Targeting the deubiquitinase USP7 for degradation with PROTACs von Murgai, Arunima, Sosi, Izidor, Gobec, Martina, Lemnitzer, Patricia, Proj, Matic, Wittenburg, Sophie, Voget, Rabea, Gütschow, Michael, Krönke, Jan, Steinebach, Christian

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Synthesis and biochemical evaluation of new 3-amido-4-substituted monocyclic ß-lactams as inhibitors of penicillin-binding protein(s) von Grabrijan, Katarina, Benedik, Nika Strašek, Krajnc, Alen, Bozovičar, Krištof, Knez, Damijan, Proj, Matic, Zdovc, Irena, Sosič, Izidor, Contreras-Martel, Carlos, Dessen, Andréa, Rambaher, Martina Hrast, Gobec, Stanislav

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Discovery of a fragment hit compound targeting D-Ala:D-Ala ligase of bacterial peptidoglycan biosynthesis von Proj, Matic, Hrast, Martina, Bajc, Gregor, Frlan, Rok, Meden, Anže, Butala, Matej, Gobec, Stanislav

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Boosting the Impact of EFMC Young Scientists Network Through the Creation of Working Groups von Mari, Michele, Lanthier, Caroline, Proj, Matic, Donckele, Etienne J., Josa‐Culleré, Laia, Goncharenko, Kristina, Leroy, Salomé, Matagne, Brieuc, McKenna, Sean M., Borsari, Chiara

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Synthesis and Biochemical Evaluation of Warhead-Decorated Psoralens as (Immuno)Proteasome Inhibitors von Schiffrer, Eva Shannon, Proj, Matic, Gobec, Martina, Rejc, Luka, Sterman, Andrej, Mravljak, Janez, Gobec, Stanislav, Sosic, Izidor

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Andrographolide Derivatives Target the KEAP1/NRF2 Axis and Possess Potent Anti‐SARS‐CoV‐2 Activity von Schulte, Bianca, König, Maria, Escher, Beate I., Wittenburg, Sophie, Proj, Matic, Wolf, Valentina, Lemke, Carina, Schnakenburg, Gregor, Sosič, Izidor, Streeck, Hendrik, Müller, Christa E., Gütschow, Michael, Steinebach, Christian

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Discovery of Immunoproteasome Inhibitors Using Large-Scale Covalent Virtual Screening von Scarpino, Andrea, Bajusz, Dávid, Proj, Matic, Gobec, Martina, Sosič, Izidor, Gobec, Stanislav, Ferenczy, György G, Keserű, György M

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Discovery of compounds with viscosity-reducing effects on biopharmaceutical formulations with monoclonal antibodies von Proj, Matic, Zidar, Mitja, Lebar, Blaž, Strašek, Nika, Miličić, Goran, Žula, Aleš, Gobec, Stanislav

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Encoding BRAF inhibitor functions in protein degraders von Miller, Daniel S. J, Voell, Sabine A, Sosi, Izidor, Proj, Matic, Rossanese, Olivia W, Schnakenburg, Gregor, Gütschow, Michael, Collins, Ian, Steinebach, Christian

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A Set of Experimentally Validated Decoys for the Human CC Chemokine Receptor 7 (CCR7) Obtained by Virtual Screening von Proj, Matic, De Jonghe, Steven, Van Loy, Tom, Jukič, Marko, Meden, Anže, Ciber, Luka, Podlipnik, Črtomir, Grošelj, Uroš, Konc, Janez, Schols, Dominique, Gobec, Stanislav

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Towards discovery of inhibitors of the undecaprenyl-pyrophosphate phosphatase BacA by virtual high-throughput screening von Jukič, Marko, Auger, Rodolphe, Folcher, Victor, Proj, Matic, Barreteau, Hélène, Gobec, Stanislav, Touzé, Thierry

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New inhibitors of cathepsin V impair tumor cell proliferation and elastin degradation and increase immune cell cytotoxicity von Mitrović, Ana, Senjor, Emanuela, Jukić, Marko, Bolčina, Lara, Prunk, Mateja, Proj, Matic, Nanut, Milica Perišić, Gobec, Stanislav, Kos, Janko

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Virtual Screening and Biochemical Testing of Borocycles as Immunoproteasome Inhibitors von Kollar, Levente, Frenczy, Gyorgy Gabor, Proj, Matic, Gobec, Martina, Gobec, Stanislav, Sosi, Izidor, Keser, Gyorgy Miklos

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Fragment-Sized and Bidentate (Immuno)Proteasome Inhibitors Derived from Cysteine and Threonine Targeting Warheads von Kollar, Levente, Gobec, Martina, Proj, Matic, Smrdel, Lara, Knez, Damijan, Imre, Timea, Gomory, Agnes, Petri, Laszlo, Abranyi-Balogh, Peter, Csanyi, Dorottya, Ferenczy, Gyoergy G., Gobec, Stanislav, Sosic, Izidor, Keseru, Gyoergy M.

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Redox active or thiol reactive? Optimization of rapid screens to identify less evident nuisance compounds von Proj, Matic, Knez, Damijan, Sosič, Izidor, Gobec, Stanislav

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Synthesis and NMR spectroscopic assignment of chlorinated benzimidazole-2-thione derivatives von Proj, Matic, Sosič, Izidor, Gobec, Stanislav

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Tunable Heteroaromatic Nitriles for Selective Bioorthogonal Click Reaction with Cysteine von Proj, Matic, Strašek, Nika, Pajk, Stane, Knez, Damijan, Sosič, Izidor

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DNA-encoded library screening on two validated enzymes of the peptidoglycan biosynthetic pathway von Proj, Matic, Bozovičar, Krištof, Hrast, Martina, Frlan, Rok, Gobec, Stanislav

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Optimization of triazolo[4,5-d]pyrimidines towards human CC chemokine receptor 7 (CCR7) antagonists von Van Hoof, Max, Claes, Sandra, Proj, Matic, Van Loy, Tom, Schols, Dominique, Gobec, Stanislav, Dehaen, Wim, De Jonghe, Steven

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Optimization of triazolo[4,5-d]pyrimidines towards human CC chemokine receptor 7 (CCR7) antagonists von Van Hoof, Max, Claes, Sandra, Proj, Matic, Van Loy, Tom, Schols, Dominique, Gobec, Stanislav, Dehaen, Wim, De Jonghe, Steven

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