Trends in Research on Traditional Chinese Health Exercises for Improving Cognitive Function: A Bibliometric Analysis of the Literature From 2001 to 2020 von Li, Wenlong, Weng, Linman, Xiang, Qiuping, Fan, Tonggang

Volltext

Effect of different conditioning methods of traditional Chinese health exercise on lung function in healthy middle-aged and elderly people: study protocol for a randomized controll... von Li, Wenlong, Song, Yapei, Xiang, Qiuping, Wang, Xinlei, Wei, Xiaoyun, Fan, Tonggang

Volltext

CBP/p300 bromodomain: new promising epigenetic target von Xiang, Qiuping, Zhou, Yang, Zhang, Yan, Xu, Yong

Volltext

Structural insights revealed by the cocrystal structure of CCS1477 in complex with CBP bromodomain von Xu, Hongrui, Luo, Guolong, Wu, Tianbang, Hu, Jiankang, Wang, Chao, Wu, Xishan, Zhang, Yan, Xu, Yong, Xiang, Qiuping

Volltext

Design, synthesis, and biological evaluation of 2-(naphthalen-1-yloxy)-N-phenylacetamide derivatives as TRPM4 inhibitors for the treatment of prostate cancer von Niu, Le, Liu, Huina, Li, Xiaomei, Wang, Lin, Hua, Hui, Cao, Qiaofeng, Xiang, Qiuping, Cai, Ting, Zhu, Dongsheng

Volltext

Discovery of Benzo[cd]indol-2(1H)‑ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation von Xue, Xiaoqian, Zhang, Yan, Liu, Zhaoxuan, Song, Ming, Xing, Yanli, Xiang, Qiuping, Wang, Zhen, Tu, Zhengchao, Zhou, Yulai, Ding, Ke, Xu, Yong

Volltext

Design, Synthesis, and Biological Evaluation of 1‑(Indolizin-3-yl)ethan-1-ones as CBP Bromodomain Inhibitors for the Treatment of Prostate Cancer von Xiang, Qiuping, Wang, Chao, Wu, Tianbang, Zhang, Cheng, Hu, Qingqing, Luo, Guolong, Hu, Jiankang, Zhuang, Xiaoxi, Zou, Lingjiao, Shen, Hui, Wu, Xishan, Zhang, Yan, Kong, Xiangqian, Liu, Jinsong, Xu, Yong

Volltext

Design, Synthesis, and Biological Evaluation of Hydrophobic-Tagged Glutathione Peroxidase 4 (GPX4) Degraders von Li, Xiaomei, Hu, Mengdie, Zhang, Yanping, Hua, Hui, Sun, Yujie, Xiang, Qiuping, Zhu, Dongsheng

Volltext

Discovery of a Promising CBP/p300 Degrader XYD129 for the Treatment of Acute Myeloid Leukemia von Wu, Tianbang, Hu, Jiankang, Zhao, Xiaofan, Zhang, Cheng, Dong, Ruibo, Hu, Qingqing, Xu, Hongrui, Shen, Hui, Zhang, Xiaohan, Zhang, Yan, Lin, Bin, Wu, Xishan, Xiang, Qiuping, Xu, Yong

Volltext

ROR-γ drives androgen receptor expression and represents a therapeutic target in castration-resistant prostate cancer von Wang, Junjian, Zou, June X, Xue, Xiaoqian, Cai, Demin, Zhang, Yan, Duan, Zhijian, Xiang, Qiuping, Yang, Joy C, Louie, Maggie C, Borowsky, Alexander D, Gao, Allen C, Evans, Christopher P, Lam, Kit S, Xu, Jianzhen, Kung, Hsing-Jien, Evans, Ronald M, Xu, Yong, Chen, Hong-Wu

Volltext

Structure-Based Discovery and Optimization of Benzo[d]­isoxazole Derivatives as Potent and Selective BET Inhibitors for Potential Treatment of Castration-Resistant Prostate Cancer... von Zhang, Maofeng, Zhang, Yan, Song, Ming, Xue, Xiaoqian, Wang, Junjian, Wang, Chao, Zhang, Cheng, Li, Chenchang, Xiang, Qiuping, Zou, Lingjiao, Wu, Xishan, Wu, Chun, Dong, Baijun, Xue, Wei, Zhou, Yulai, Chen, Hongwu, Wu, Donghai, Ding, Ke, Xu, Yong

