No Denying It: Medicinal Chemistry Training Is in Big Trouble von Rafferty, Michael F

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No Denying It: Medicinal Chemistry Training Is in Big Trouble: Miniperspective von Rafferty, Michael F

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The design and synthesis of human branched-chain amino acid aminotransferase inhibitors for treatment of neurodegenerative diseases von Hu, Lain-Yen, Boxer, Peter A., Kesten, Suzanne R., Lei, Huangshu J., Wustrow, David J., Moreland, David W., Zhang, Liming, Ahn, Kay, Ryder, Todd R., Liu, Xiaohong, Rubin, John R., Fahnoe, Kelly, Carroll, Richard T., Dutta, Satavisha, Fahnoe, Douglass C., Probert, Albert W., Roof, Robin L., Rafferty, Michael F., Kostlan, Catherine R., Scholten, Jeffrey D., Hood, Molly, Ren, Xiao-Dan, Schielke, Gerald P., Su, Ti-Zhi, Taylor, Charles P., Mistry, Anil, McConnell, Patrick, Hasemann, Charles, Ohren, Jeffrey

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New Synthesis of Substituted Benzylamines. Novel Application of the Mitsunobu Reaction To Convert Substituted Benzyl Alcohols to Amines von Nikam, Sham S, Kornberg, Brian E, Rafferty, Michael F

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Synthesis of a Series of 4-Benzyloxyaniline Analogues as Neuronal N-Type Calcium Channel Blockers with Improved Anticonvulsant and Analgesic Properties von Hu, Lain-Yen, Ryder, Todd R, Rafferty, Michael F, Feng, M. Rose, Lotarski, Susan M, Rock, David M, Sinz, Michael, Stoehr, Sally J, Taylor, Charles P, Weber, Mark L, Bowersox, S. Scott, Miljanich, George P, Millerman, Elizabeth, Wang, Yong-Xiang, Szoke, Balazs G

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(S)-4-Methyl-2-(methylamino)pentanoic Acid [4,4-Bis(4-fluorophenyl)butyl]amide Hydrochloride, a Novel Calcium Channel Antagonist, Is Efficacious in Several Animal Models of Pain von Song, Yuntao, Bowersox, S. Scott, Connor, David T, Dooley, David J, Lotarski, Susan M, Malone, Thomas, Miljanich, George, Millerman, Elizabeth, Rafferty, Michael F, Rock, David, Roth, Bruce D, Schmidt, Joann, Stoehr, Sally, Szoke, Balazs G, Taylor, Charles, Vartanian, Mark, Wang, Yong-Xiang

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N-Substituted dibenzoxazepines as analgesic PGE2 antagonists von Hallinan, E. Ann, Hagen, Timothy J, Husa, Robert K, Tsymbalov, Sofya, Rao, Shashidhar N, vanHoeck, Jean Pierre, Rafferty, Michael F, Stapelfeld, Awilda, Savage, Michael A, Reichman, Melvin

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N, N-Dialkyl-dipeptidylamines as novel N-type calcium channel blockers von Hu, Lain-Yen, Ryder, Todd R, Rafferty, Michael F, Cody, Wayne L, Lotarski, Susan M, Miljanich, George P, Millerman, Elizabeth, Rock, David M, Song, Yuntao, Stoehr, Sally J, Taylor, Charles P, Weber, Mark L, Szoke, Balazs G, Vartanian, Mark G

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Novel Use of Substituted 1,4-Dihydrobenz[d][1,3]oxazin-2-ones in the Synthesis of Important Aminomethyl o-Nitroanilines von Nikam, Sham S, Yuen, Po-Wai, Kornberg, Brian E, Tobias, Brian, Rafferty, Michael F

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Design and Synthesis of Novel Quinoxaline-2,3-dione AMPA/GlyN Receptor Antagonists:  Amino Acid Derivatives von Nikam, Sham S, Cordon, John J, Ortwine, Daniel F, Heimbach, Tycho H, Blackburn, Anthony C, Vartanian, Mark G, Nelson, Carrie B, Schwarz, Roy D, Boxer, Peter A, Rafferty, Michael F

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In Silico Pharmaceutical Property Prediction von Pil H. LeeMichael F. Rafferty

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Acute but not chronic activation of the NMDA-coupled glycine receptor with D-cycloserine facilitates learning and retention von Quartermain, David, Mower, Jay, Rafferty, Michael F., Herting, Robert L., Lanthorn, Thomas H.

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Editorial preface von Flynn, Daniel, Rafferty, Michael F.

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The discovery of [1-(4-dimethylamino-benzyl)-piperidin-4-yl]-[4-(3,3-dimethylbutyl)-phenyl]-(3-me thyl-but-2-enyl)-amine, an N-type Ca+2 channel blocker with oral activity for anal... von HU, L.-Y, RYDER, T. R, SZOKE, B. G, RAFFERTY, M. F, TAYLOR, C. P, FENG, M. R, KUO, B.-S, LOTARSKI, S. M, MILJANICH, G. P, MILLERMAN, E, SIEBERS, K. M

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Antinociceptive effect of spinally delivered prostaglandin E receptor antagonists in the formalin test on the rat von Malmberg, Annika B., Rafferty, Michael F., Yaksh, Tony L.

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Synthesis and biological evaluation of substituted 4-(OBz)phenylalanine derivatives as novel N-type calcium channel blockers von Hu, Lain-Yen, Ryder, Todd R., Nikam, Sham S., Millerman, Elizabeth, Szoke, Balazs G., Rafferty, Michael F.

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Multiple parallel synthesis of N, N-dialkyldipeptidylamines as N-type calcium channel blockers von Ryder, Todd R., Hu, Lain-Yen, Rafferty, Michael F., Millerman, Elizabeth, Szoke, Balazs G., Tarczy-Hornoch, Katalin

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Synthesis, configuration, and evaluation of two conformationally restrained analogs of phencyclidine von De Costa, Brian R, George, Clifford, Burke, Terrence R, Rafferty, Michael F, Contreras, Patricia C, Mick, Stephen J, Jacobson, Arthur E, Rice, Kenner C

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Editorial announcement von Flynn, Daniel L., Rafferty, Michael F.

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Editorial announcement von Flynn, Daniel L., Rafferty, Michael F.

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