Tau protein aggregation in Alzheimer's disease: An attractive target for the development of novel therapeutic agents von Jouanne, Marie, Rault, Sylvain, Voisin-Chiret, Anne-Sophie

Volltext

Selective ortho-Bromination of Substituted Benzaldoximes Using Pd-Catalyzed C–H Activation: Application to the Synthesis of Substituted 2-Bromobenzaldehydes von Dubost, Emmanuelle, Fossey, Christine, Cailly, Thomas, Rault, Sylvain, Fabis, Frederic

Volltext

Discovery of Bis-Imidazoline Derivatives as New CXCR4 Ligands von Zhou, Zhicheng, Staropoli, Isabelle, Brelot, Anne, Suzanne, Peggy, Lesnard, Aurélien, Fontaine, Fanny, Perato, Serge, Rault, Sylvain, Helynck, Olivier, Arenzana-Seisdedos, Fernando, Sopkova-de Oliveira Santos, Jana, Lagane, Bernard, Munier-Lehmann, Hélène, Colin, Philippe

Volltext

Recent progress in the synthesis of five-membered heterocycle boronic acids and esters von Primas, Nicolas, Bouillon, Alexandre, Rault, Sylvain

Volltext

Synthesis and Structure–Affinity Relationships of Selective High-Affinity 5‑HT4 Receptor Antagonists: Application to the Design of New Potential Single Photon Emission Computed Tom... von Dubost, Emmanuelle, Dumas, Noé, Fossey, Christine, Magnelli, Rosa, Butt-Gueulle, Sabrina, Ballandonne, Céline, Caignard, Daniel H, Dulin, Fabienne, Sopkova de-Oliveira Santos, Jana, Millet, Philippe, Charnay, Yves, Rault, Sylvain, Cailly, Thomas, Fabis, Frederic

Volltext

Two-Step Synthesis of Substituted 3-Aminoindazoles from 2-Bromobenzonitriles von Lefebvre, Valerie, Cailly, Thomas, Fabis, Frederic, Rault, Sylvain

Volltext

Use of allostery to identify inhibitors of calmodulin-induced activation of Bacillus anthracis edema factor von Laine, Elodie, Goncalves, Christophe, Karst, Johanna C., Lesnard, Aurélien, Rault, Sylvain, Tang, Wei-Jen, Malliavin, Thérèse E., Ladant, Daniel, Blondel, Arnaud, Kuriyan, John

Volltext

Sonogashira cross-coupling reaction in 4-chloro-2-trichloromethylquinazoline series is possible despite a side dimerization reaction von Kieffer, Charline, Verhaeghe, Pierre, Primas, Nicolas, Castera-Ducros, Caroline, Gellis, Armand, Rosas, Roselyne, Rault, Sylvain, Rathelot, Pascal, Vanelle, Patrice

Volltext

Synthesis of 5-arylthiazoles. Comparative study between Suzuki cross-coupling reaction and direct arylation von Primas, Nicolas, Bouillon, Alexandre, Lancelot, Jean-Charles, El-Kashef, Hussein, Rault, Sylvain

Volltext

Synthesis and in vitro antiplasmodial evaluation of 4-anilino-2-trichloromethylquinazolines von VERHAEGHE, Pierre, AZAS, Nadine, VANELLE, Patrice, HUTTER, Sébastien, CASTERA-DUCROS, Caroline, LAGET, Michèle, DUMETRE, Aurélien, GASQUET, Monique, REBOUL, Jean-Pierre, RAULT, Sylvain, RATHELOT, Pascal

Volltext

A general synthesis of halo-oligopyridines. The Garlanding concept von Voisin-Chiret, Anne Sophie, Bouillon, Alexandre, Burzicki, Grégory, Célant, Melanie, Legay, Rémi, El-Kashef, Hussein, Rault, Sylvain

Volltext

Synthesis of novel halopyridinylboronic acids and esters. Part 4: Halopyridin-2-yl-boronic acids and esters are stable, crystalline partners for classical Suzuki cross-coupling von Bouillon, Alexandre, Lancelot, Jean-Charles, Sopkova de Oliveira Santos, Jana, Collot, Valérie, Bovy, Philipppe R, Rault, Sylvain

Volltext

Efficient and simple synthesis of 6-aryl-1,4-dimethyl-9H-carbazoles von Caruso, Anna, Voisin-Chiret, Anne Sophie, Lancelot, Jean-Charles, Sinicropi, Maria Stefania, Garofalo, Antonio, Rault, Sylvain

Volltext

One-pot synthesis of new aza- and diaza-aminophenanthrenes von Rochais, Christophe, Yougnia, Rodrigue, Cailly, Thomas, Sopková-de Oliveira Santos, Jana, Rault, Sylvain, Dallemagne, Patrick

Volltext

Synthesis of 2-TIPS-oxazol-5-ylboronic acid pinacol ester: efficient route to 5-(het)aryloxazoles via Suzuki cross-coupling reaction von Primas, Nicolas, Bouillon, Alexandre, Lancelot, Jean-Charles, Rault, Sylvain

Volltext

A new synthetic route to original sulfonamide derivatives in 2-trichloromethylquinazoline series: a structure-activity relationship study of antiplasmodial activity von Primas, Nicolas, Verhaeghe, Pierre, Cohen, Anita, Kieffer, Charline, Dumètre, Aurélien, Hutter, Sébastien, Rault, Sylvain, Rathelot, Pascal, Azas, Nadine, Vanelle, Patrice

Volltext

Synthesis of novel halopyridinylboronic acids and esters. Part 1: 6-Halopyridin-3-yl-boronic acids and esters von Bouillon, Alexandre, Lancelot, Jean-Charles, Collot, Valérie, Bovy, Philippe R, Rault, Sylvain

Volltext

Reactivity of 3-Iodoimidazo[1,2-a]pyridines Using a Suzuki-Type Cross-Coupling Reaction von Enguehard, Cécile, Renou, Jean-Louis, Collot, Valérie, Hervet, Maud, Rault, Sylvain, Gueiffier, Alain

Volltext

Synthesis of novel halopyridinylboronic acids and esters. Part 2: 2,4, or 5-Halopyridin-3-yl-boronic acids and esters von Bouillon, Alexandre, Lancelot, Jean-Charles, Collot, Valérie, Bovy, Philippe R, Rault, Sylvain

Volltext

An Efficient Two-Step Total Synthesis of the Quaterpyridine Nemertelline von Bouillon, Alexandre, Voisin, Anne Sophie, Robic, Audrey, Lancelot, Jean-Charles, Collot, Valérie, Rault, Sylvain

Volltext