Structural Basis of Constitutive Activity and a Unique Nucleotide Binding Mode of Human Pim-1 Kinase von Qian, Kevin C., Wang, Lian, Hickey, Eugene R., Studts, Joey, Barringer, Kevin, Peng, Charline, Kronkaitis, Anthony, Li, Jun, White, Andre, Mische, Sheenah, Farmer, Bennett

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Benzimidazolone as potent chymase inhibitor: Modulation of reactive metabolite formation in the hydrophobic (P 1) region von Lo, Ho Yin, Nemoto, Peter A., Kim, Jin Mi, Hao, Ming-Hong, Qian, Kevin C., Farrow, Neil A., Albaugh, Daniel R., Fowler, Danielle M., Schneiderman, Richard D., Michael August, E., Martin, Leslie, Hill-Drzewi, Melissa, Pullen, Steven S., Takahashi, Hidenori, De Lombaert, Stéphane

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Discovery and design of benzimidazolone based inhibitors of p38 MAP kinase von Hammach, Abdelhakim, Barbosa, Antonio, Gaenzler, Faith Corbo, Fadra, Tazmeen, Goldberg, Daniel, Hao, Ming-Hong, Kroe, Rachel R., Liu, Pingrong, Qian, Kevin C., Ralph, Mark, Sarko, Christopher, Soleymanzadeh, Fariba, Moss, Neil

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Discovery and Optimization of p38 Inhibitors via Computer-Assisted Drug Design von Goldberg, Daniel R, Hao, Ming-Hong, Qian, Kevin C, Swinamer, Alan D, Gao, Donghong A, Xiong, Zhaoming, Sarko, Chris, Berry, Angela, Lord, John, Magolda, Ronald L, Fadra, Tazmeen, Kroe, Rachel R, Kukulka, Alison, Madwed, Jeffrey B, Martin, Leslie, Pargellis, Christopher, Skow, Donna, Song, Jinhua J, Tan, Zhulin, Torcellini, Carol A, Zimmitti, Clare S, Yee, Nathan K, Moss, Neil

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Second-Generation Lymphocyte Function-Associated Antigen-1 Inhibitors:  1H-Imidazo[1,2-α]imidazol-2-one Derivatives von Wu, Jiang-Ping, Emeigh, Jonathan, Gao, Donghong A, Goldberg, Daniel R, Kuzmich, Daniel, Miao, Clara, Potocki, Ian, Qian, Kevin C, Sorcek, Ronald J, Jeanfavre, Deborah D, Kishimoto, Kei, Mainolfi, Elizabeth A, Nabozny, Gerald, Peng, Charline, Reilly, Patricia, Rothlein, Robert, Sellati, Rosemarie H, Woska, Joseph R, Chen, Shirlynn, Gunn, Jocelyn A, O'Brien, Drane, Norris, Stephen H, Kelly, Terence A

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New modifications to the area of pyrazole-naphthyl urea based p38 MAP kinase inhibitors that bind to the adenine/ATP site von Moss, Neil, Breitfelder, Steffen, Betageri, Raj, Cirillo, Pier F., Fadra, Tazmeen, Hickey, Eugene R., Kirrane, Thomas, Kroe, Rachel R., Madwed, Jeffrey, Nelson, Richard M., Pargellis, Christopher A., Qian, Kevin C., Regan, John, Swinamer, Alan, Torcellini, Carol

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Discovery and characterization of the N-phenyl- N′-naphthylurea class of p38 kinase inhibitors von Cirillo, Pier F., Hickey, Eugene R., Moss, Neil, Breitfelder, Steffen, Betageri, Raj, Fadra, Tazmeen, Gaenzler, Faith, Gilmore, Thomas, Goldberg, Daniel R., Kamhi, Victor, Kirrane, Thomas, Kroe, Rachel R., Madwed, Jeffrey, Moriak, Monica, Netherton, Matthew, Pargellis, Christopher A., Patel, Usha R., Qian, Kevin C., Sharma, Rajiv, Sun, Sanxing, Swinamer, Alan, Torcellini, Carol, Takahashi, Hidenori, Tsang, Michele, Xiong, Zhaoming

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Expression, purification, crystallization and preliminary crystallographic analysis of human Pim-­1 kinase von Qian, Kevin C., Studts, Joey, Wang, Lian, Barringer, Kevin, Kronkaitis, Anthony, Peng, Charline, Baptiste, Alistair, LaFrance, Roger, Mische, Sheenah, Farmer, Bennett

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Second-Generation Lymphocyte Function-Associated Antigen-1 Inhibitors:  1 H -Imidazo[1,2-α]imidazol-2-one Derivatives von Wu, Jiang-Ping, Emeigh, Jonathan, Gao, Donghong A., Goldberg, Daniel R., Kuzmich, Daniel, Miao, Clara, Potocki, Ian, Qian, Kevin C., Sorcek, Ronald J., Jeanfavre, Deborah D., Kishimoto, Kei, Mainolfi, Elizabeth A., Nabozny, Gerald, Peng, Charline, Reilly, Patricia, Rothlein, Robert, Sellati, Rosemarie H., Woska, Joseph R., Chen, Shirlynn, Gunn, Jocelyn A., O'Brien, Drane, Norris, Stephen H., Kelly, Terence A.

