUTERSHAN, Michael Hale, ALTMAN, Michael, D

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