Targeting CBP and p300: Emerging Anticancer Agents von Masci, Domiziana, Puxeddu, Michela, Silvestri, Romano, La Regina, Giuseppe

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Metabolic Rewiring in Cancer: Small Molecule Inhibitors in Colorectal Cancer Therapy von Masci, Domiziana, Puxeddu, Michela, Silvestri, Romano, La Regina, Giuseppe

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Emerging Therapeutic Agents for Colorectal Cancer von Nalli, Marianna, Puxeddu, Michela, La Regina, Giuseppe, Gianni, Stefano, Silvestri, Romano

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Recent Advances in Drug Discovery for Triple-Negative Breast Cancer Treatment von Masci, Domiziana, Naro, Chiara, Puxeddu, Michela, Urbani, Andrea, Sette, Claudio, La Regina, Giuseppe, Silvestri, Romano

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A Novel Validated UHPLC Method for the Estimation of Rosuvastatin and Its Complete Impurity Profile in Tablet Formulations von Mammone, Francesca Romana, Zanitti, Leo, Puxeddu, Michela, La Regina, Giuseppe, Silvestri, Romano, Borioni, Anna, Cirilli, Roberto

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Discovery of a Novel Class of Norovirus Inhibitors with High Barrier of Resistance von Van Dycke, Jana, Puxeddu, Michela, La Regina, Giuseppe, Mastrangelo, Eloise, Tarantino, Delia, Rymenants, Jasper, Sebastiani, Jessica, Nalli, Marianna, Matthijnssens, Jelle, Neyts, Johan, Silvestri, Romano, Rocha-Pereira, Joana

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Targeting the Interaction between the SH3 Domain of Grb2 and Gab2 von Malagrino, Francesca, Coluccia, Antonio, Bufano, Marianna, La Regina, Giuseppe, Puxeddu, Michela, Toto, Angelo, Visconti, Lorenzo, Paone, Alessio, Magnifico, Maria Chiara, Troilo, Francesca, Cutruzzola, Francesca, Silvestri, Romano, Gianni, Stefano

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Chemo- and enantio-selective reversed-phase HPLC analysis of rosuvastatin using a cellulose-based chiral stationary phase in gradient elution mode von Mammone, Francesca Romana, Rotundo, Paola, Ferretti, Rosella, Puxeddu, Michela, Silvestri, Romano, Cirilli, Roberto

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Induction of Ferroptosis in Glioblastoma and Ovarian Cancers by a New Pyrrole Tubulin Assembly Inhibitor von Puxeddu, Michela, Wu, Jianchao, Bai, Ruoli, D’Ambrosio, Michele, Nalli, Marianna, Coluccia, Antonio, Manetto, Simone, Ciogli, Alessia, Masci, Domiziana, Urbani, Andrea, Fionda, Cinzia, Coni, Sonia, Bordone, Rosa, Canettieri, Gianluca, Bigogno, Chiara, Dondio, Giulio, Hamel, Ernest, Liu, Te, Silvestri, Romano, La Regina, Giuseppe

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RS6077 induces mitotic arrest and selectively activates cell death in human cancer cell lines and in a lymphoma tumor in vivo von Sebastiani, Jessica, Puxeddu, Michela, Nalli, Marianna, Bai, Ruoli, Altieri, Ludovica, Rovella, Paola, Gaudio, Eugenio, Trisciuoglio, Daniela, Spriano, Filippo, Lavia, Patrizia, Fionda, Cinzia, Masci, Domiziana, Urbani, Andrea, Bigogno, Chiara, Dondio, Giulio, Hamel, Ernest, Bertoni, Francesco, Silvestri, Romano, La Regina, Giuseppe

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Development of N -(4-(1 H -Imidazol-1-yl)phenyl)-4-chlorobenzenesulfonamide, a Novel Potent Inhibitor of β-Catenin with Enhanced Antitumor Activity and Metabolic Stability von Puxeddu, Michela, Ling, Lele, Ripa, Silvia, D’Ambrosio, Michele, Nalli, Marianna, Parisi, Anastasia, Sciò, Pietro, Coluccia, Antonio, Granese, Arianna, Santelli, Martina, Masci, Domiziana, Cuřínová, Petra, Naro, Chiara, Sette, Claudio, Pastore, Arianna, Stornaiuolo, Mariano, Bigogno, Chiara, Dondio, Giulio, Di Magno, Laura, Canettieri, Gianluca, Liu, Te, Silvestri, Romano, La Regina, Giuseppe

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4-(3-Phenyl-4-(3,4,5-trimethoxybenzoyl)-1 H -pyrrol-1-yl)benzenesulfonamide, a Novel Carbonic Anhydrase and Wnt/β-Catenin Signaling Pathway Dual-Targeting Inhibitor with Potent Act... von Masci, Domiziana, Puxeddu, Michela, Di Magno, Laura, D'Ambrosio, Michele, Parisi, Anastasia, Nalli, Marianna, Bai, Ruoli, Coluccia, Antonio, Sciò, Pietro, Orlando, Viviana, D'Angelo, Sara, Biagioni, Stefano, Urbani, Andrea, Hamel, Ernest, Nocentini, Alessio, Filiberti, Serena, Turati, Marta, Ronca, Roberto, Kopecka, Joanna, Riganti, Chiara, Fionda, Cinzia, Bordone, Rosa, Della Rocca, Giorgia, Canettieri, Gianluca, Supuran, Claudiu T, Silvestri, Romano, La Regina, Giuseppe

