Catalytic enantioselective synthesis of quaternary carbon stereocentres von Quasdorf, Kyle W., Overman, Larry E.

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Direct Construction of Quaternary Carbons from Tertiary Alcohols via Photoredox-Catalyzed Fragmentation of tert-Alkyl N‑Phthalimidoyl Oxalates von Lackner, Gregory L, Quasdorf, Kyle W, Overman, Larry E

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Nickel-Catalyzed Cross-Couplings Involving Carbon−Oxygen Bonds von Rosen, Brad M, Quasdorf, Kyle W, Wilson, Daniella A, Zhang, Na, Resmerita, Ana-Maria, Garg, Neil K, Percec, Virgil

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Cross-Coupling Reactions of Aryl Pivalates with Boronic Acids von Quasdorf, Kyle W, Tian, Xia, Garg, Neil K

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Fragment Coupling and the Construction of Quaternary Carbons Using Tertiary Radicals Generated From tert-Alkyl N‑Phthalimidoyl Oxalates By Visible-Light Photocatalysis von Lackner, Gregory L, Quasdorf, Kyle W, Pratsch, Gerald, Overman, Larry E

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Suzuki−Miyaura Cross-Coupling of Aryl Carbamates and Sulfamates: Experimental and Computational Studies von Quasdorf, Kyle W, Antoft-Finch, Aurora, Liu, Peng, Silberstein, Amanda L, Komaromi, Anna, Blackburn, Tom, Ramgren, Stephen D, Houk, K. N, Snieckus, Victor, Garg, Neil K

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Total Synthesis of (−)-N-Methylwelwitindolinone C Isothiocyanate von Huters, Alexander D, Quasdorf, Kyle W, Styduhar, Evan D, Garg, Neil K

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Total Synthesis of Oxidized Welwitindolinones and (−)-N-Methylwelwitindolinone C Isonitrile von Quasdorf, Kyle W, Huters, Alexander D, Lodewyk, Michael W, Tantillo, Dean J, Garg, Neil K

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Mechanistic Insights into the Racemization of Fused Cyclopropyl Isoxazolines von Quasdorf, Kyle W, Birkholz, Adam B, Bartberger, Michael D, Colyer, John, Osgood, Stephen, Crossley, Kevin, Caille, Seb

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Suzuki−Miyaura Coupling of Aryl Carbamates, Carbonates, and Sulfamates von Quasdorf, Kyle W, Riener, Michelle, Petrova, Krastina V, Garg, Neil K

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Ipso Nitration of Aryl Boronic Acids Using Fuming Nitric Acid von Murray, James I, Silva Elipe, Maria V, Baucom, Kyle D, Brown, Derek B, Quasdorf, Kyle, Caille, Seb

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Kinetic Investigations To Enable Development of a Robust Radical Benzylic Bromination for Commercial Manufacturing of AMG 423 Dihydrochloride Hydrate von Murray, James I, Silva Elipe, Maria V, Cosbie, Andrew, Baucom, Kyle, Quasdorf, Kyle, Caille, Seb

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Ni-Catalyzed Enantioselective Desymmetrization: Development of Divergent Acyl and Decarbonylative Cross-Coupling Reactions von Hernández-Mejías, Ángel D, Shimozono, Alexander M, Hazra, Avijit, Richter, Sven, Tong, Zhengjia, Langille, Neil F, Quasdorf, Kyle, Parsons, Andrew T, Sigman, Matthew S, Reisman, Sarah E

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Catalytic Enantioselective Synthesis of Quaternary Carbon Stereocenters von Quasdorf, Kyle W., Overman, Larry E.

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Structural Elucidation and Absolute Stereochemistry for Pharma Compounds Using MicroED von de Moraes, Lygia Silva, Burch, Jessica E., Delgadillo, David A., Rodriguez, Isabel Hernandez, Mai, Huanghao, Smith, Austin G., Caille, Seb, Walker, Shawn D., Wurz, Ryan P., Cee, Victor J., Rodriguez, Jose A., Gostovic, Dan, Quasdorf, Kyle, Nelson, Hosea M.

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Development of a Continuous Photochemical Bromination/Alkylation Sequence En Route to AMG 423 von Quasdorf, Kyle, Murray, James I, Nguyen, Hanh, Silva Elipe, Maria V, Ericson, Ari, Kircher, Eric, Guan, Lianxiu, Caille, Seb

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Development of a scalable route to a complex cyclobutane linchpin via a diastereoselective CuI-catalyzed vinylation of a cyclobutanyl aldehyde von Corbett, Michael T., Baucom, Kyle, Cui, Sheng, Dornan, Peter K., Jiao, Fangxia, Han, Jun, Langille, Neil F., Osgood, Steve, Parsons, Andrew T., Quasdorf, Kyle W., Rötheli, Andreas R., Elipe, Maria Victoria Silva, Sangodkar, Rahul P., Smith, Austin G., Spada, Simone, Stahl, Amanda E., St-Pierre, Gabrielle, Thiel, Oliver R., Walker, Shawn D., Xie, Yong, Yang, Ning

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Development of a Commercial Manufacturing Process for Sotorasib, a First-in-Class KRASG12C Inhibitor von Zhang, Liang, Griffin, Daniel J., Beaver, Matthew G., Blue, Laura E., Borths, Christopher J., Brown, Derek B., Caille, Seb, Chen, Ying, Cherney, Alan H., Cochran, Brian M., Colyer, John T., Corbett, Michael T., Correll, Tiffany L., Crockett, Richard D., Dai, Xi-Jie, Dornan, Peter K., Farrell, Robert P., Hedley, Simon J., Hsieh, Hsiao-Wu, Huang, Liang, Huggins, Seth, Liu, Min, Lovette, Michael A., Quasdorf, Kyle, Reifman, Jonathan, Robinson, Jo Anna, Sangodkar, Rahul P., Sharma, Sonika, Kumar, Srividya Sharvan, Smith, Austin G., St-Pierre, Gabrielle, Tedrow, Jason S., Thiel, Oliver R., Truong, Jonathan V., Walker, Shawn D., Wei, Carolyn S., Wilsily, Ashraf, Xie, Yong, Yang, Ning, Parsons, Andrew T.

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Development of a Commercial Manufacturing Process for Sotorasib, a First-in-Class KRAS G12C Inhibitor von Zhang, Liang, Griffin, Daniel J., Beaver, Matthew G., Blue, Laura E., Borths, Christopher J., Brown, Derek B., Caille, Seb, Chen, Ying, Cherney, Alan H., Cochran, Brian M., Colyer, John T., Corbett, Michael T., Correll, Tiffany L., Crockett, Richard D., Dai, Xi-Jie, Dornan, Peter K., Farrell, Robert P., Hedley, Simon J., Hsieh, Hsiao-Wu, Huang, Liang, Huggins, Seth, Liu, Min, Lovette, Michael A., Quasdorf, Kyle, Powazinik, William, Reifman, Jonathan, Robinson, Jo Anna, Sangodkar, Rahul P., Sharma, Sonika, Kumar, Srividya Sharvan, Smith, Austin G., St-Pierre, Gabrielle, Tedrow, Jason S., Thiel, Oliver R., Truong, Jonathan V., Walker, Shawn D., Wei, Carolyn S., Wilsily, Ashraf, Xie, Yong, Yang, Ning, Parsons, Andrew T.

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A fluorophosphate-based inverse Keggin structure von Fielden, John, Quasdorf, Kyle, Cronin, Leroy, Kögerler, Paul

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