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Cytokine Inhibitors von SWINAMER ALAN D, HAO MING-HONG, COGAN DEREK A, QIAN KEVIN C

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Cytokine Inhibitors von HAO MING-HONG, RALPH MARK S, KAMHI VICTOR M, QIAN KEVIN C, CIRILLO PIER F, HAMMACH ABDELHAKIM, GOLDBERG DANIEL R, WU LIFEN, AUNGST RONALD A.JR, GAO DONGHONG A, MOSS NEIL, NETHERTON MATTHEW R, XIONG ZHAOMING

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Cytokine inhibitors von MING-HONG HAO, ZHAOMING XIONG, AUNGST, RONALD, A, JR, GOLDBERG, DANIEL, R, NEIL MOSS, QIAN, KEVIN, C, MARC VICTOR, ABDELHAKIM HAMMACH, RUSSEL NETHERTON, LIFEN WU, GAO, DONGHONG, A, RALPH, MARK, S, CIRILLO, PIER, F, VITOR KAHMHI

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Heterocyclic N-aryl carboxamides as cytokine inhibitors von CIRILLO PIER F.,GAO DONGHONG,GOLDBERG D. R.,HAMMACH A.,HAO MING-HONG,KAMHI VICTOR M.,MOSS NEIL,NETHERTON R.,QIAN KEVIN C.,RALPH MARK S.,WU LIFEN,XIONG ZHAOMING,AUNGST RONALD A. JR. ALBANY MOLE

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HETEROCYCLIC N-ARYL CARBOXAMIDES AS CYTOKINE INHIBITORS von WU, LIFEN, HAO, MING-HONG, AUNGST, RONALD A. JR, GAO, DONGHONG A, CIRILLO, PIER F, MOSS, NEIL, GOLDBERG, D.R, HAMMACH, A, RALPH, MARK S, KAMHI, VICTOR M, XIONG, ZHAOMING, NETHERTON, R, QIAN, KEVIN C

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Novel BET protein proteolysis-targeting chimera exerts superior lethal activity than bromodomain inhibitor (BETi) against post-myeloproliferative neoplasm secondary (s) AML cells von Saenz, D T, Fiskus, W, Qian, Y, Manshouri, T, Rajapakshe, K, Raina, K, Coleman, K G, Crew, A P, Shen, A, Mill, C P, Sun, B, Qiu, P, Kadia, T M, Pemmaraju, N, DiNardo, C, Kim, M-S, Nowak, A J, Coarfa, C, Crews, C M, Verstovsek, S, Bhalla, K N

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Video-rate high-precision time-frequency multiplexed 3D coherent ranging von Qian, Ruobing, Zhou, Kevin C., Zhang, Jingkai, Viehland, Christian, Dhalla, Al-Hafeez, Izatt, Joseph A.

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Spatial multiomics map of trophoblast development in early pregnancy von Arutyunyan, Anna, Roberts, Kenny, Troulé, Kevin, Wong, Frederick C. K., Sheridan, Megan A., Kats, Ilia, Garcia-Alonso, Luz, Velten, Britta, Hoo, Regina, Ruiz-Morales, Elias R., Sancho-Serra, Carmen, Shilts, Jarrod, Handfield, Louis-Francois, Marconato, Luca, Tuck, Elizabeth, Gardner, Lucy, Mazzeo, Cecilia Icoresi, Li, Qian, Kelava, Iva, Wright, Gavin J., Prigmore, Elena, Teichmann, Sarah A., Bayraktar, Omer Ali, Moffett, Ashley, Stegle, Oliver, Turco, Margherita Y., Vento-Tormo, Roser

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Brain Insulin Lowers Circulating BCAA Levels by Inducing Hepatic BCAA Catabolism von Shin, Andrew C., Fasshauer, Martin, Filatova, Nika, Grundell, Linus A., Zielinski, Elizabeth, Zhou, Jian-Ying, Scherer, Thomas, Lindtner, Claudia, White, Phillip J., Lapworth, Amanda L., Ilkayeva, Olga, Knippschild, Uwe, Wolf, Anna M., Scheja, Ludger, Grove, Kevin L., Smith, Richard D., Qian, Wei-Jun, Lynch, Christopher J., Newgard, Christopher B., Buettner, Christoph

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Biomarker Changes Associated With Both Dulaglutide and Cardiovascular Events in the REWIND Randomized Controlled Trial: A Nested Case-Control Post Hoc Analysis von Gerstein, Hertzel C, Lee, Shun-Fu, Paré, Guillaume, Bethel, M Angelyn, Colhoun, Helen M, Hoover, Anastasia, Lakshmanan, Mark, Lin, Yanzhu, Pirro, Valentino, Qian, Hui-Rong, Ruotolo, Giacomo, Ryden, Lars, Wilson, Jonathan M, Duffin, Kevin L

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High thermoelectric performance by resonant dopant indium in nanostructured SnTe von Zhang, Qian, Liao, Bolin, Lan, Yucheng, Lukas, Kevin, Liu, Weishu, Esfarjani, Keivan, Opeil, Cyril, Broido, David, Chen, Gang, Ren, Zhifeng

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