Design, Synthesis and Characterization of a New Series of Fluorescent Metabotropic Glutamate Receptor Type 5 Negative Allosteric Modulators von Fernández-Dueñas, Víctor, Qian, Mingcheng, Argerich, Josep, Amaral, Carolina, Risseeuw, Martijn D P, Van Calenbergh, Serge, Ciruela, Francisco

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Visible-Light-Mediated Cyclopropanation Reactions of 3-Diazooxindoles with Arenes von Zhao, Shuai, Chen, Xiang-Xiang, Gao, Nan, Qian, Mingcheng, Chen, Xin

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Pyrazolone structural motif in medicinal chemistry: Retrospect and prospect von Zhao, Zefeng, Dai, Xufen, Li, Chenyang, Wang, Xiao, Tian, Jiale, Feng, Ying, Xie, Jing, Ma, Cong, Nie, Zhuang, Fan, Peinan, Qian, Mingcheng, He, Xirui, Wu, Shaoping, Zhang, Yongmin, Zheng, Xiaohui

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Visible-light-mediated cyclopropanation reactions of 3-diazooxindoles with olefins von Mu, Zhuangzhuang, Xie, Haochi, Gan, Shundong, Li, Hujin, Hou, Yanan, Qian, Mingcheng, Zhao, Shuai, Chen, Xin

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Visible-light-mediated O–H functionalization reactions of acetylenic alcohols with 3-diazooxindoles: Facile access to spirooxindole-fused oxacycles von Xu, Liqin, Wang, Jing, Li, Hujin, Xie, Haochi, Qian, Mingcheng, Hou, Yanan, Zhao, Shuai, Chen, Xin

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Study of G protein-coupled receptors dimerization: From bivalent ligands to drug-like small molecules von Qian, Mingcheng, Sun, Zhengyang, Chen, Xin, Van Calenbergh, Serge

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Structure optimization of Cmpd-15 as negative allosteric modulators for the β2-adrenergic receptor von Guo, Xue, Luo, Zhijie, Qi, Ying, Hei, Xiaoyuan, Zhang, Xin, Cao, Xuli, Qian, Mingcheng, Zhao, Shuai, Hou, Yanan, Chen, Xin

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Discovery and biological evaluation of cholic acid derivatives as potent TGR5 positive allosteric modulators von Li, Yan, Sun, Jingjing, Wang, Xiao, Luo, Zhijie, Shao, Xuemei, Li, Yingxiu, Cao, Qirong, Zhao, Shuai, Qian, Mingcheng, Chen, Xin

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Stereoselective Synthesis of Tetrasubstituted Olefins via Visible-Light-Promoted Iodine-Mediated Homo-Coupling of Diazo von Zhao, Shuai, Gao, Nan, Bao, Ning, Qian, Mingcheng, Chen, Zi-Yun, Zhang, Meng-Jia, Chen, Xin

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Allosteric Inhibition of the β 2 -Adrenergic Receptor: Design and Synthesis of Cmpd-15 Analogs von Ye, Kexin, Li, Qing, Luo, Zhijie, Lu, Qianchen, Rui, Xue, Li, Yan, Jin, Jie, Jing, Chenchen, Hong, Meiling, Qian, Mingcheng, Zhao, Shuai, Hou, Yanan, Chen, Xin

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Allosteric Inhibition of the β2‐Adrenergic Receptor: Design and Synthesis of Cmpd‐15 Analogs von Ye, Kexin, Li, Qing, Luo, Zhijie, Lu, Qianchen, Rui, Xue, Li, Yan, Jin, Jie, Jing, Chenchen, Hong, Meiling, Qian, Mingcheng, Zhao, Shuai, Hou, Yanan, Chen, Xin

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Synthesis, Biological Evaluation, and Docking Study of Ring‐Opening Amide Analogs of Matrine as Antitumor Agents von Qian, Mingcheng, Jiang, Xinyu, Zhang, Mingting, Hu, Lijuan, Liu, Huimin, Zhao, Shuai, Zhou, Xiaoying, Chen, Xin

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Synthesis of Bitopic Ligands as Potent Dopamine D 2 Receptor Agonists von Qian, Mingcheng, Zhou, Kuo, Wu, Yi, Luo, Zhijie, Xiao, Zhekai, Sun, Jingjing, Zeng, Siyu, Yao, Yi, Zhao, Shuai, Chen, Xin

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Discovery of a true bivalent dopamine D2 receptor agonist von Qian, Mingcheng, Ricarte, Adrián, Wouters, Elise, Dalton, James A.R., Risseeuw, Martijn D.P., Giraldo, Jesús, Van Calenbergh, Serge

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Stereoselective Synthesis of Enamides through Palladium‐Catalyzed Oxidative Amidation of Conjugated Olefins with 2‐Pyridones von Zhao, Shuai, Lu, Bin‐Wei, Bao, Ning, Yin, Zi‐Jian, Qian, Mingcheng, Cao, Lin, Geng, Min, Lin, Ye, Chen, Xin

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Design, synthesis and characterization of a new series of fluorescent metabotropic glutamate receptor type 5 negative allosteric modulators von Fernández-Dueñas, Víctor, Qian, Mingcheng, Argerich, Josep, Amaral, Carolina, Risseeuw, Martijn, Van Calenbergh, Serge, Ciruela, Francisco

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Front Cover: Synthesis, Biological Evaluation, and Docking Study of Ring‐Opening Amide Analogs of Matrine as Antitumor Agents (4/2021) von Qian, Mingcheng, Jiang, Xinyu, Zhang, Mingting, Hu, Lijuan, Liu, Huimin, Zhao, Shuai, Zhou, Xiaoying, Chen, Xin

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Design, synthesis and characterization of a new series of fluorescent metabotropic glutamate receptor type 5 negative allosteric modulators von Fernández Dueñas, Víctor, Qian, Mingcheng, Argerich, Josep, Amaral, Carolina, Risseeuw, Martijn D.P, Van Calenbergh, Serge, Ciruela Alférez, Francisco

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Discovery of novel cholic acid derivatives as highly potent agonists for G protein-coupled bile acid receptor von Qian, Mingcheng, Luo, Zhijie, Hou, Wenwen, Sun, Jingjing, Lu, Xin, Zhang, Qianxi, Wu, Yi, Xue, Caile, Zhao, Shuai, Chen, Xin

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Discovery of a true bivalent dopamine D 2 receptor agonist von Qian, Mingcheng, Ricarte, Adrián, Wouters, Elise, Dalton, James A R, Risseeuw, Martijn D P, Giraldo, Jesús, Van Calenbergh, Serge

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