Volltext

Discovery of the First BRD4 Second Bromodomain (BD2)-Selective Inhibitors von Li, Junhua, Hu, Qingqing, Zhu, Run, Dong, Ruibo, Shen, Hui, Hu, Jiankang, Zhang, Cheng, Zhang, Xiaohan, Xu, Tingting, Xiang, Qiuping, Zhang, Yan, Lin, Bin, Zhao, Linxiang, Wu, Xishan, Xu, Yong

Volltext

Discovery of Highly Potent and Efficient CBP/p300 Degraders with Strong In Vivo Antitumor Activity von Hu, Jiankang, Xu, Hongrui, Wu, Tianbang, Zhang, Cheng, Shen, Hui, Dong, Ruibo, Hu, Qingqing, Xiang, Qiuping, Chai, Shuang, Luo, Guolong, Chen, Xiaoshan, Huang, Yumin, Zhao, Xiaofan, Peng, Chao, Wu, Xishan, Lin, Bin, Zhang, Yan, Xu, Yong

Volltext

ZX703: A Small-Molecule Degrader of GPX4 Inducing Ferroptosis in Human Cancer Cells von Hu, Mengdie, Li, Xiaomei, Wang, Lin, Zhang, Yanping, Sun, Yujie, Hua, Hui, Liu, Huina, Cai, Ting, Zhu, Dongsheng, Xiang, Qiuping

Volltext

Discovery of a Highly Selective and H435R-Sensitive Thyroid Hormone Receptor β Agonist von Li, Qiu, Yao, Benqiang, Zhao, Shiting, Lu, Zhou, Zhang, Yan, Xiang, Qiuping, Wu, Xishan, Yu, Haonan, Zhang, Cheng, Li, Junhua, Zhuang, Xiaoxi, Wu, Donghai, Li, Yong, Xu, Yong

Volltext

2-Amino-2,3-dihydro-1 H -indene-5-carboxamide-Based Discoidin Domain Receptor 1 (DDR1) Inhibitors: Design, Synthesis, and in Vivo Antipancreatic Cancer Efficacy von Zhu, Dongsheng, Huang, Huocong, Pinkas, Daniel M, Luo, Jinfeng, Ganguly, Debolina, Fox, Alice E, Arner, Emily, Xiang, Qiuping, Tu, Zheng-Chao, Bullock, Alex N, Brekken, Rolf A, Ding, Ke, Lu, Xiaoyun

Volltext

2‑Amino-2,3-dihydro‑1H‑indene-5-carboxamide-Based Discoidin Domain Receptor 1 (DDR1) Inhibitors: Design, Synthesis, and in Vivo Antipancreatic Cancer Efficacy von Zhu, Dongsheng, Huang, Huocong, Pinkas, Daniel M, Luo, Jinfeng, Ganguly, Debolina, Fox, Alice E, Arner, Emily, Xiang, Qiuping, Tu, Zheng-Chao, Bullock, Alex N, Brekken, Rolf A, Ding, Ke, Lu, Xiaoyun

Volltext

Discovery and optimization of 1-(1H-indol-1-yl)ethanone derivatives as CBP/EP300 bromodomain inhibitors for the treatment of castration-resistant prostate cancer von Xiang, Qiuping, Wang, Chao, Zhang, Yan, Xue, Xiaoqian, Song, Ming, Zhang, Cheng, Li, Chenchang, Wu, Chun, Li, Kuai, Hui, Xiaoyan, Zhou, Yulai, Smaill, Jeff B., Patterson, Adam V., Wu, Donghai, Ding, Ke, Xu, Yong

Volltext

Discovery and Characterization of Benzimidazole Derivative XY123 as a Potent, Selective, and Orally Available RORγ Inverse Agonist von Wu, Xishan, Shen, Hui, Zhang, Yan, Wang, Chao, Li, Qiu, Zhang, Cheng, Zhuang, Xiaoxi, Li, Chenchang, Shi, Yudan, Xing, Yanli, Xiang, Qiuping, Xu, Jinxin, Wu, Donghai, Liu, Jinsong, Xu, Yong

Volltext

Optimization of the synthesis of BET BD2 selective inhibitor XY153 von Zhu, Run, Li, Junhua, Dong, Ruibo, Hu, Qingqing, Chen, Zhiming, Chen, Xiaoshan, Zhong, Zhixin, Xiang, Qiuping, Huang, Cen, Lin, Bin, Wu, Xishan, Zhang, Yan, Zhao, Linxiang, Xu, Yong

Volltext