Mechanism-Based Inhibition of Human Steroid 5α-Reductase by Finasteride:  Enzyme-Catalyzed Formation of NADP−Dihydrofinasteride, a Potent Bisubstrate Analog Inhibitor von Bull, Herbert G, Garcia-Calvo, Margarita, Andersson, Stefan, Baginsky, Walter F, Chan, H. Karen, Ellsworth, Dina E, Miller, Randall R, Stearns, Ralph A, Bakshi, Raman K, Rasmusson, Gary H, Tolman, Richard L, Myers, Robert W, Kozarich, John W, Harris, Georgianna S

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4-Aza-3-oxo-5.alpha.-androst-1-ene-17.beta.-N-arylcarboxamides as Dual Inhibitors of Human Type 1 and Type 2 Steroid 5.alpha.-Reductases. Dramatic Effect of N-Aryl Substituents on... von Bakshi, Raman K, Rasmusson, Gary H, Patel, Gool F, Mosley, Ralph T, Chang, Benedict, Ellsworth, Kenneth, Harris, Georgianna S, Tolman, Richard L

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Azasteroids: structure-activity relationships for inhibition of 5.alpha.-reductase and of androgen receptor binding von Rasmusson, Gary H, Reynolds, Glenn F, Steinberg, Nathan G, Walton, Edward, Patel, Gool F, Liang, Tehming, Cascieri, Margaret A, Cheung, Anne H, Brooks, Jerry R, Berman, Charles

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4-Aza-3-oxo-5α-androst-1-ene-17β-N-arylcarboxamides as Dual Inhibitors of Human Type 1 and Type 2 Steroid 5α-Reductases. Dramatic Effect of N-Aryl Substituents on Type 1 and Type 2... von Bakshi, Raman K, Rasmusson, Gary H, Patel, Gool F, Mosley, Ralph T, Chang, Benedict, Ellsworth, Kenneth, Harris, Georgianna S, Tolman, Richard L

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Azasteroids as inhibitors of rat prostatic 5.alpha.-reductase von Rasmusson, Gary H, Reynolds, Glenn F, Utne, Torleif, Jobson, Ronald B, Primka, Raymond L, Berman, Charles, Brooks, Jerry R

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Identification and Selective Inhibition of an Isozyme of Steroid 5α- Reductase in Human Scalp von Harris, Georgianna, Azzolina, Barbara, Baginsky, Walter, Cimis, George, Rasmusson, Gary H., Tolman, Richard L., Christian R. H. Raetz, Ellsworth, Kenneth

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16-SUBSTITUTED-4-AZA-ANDROSTANE 5-ALPHA-REDUCTASE 16-SUBSTITUTED-4-AZA-ANDROSTANE 5-ALPHA-REDUCTASE ISOZYME 1 INHIBITORS ISOZYME 1 INHIBITORS von DURETTE,PHILIPPE, L. DURETTE,PHILIPPE, L, TOLMAN,RICHARD, L. TOLMAN,RICHARD, L, RASMUSSON,GARY H. RASMUSSON,GARY H, HAGMANN,WILLIAM, K. HAGMANN,WILLIAM, K, VON LANGEN,DEREK VON LANGEN,DEREK, LANZA,THOMAS, J., JR. LANZA,THOMAS, J., JR, SAHOO,SOUMYA, P. SAHOO,SOUMYA, P

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4-Aza-3-oxo-5α-androst-1-ene-17β-N-aryl-carboxamides as dual inhibitors of human type 1 and type 2 steroid 5α-reductases. Dramatic effect of N-aryl substituents on type 1 and type... von BAKSHI, R. K, RASMUSSON, G. H, PATEL, G. F, MOSLEY, R. T, CHANG, B, ELLSWORTH, K, HARRIS, G. S, TOLMAN, R. L

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Perhydroindanone Derivatives. I. Applicability of the Diels-Alder Reaction von House, Herbert O, Rasmusson, Gary H

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Stereoselective Synthesis of α-Substituted α,β-Unsaturated Esters von HOUSE, HERBERT O, RASMUSSON, GARY H

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Azasteroids as inhibitors of testosterone 5α-reductase in mammalian skin von MELLIN, T. N, BUSCH, R. D, RASMUSSON, G. H

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Solvolytic rearrangement route to D-homosteroids von Steinberg, Nathan G, Rasmusson, Gary H, Reamer, Robert A

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Photocatalyzed reaction of trifluoromethyl iodide with steroidal dienones von Rasmusson, Gary H, Brown, Ronald D, Arth, Glen E

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Synthesis of 7.alpha.-trifluoromethyltestosterone acetate von Rasmusson, Gary H, Chen, Anna, Arth, Glen E

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Perhydroindanone Derivatives. II. Stability Relationships von House, Herbert O, Rasmusson, Gary H

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A stereoselective synthesis of 7β-phenyl and 7β-methylcholesterol von Bakshi, Raman K., Rasmusson, Gary H.

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4-Methyl-1,2,5,6-tetrahydrobenzo[f]quinolin-3(4H)-one. The Cyclization Product Derived from Methyl 3-[(3,4-Dihydro-2-naphthyl)methyl-amino]propionate von Horii, Zen-Ichi, Iwata, Chuzo, Tamura, Yasumitsu, Nelson, Norman A, Rasmusson, Gary H

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4-AZASTEROIDS AS 5α-REDUCTASE INHIBITORS: IDENTIFICATION OF 4,7β-DIMETHYL-4-AZA-5α-CHOLESTAN-3-ONE (MK-386) AS A SCALP ISOZYME SELECTIVE INHIBITOR von Tolman, Richard L., Aster, Susan, Bakshi, Raman K., Bergman, Jeffrey P., Bull, Herb G., Chang, Benedict, Cimis, George, Dolenga, Michael P., Durette, Phillippe, Ellsworth, Kenneth, Esser, Craig, Graham, Donald W., Hagmann, William K., Harris, Georgianna, Kopka, Ihor, Lanza, Thomas, Patel, Gool, Polo, Scott, Rasmusson, Gary H., Sahoo, Soumya, Toney, Jeffrey H., Von Langen, Derek, Witzel, Bruce

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By-products of the Robinson Annelation Reaction with Cyclohexanone, Cyclopentanone, and Cyclopentane-1,2-dione1 von House, Herbert O, Trost, Barry M, Magin, Ralph W, Carlson, Robert G, Franck, Richard W, Rasmusson, Gary H

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Biochemical and biological studies with 4-aza-steroidal 5α-reductase inhibitors von Liang, Tehming, Rasmusson, Gary H., Brooks, Jerry R.

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