Copper-Catalyzed Domino Cycloaddition/CN Coupling/Cyclization/(CH Arylation): An Efficient Three-Component Synthesis of Nitrogen Polyheterocycles von Qian, Wenyuan, Wang, Hao, Allen, Jennifer

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A new wave of innovations within the DNA damage response von Li, Qi, Qian, Wenyuan, Zhang, Yang, Hu, Lihong, Chen, Shuhui, Xia, Yuanfeng

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A “Click and Activate” Approach in One-Pot Synthesis of a Triazolyl-Pyridazinone Library von Qian, Wenyuan, Winternheimer, David, Allen, Jennifer

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One-pot synthesis of [1,2,3]triazole-fused pyrazinopyridazindione tricycles by a ‘click and activate’ approach von Qian, Wenyuan, Winternheimer, David, Amegadzie, Albert, Allen, Jennifer

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Convergent, Regioselective Synthesis of Tetrakisfulleroids from C60 von Qian, Wenyuan, Rubin, Yves

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Discovery of dihydroquinoxalinone acetamides containing bicyclic amines as potent Bradykinin B1 receptor antagonists von Chen, Jian Jeffrey, Qian, Wenyuan, Biswas, Kaustav, Viswanadhan, Vellarkad N., Askew, Benny C., Hitchcock, Stephen, Hungate, Randall W., Arik, Leyla, Johnson, Eileen

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Total Synthesis and Structural Elucidation of Azaspiracid-1. Construction of Key Building Blocks for Originally Proposed Structure von Nicolaou, K. C, Pihko, Petri M, Bernal, Federico, Frederick, Michael O, Qian, Wenyuan, Uesaka, Noriaki, Diedrichs, Nicole, Hinrichs, Jürgen, Koftis, Theocharis V, Loizidou, Eriketi, Petrovic, Goran, Rodriquez, Manuela, Sarlah, David, Zou, Ning

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Total Synthesis of the Proposed Azaspiracid-1 Structure, Part 1: Construction of the Enantiomerically Pure C1-C20, C21-C27, and C28-C40 Fragments von Nicolaou, K. C., Li, Yiwei, Uesaka, Noriaki, Koftis, Theocharis V., Vyskocil, Stepan, Ling, Taotao, Govindasamy, Mugesh, Qian, Wenyuan, Bernal, Federico, Chen, David Y.-K.

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Towards Sixfold Functionalization of Buckminsterfullerene (C60) at Fully Addressable Octahedral Sites von Qian, Wenyuan, Rubin, Yves

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Discovery of dehydro-oxopiperazine acetamides as novel bradykinin B1 receptor antagonists with enhanced in vitro potency von Qian, Wenyuan, Chen, Jian Jeffrey, Human, Jason, Aya, Toshihiro, Zhu, Jiawang, Biswas, Kaustav, Peterkin, Tanya, Hungate, Randall W., Arik, Leyla, Johnson, Eileen, Kumar, Gondi, Joseph, Smriti, Jona, Janan, Guo, Hong-Xun, Wu, Zufan

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Synthesis of Stable Derivatives of C62:  The First Nonclassical Fullerene Incorporating a Four-Membered Ring von Qian, Wenyuan, Chuang, Shih-Ching, Amador, Roberto B, Jarrosson, Thibaut, Sander, Michael, Pieniazek, Susan, Khan, Saeed I, Rubin, Yves

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One-Pot Synthesis of 3‑Triazolyl-2-iminochromenes via a Catalytic Three Component Cascade Reaction von Qian, Wenyuan, Amegadzie, Albert, Winternheimer, David, Allen, Jennifer

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Copper-Catalyzed Domino Cycloaddition/CN Coupling/Cyclization/(CH Arylation): An Efficient Three-Component Synthesis of Nitrogen Polyheterocycles von Qian, Wenyuan, Wang, Hao, Allen, Jennifer

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Identification of TUL01101: A Novel Potent and Selective JAK1 Inhibitor for the Treatment of Rheumatoid Arthritis von Zhou, Shuhao, Mao, Weiwei, Su, Yuan, Zheng, Xuejian, Qian, Wenyuan, Shen, Meiyue, Shan, Ningli, Li, Yaoshuang, Wang, Degang, Wu, Shouting, Sun, Tiemin, Mu, Liwei

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3-Oxo-2-piperazinyl acetamides as potent bradykinin B1 receptor antagonists for the treatment of pain and inflammation von Chen, Jian Jeffrey, Nguyen, Thomas, D’Amico, Derin C., Qian, Wenyuan, Human, Jason, Aya, Toshihiro, Biswas, Kaustav, Fotsch, Christopher, Han, Nianhe, Liu, Qingyian, Nishimura, Nobuko, Peterkin, Tanya A.N., Yang, Kevin, Zhu, Jiawang, Riahi, Babak Bobby, Hungate, Randall W., Andersen, Neil G., Colyer, John T., Faul, Margaret M., Kamassah, Augustus, Wang, Judy, Jona, Janan, Kumar, Gondi, Johnson, Eileen, Askew, Benny C.

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Aryl sulfones as novel Bradykinin B1 receptor antagonists for treatment of chronic pain von Biswas, Kaustav, Aya, Toshihiro, Qian, Wenyuan, Peterkin, Tanya A.N., Chen, Jian Jeffrey, Human, Jason, Hungate, Randall W., Kumar, Gondi, Arik, Leyla, Lester-Zeiner, Dianna, Biddlecome, Gloria, Manning, Barton H., Sun, Hong, Dong, Hong, Huang, Ming, Loeloff, Richard, Johnson, Eileen J., Askew, Benny C.

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Aryl sulfonamides containing tetralin allylic amines as potent and selective bradykinin B1 receptor antagonists von Liu, Qingyian, Qian, Wenyuan, Li, Aiwen, Biswas, Kaustav, Chen, Jian Jeffrey, Fotsch, Christopher, Han, Nianhe, Yuan, Chester, Arik, Leyla, Biddlecome, Gloria, Johnson, Eileen, Kumar, Gondi, Lester-Zeiner, Dianna, Ng, Gordon Y., Hungate, Randall W., Askew, Benny C.

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Accelerating Effect of Triazolyl and Related Heteroaryl Substituents on S N Ar Reactions: Evidence of Hydrogen-Bond Stabilized Transition States von Qian, Wenyuan, Wang, Hao, Bartberger, Michael D.

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Synthesis and evaluation of hydrazinyl-containing pyrrolo[2,3-d]pyrimidine series as potent, selective and oral JAK1 inhibitors for the treatment of rheumatoid arthritis von Mao, Weiwei, Wu, Hao, Guo, Qiang, Zheng, Xuejian, Wei, Changqing, Liao, Yonggang, Shen, Liang, Mi, Jingyu, Li, Jian, Chen, Shuhui, Qian, Wenyuan

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One-pot synthesis of 3-triazolyl-quinolin-2-(1H)-ones via sequential Ugi-“click”-Knoevenagel condensations von Qian, Wenyuan, Wang, Dahai, Wang, Honglin, Yu, Peng, Liu, Shilan, Chen, Shuhui

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