(+)-and (−)-Phenazocine enantiomers: Evaluation of their dual opioid agonist/σ1 antagonist properties and antinociceptive effects von Prezzavento, O., Arena, E., Sánchez-Fernández, C., Turnaturi, R., Parenti, C., Marrazzo, A., Catalano, R., Amata, E., Pasquinucci, L., Cobos, E.J.

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Design and Synthesis of New Bifunctional Sigma‑1 Selective Ligands with Antioxidant Activity von Prezzavento, O, Arena, E, Parenti, C, Pasquinucci, L, Aricò, G, Scoto, G. M, Grancara, S, Toninello, A, Ronsisvalle, S

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(2S)-N-2-methoxy-2-phenylethyl-6,7-benzomorphan compound (2S-LP2): Discovery of a biased mu/delta opioid receptor agonist von Pasquinucci, Lorella, Turnaturi, Rita, Calò, Girolamo, Pappalardo, Francesco, Ferrari, Federica, Russo, Giulia, Arena, Emanuela, Montenegro, Lucia, Chiechio, Santina, Prezzavento, Orazio, Parenti, Carmela

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The benzomorphan-based LP1 ligand is a suitable MOR/DOR agonist for chronic pain treatment von Pasquinucci, Lorella, Parenti, Carmela, Turnaturi, Rita, Aricò, Giuseppina, Marrazzo, Agostino, Prezzavento, Orazio, Ronsisvalle, Simone, Georgoussi, Zafiroula, Fourla, Danai-Dionysia, Scoto, Giovanna M., Ronsisvalle, Giuseppe

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Effects of a Selective Sigma 1 Antagonist Compound on Inflammatory Pain von Parenti, Carmela, Marrazzo, Agostino, Aricò, Giuseppina, Cantarella, Giuseppina, Prezzavento, Orazio, Ronsisvalle, Simone, Scoto, Giovanna Maria, Ronsisvalle, Giuseppe

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New benzomorphan derivatives of MPCB as MOP and KOP receptor ligands von Pasquinucci, L., Iadanza, M., Marrazzo, A., Prezzavento, O., Ronsisvalle, S., Scoto, G. M., Parenti, C., De Luca, L., Ronsisvalle, G.

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Novel Sigma Receptor Ligands:  Synthesis and Biological Profile von Prezzavento, Orazio, Campisi, Agata, Ronsisvalle, Simone, Li Volti, Giovanni, Marrazzo, Agostino, Bramanti, Vincenzo, Cannavò, Giuseppe, Vanella, Luca, Cagnotto, Alfredo, Mennini, Tiziana, Ientile, Riccardo, Ronsisvalle, Giuseppe

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Nonpeptide Analogues of Dynorphin A(1−8):  Design, Synthesis, and Pharmacological Evaluation of κ-Selective Agonists von Ronsisvalle, Giuseppe, Pasquinucci, Lorella, Pittalà, Valeria, Marrazzo, Agostino, Prezzavento, Orazio, Di Toro, Rosanna, Falcucci, Barbara, Spampinato, Santi

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(+)-and (-)-Phenazocine enantiomers: Evaluation of their dual opioid agonist/σ 1 antagonist properties and antinociceptive effects von Prezzavento, O, Arena, E, Sánchez-Fernández, C, Turnaturi, R, Parenti, C, Marrazzo, A, Catalano, R, Amata, E, Pasquinucci, L, Cobos, E J

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Synthesis and Structure−Activity Relationships of 1-Aralkyl-4-Benzylpiperidine and 1-Aralkyl-4-Benzylpiperazine Derivatives as Potent σ Ligands von Costantino, Luca, Gandolfi, Francesca, Sorbi, Claudia, Franchini, Silvia, Prezzavento, Orazio, Vittorio, Franco, Ronsisvalle, Giuseppe, Leonardi, Amedeo, Poggesi, Elena, Brasili, Livio

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Synthesis and anti-measles virus activity of new isoquinolin-4-one derivatives von Santagati, N.A, Bousquet, E, Garozzo, A, Prezzavento, O, Spadaro, A, Ronsisvalle, G

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Intrastriatal administration of sigma ligands inhibits basal dopamine release in vivo von Moison, Delphine, De Deurwaerdère, Philippe, Cagnotto, Alfredo, Marrazzo, Agostino, Prezzavento, Orazio, Ronsisvalle, Giuseppe, Mennini, Tiziana, Spampinato, Umberto

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Opioid and sigma receptor studies. New developments in the design of selective sigma ligands von Ronsisvalle, Giuseppe, Marrazzo, Agostino, Prezzavento, Orazio, Cagnotto, Alfredo, Mennini, Tiziana, Parenti, Carmela, Scoto, Giovanna M.

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CCB, a novel specific κ opioid agonist, which discriminates between opioid and σ 1 recognition sites von Ronsisvalle, G., Prezzavento, O., Pasquinucci, L., Marrazzo, A., Vittorio, F., Gomez-Vidal, J.A., Carboni, L., Spampinato, S.

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CCB: A novel anologue of MPCB with high binding affinity and specific kappa opioid receptor agonist von Ronsisvalle, G, Prezzavento, O, Pasquinucci, L, Carboni, L, Pistacchio, E, Spampinato, S

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Synthesis of (+)-cis-N-(4-isothiocyanatobenzyl)-N-normetazocine, an isothiocyanate derivative of N-benzylnormetazocine as acylant agent for the sigma(1) receptor von Ronsisvalle, Giuseppe, Prezzavento, Orazio, Marrazzo, Agostino, Vittorio, Franco, Massimino, Michele, Murari, Giovanna, Spampinato, Santi

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Synthesis and spasmolytic action of 2-substituted thienopyrimidin-4-one derivatives von Santagati, Natale Alfredo, Prezzavento, Orazio, Bousquet, Ennio, Ronsisvalle, Giuseppe, Spampinato, Santi

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1-Phenyl-3-azabicyclo[3.1.0]hexane derivatives as new ligands for sigma receptors von Marrazzo, Agostino, Pappalardo, Andrea, Prezzavento, Orazio, Vittorio, Franco

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Substituted 1-phenyl-2-cyclopropylmethylamines with high affinity and selectivity for sigma sites von RONSISVALLE, G, MARRAZZO, A, PREZZAVENTO, O, PASQUINUCCI, L, FALCUCCI, B, DI TORO, R, SPAMPINATO, S

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Synthesis and binding affinity of cis-(-)- and cis-(+)-N-ethyleneamino-N-nordeoxymetazocine and cis-(-)-N-normetazocine analogues at sigma1, sigma2 and kappa opioid receptors von Ronsisvalle, G, Prezzavento, O, Marrazzo, A, Vittorio, F, Bousquet, E, Di Toro, R, Spampinato, S

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