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CXCR4 antagonism sensitizes cancer cells to novel indole-based MDM2/4 inhibitors in glioblastoma multiforme von Daniele, Simona, La Pietra, Valeria, Piccarducci, Rebecca, Pietrobono, Deborah, Cavallini, Chiara, D'Amore, Vincenzo Maria, Cerofolini, Linda, Giuntini, Stefano, Russomanno, Pasquale, Puxeddu, Michela, Nalli, Marianna, Pedrini, Martina, Fragai, Marco, Luchinat, Claudio, Novellino, Ettore, Taliani, Sabrina, La Regina, Giuseppe, Silvestri, Romano, Martini, Claudia, Marinelli, Luciana

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4‑(3-Phenyl-4-(3,4,5-trimethoxybenzoyl)‑1H‑pyrrol-1-yl)benzenesulfonamide, a Novel Carbonic Anhydrase and Wnt/β-Catenin Signaling Pathway Dual-Targeting Inhibitor with Potent Activ... von Masci, Domiziana, Puxeddu, Michela, Di Magno, Laura, D’Ambrosio, Michele, Parisi, Anastasia, Nalli, Marianna, Bai, Ruoli, Coluccia, Antonio, Sciò, Pietro, Orlando, Viviana, D’Angelo, Sara, Biagioni, Stefano, Urbani, Andrea, Hamel, Ernest, Nocentini, Alessio, Filiberti, Serena, Turati, Marta, Ronca, Roberto, Kopecka, Joanna, Riganti, Chiara, Fionda, Cinzia, Bordone, Rosa, Della Rocca, Giorgia, Canettieri, Gianluca, Supuran, Claudiu T., Silvestri, Romano, La Regina, Giuseppe

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Discovery of pyrrole derivatives for the treatment of glioblastoma and chronic myeloid leukemia von Puxeddu, Michela, Shen, Hongliang, Bai, Ruoli, Coluccia, Antonio, Bufano, Marianna, Nalli, Marianna, Sebastiani, Jessica, Brancaccio, Diego, Da Pozzo, Eleonora, Tremolanti, Chiara, Martini, Claudia, Orlando, Viviana, Biagioni, Stefano, Sinicropi, Maria Stefania, Ceramella, Jessica, Iacopetta, Domenico, Coluccia, Addolorata Maria Luce, Hamel, Ernest, Liu, Te, Silvestri, Romano, La Regina, Giuseppe

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Targeting the Grb2 cSH3 domain: Design, synthesis and biological evaluation of the first series of modulators von Bufano, Marianna, Puxeddu, Michela, Nalli, Marianna, La Regina, Giuseppe, Toto, Angelo, Liberati, Francesca Romana, Paone, Alessio, Cutruzzolà, Francesca, Masci, Domiziana, Bigogno, Chiara, Dondio, Giulio, Silvestri, Romano, Gianni, Stefano, Coluccia, Antonio

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Structure-activity relationship studies and in vitro and in vivo anticancer activity of novel 3-aroyl-1,4-diarylpyrroles against solid tumors and hematological malignancies von Puxeddu, Michela, Shen, Hongliang, Bai, Ruoli, Coluccia, Antonio, Nalli, Marianna, Mazzoccoli, Carmela, Da Pozzo, Eleonora, Cavallini, Chiara, Martini, Claudia, Orlando, Viviana, Biagioni, Stefano, Mazzoni, Cristina, Coluccia, Addolorata Maria Luce, Hamel, Ernest, Liu, Te, Silvestri, Romano, La Regina, Giuseppe

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Discovery of New 1,1′-Biphenyl-4-sulfonamides as Selective Subnanomolar Human Carbonic Anhydrase II Inhibitors von La Regina, Giuseppe, Puxeddu, Michela, Nalli, Marianna, Vullo, Daniela, Gratteri, Paola, Supuran, Claudiu Trandafir, Nocentini, Alessio, Silvestri, Romano

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Sulfonamide Inhibitors of β‐Catenin Signaling as Anticancer Agents with Different Output on c‐MYC von Di Magno, Laura, Di Pastena, Fiorella, Puxeddu, Michela, La Regina, Giuseppe, Coluccia, Antonio, Ciogli, Alessia, Manetto, Simone, Maroder, Marella, Canettieri, Gianluca, Silvestri, Romano, Nalli, Marianna

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Discovery of Zika Virus NS2B/NS3 Inhibitors That Prevent Mice from Life-Threatening Infection and Brain Damage von Coluccia, Antonio, Puxeddu, Michela, Nalli, Marianna, Wei, Chih-Ku, Wu, Yu-Hsuan, Mastrangelo, Eloise, Elamin, Tasneem, Tarantino, Delia, Bugert, Joachim Jakob, Schreiner, Benno, Nolte, Juliane, Schwarze, Frank, La Regina, Giuseppe, Lee, Jin-Ching, Silvestri, Romano

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