Biased signaling due to oligomerization of the G protein-coupled platelet-activating factor receptor von Liu, Junke, Tang, Hengmin, Xu, Chanjuan, Zhou, Shengnan, Zhu, Xunying, Li, Yuanyuan, Prézeau, Laurent, Xu, Tao, Pin, Jean-Philippe, Rondard, Philippe, Ji, Wei, Liu, Jianfeng

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Design, Synthesis, Pharmacology, and In Silico Studies of (1S,2S,3S)‑2-((S)‑Amino(carboxy)methyl)-3-(carboxymethyl)cyclopropane-1-carboxylic Acid (LBG30300): A Picomolar Potency Su... von Liu, Na, Eshak, Floriane, Malhaire, Fanny, Brabet, Isabelle, Prézeau, Laurent, Renard, Emma, Pin, Jean-Philippe, Acher, Francine C., Staudt, Markus, Bunch, Lennart

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Dimers and beyond: The functional puzzles of class C GPCRs von Kniazeff, Julie, Prézeau, Laurent, Rondard, Philippe, Pin, Jean-Philippe, Goudet, Cyril

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GPCR interaction as a possible way for allosteric control between receptors von Pin, Jean-Philippe, Kniazeff, Julie, Prézeau, Laurent, Liu, Jiang-Feng, Rondard, Philippe

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The urotensin II receptor triggers an early meningeal response and a delayed macrophage-dependent vasospasm after subarachnoid hemorrhage in male mice von Pedard, Martin, Prevost, Lucie, Carpena, Camille, Holleran, Brian, Desrues, Laurence, Dubois, Martine, Nicola, Celeste, Gruel, Roxane, Godefroy, David, Deffieux, Thomas, Tanter, Mickael, Ali, Carine, Leduc, Richard, Prézeau, Laurent, Gandolfo, Pierrick, Morin, Fabrice, Wurtz, Olivier, Bonnard, Thomas, Vivien, Denis, Castel, Hélène

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Pharmacological evidence for a metabotropic glutamate receptor heterodimer in neuronal cells von Moreno Delgado, David, Møller, Thor C, Ster, Jeanne, Giraldo, Jesús, Maurel, Damien, Rovira, Xavier, Scholler, Pauline, Zwier, Jurriaan M, Perroy, Julie, Durroux, Thierry, Trinquet, Eric, Prezeau, Laurent, Rondard, Philippe, Pin, Jean-Philippe

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Synthesis and pharmacological characterization of conformationally restricted 2-amino-Adipic acid analogs and carboxycyclopropyl glycines as selective metabotropic glutamate 2 rece... von Staudt, Markus, Liu, Na, Malhaire, Fanny, Doroudian, Yasaman, Prézeau, Laurent, Renard, Emma, Hasanpour, Zahra, Pin, Jean-Philippe, Bunch, Lennart

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A nanobody activating metabotropic glutamate receptor 4 discriminates between homo- and heterodimers von Haubrich, Jordi, Font, Joan, Quast, Robert B, Goupil-Lamy, Anne, Scholler, Pauline, Nevoltris, Damien, Acher, Francine, Chames, Patrick, Rondard, Philippe, Prézeau, Laurent, Pin, Jean-Philippe

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Biased signaling regulates the pleiotropic effects of the urotensin II receptor to modulate its cellular behaviors von Brulé, Cédric, Perzo, Nicolas, Joubert, Jane‐Eileen, Sainsily, Xavier, Leduc, Richard, Castel, Hélène, Prézeau, Laurent

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Different EGF‐induced receptor dimer conformations for signaling and internalization von Haubrich, Jordi, Zwier, Jurriaan M., Charrier‐Savournin, Fabienne, Prézeau, Laurent, Pin, Jean‐Philippe

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Cell-surface protein-protein interaction analysis with time-resolved FRET and snap-tag technologies: application to GPCR oligomerization von Maurel, Damien, Comps-Agrar, Laëtitia, Brock, Carsten, Rives, Marie-Laure, Bourrier, Emmanuel, Ayoub, Mohammed Akli, Bazin, Hervé, Tinel, Norbert, Durroux, Thierry, Prézeau, Laurent, Trinquet, Eric, Pin, Jean-Philippe

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G protein‐coupled receptors can control the Hippo/YAP pathway through Gq signaling von Zindel, Diana, Mensat, Patrick, Vol, Claire, Homayed, Zeinab, Charrier‐Savournin, Fabienne, Trinquet, Eric, Banères, Jean‐Louis, Pin, Jean‐Philippe, Pannequin, Julie, Roux, Thomas, Dupuis, Elodie, Prézeau, Laurent

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Evolution, structure, and activation mechanism of family 3/C G-protein-coupled receptors von Pin, Jean-Philippe, Galvez, Thierry, Prézeau, Laurent

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The chemokine CXC4 and CC2 receptors form homo‐ and heterooligomers that can engage their signaling G‐protein effectors and βarrestin von Armando, Sylvain, Quoyer, Julie, Lukashova, Viktorya, Maiga, Arhamatoulaye, Percherancier, Yann, Heveker, Nikolaus, Pin, Jean‐Philippe, Prézeau, Laurent, Bouvier, Michel

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Closed state of both binding domains of homodimeric mGlu receptors is required for full activity von Kniazeff, Julie, Bessis, Anne-Sophie, Maurel, Damien, Ansanay, Hervé, Prézeau, Laurent, Pin, Jean-Philippe

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Nonclassical Ligand-Independent Regulation of Go Protein by an Orphan Class C G-Protein–Coupled Receptor von Hajj, Mariana, De Vita, Teresa, Vol, Claire, Renassia, Charlotte, Bologna, Jean-Charles, Brabet, Isabelle, Cazade, Magali, Pastore, Manuela, Blahos, Jaroslav, Labesse, Gilles, Pin, Jean-Philippe, Prézeau, Laurent

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The complexity of their activation mechanism opens new possibilities for the modulation of mGlu and GABAB class C G protein-coupled receptors von Rondard, Philippe, Goudet, Cyril, Kniazeff, Julie, Pin, Jean-Philippe, Prézeau, Laurent

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Quantitative Phosphoproteomics Unravels Biased Phosphorylation of Serotonin 2A Receptor at Ser280 by Hallucinogenic versus Nonhallucinogenic Agonists von Karaki, Samah, Becamel, Carine, Murat, Samy, Mannoury la Cour, Clotilde, Millan, Mark J., Prézeau, Laurent, Bockaert, Joël, Marin, Philippe, Vandermoere, Franck

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Oligomerization of a G protein-coupled receptor in neurons controlled by its structural dynamics von Møller, Thor C., Hottin, Jerome, Clerté, Caroline, Zwier, Jurriaan M., Durroux, Thierry, Rondard, Philippe, Prézeau, Laurent, Royer, Catherine A., Pin, Jean-Philippe, Margeat, Emmanuel, Kniazeff, Julie

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The Heptahelical Domain of GABAB2 Is Activated Directly by CGP7930, a Positive Allosteric Modulator of the GABAB Receptor von Virginie Binet, Carole Brajon, Laurent Le Corre, Francine Acher, Jean-Philippe Pin, Laurent Prézeau

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