Novel Derivatives of Eugenol as a New Class of PPARγ Agonists in Treating Inflammation: Design, Synthesis, SAR Analysis and In Vitro Anti-Inflammatory Activity von Anjum, Noor Fathima, Shanmugarajan, Dhivya, Prashantha Kumar, B R, Faizan, Syed, Durai, Priya, Raju, Ruby Mariam, Javid, Saleem, Purohit, Madhusudan N

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Curcumin to inhibit binding of spike glycoprotein to ACE2 receptors: computational modelling, simulations, and ADMET studies to explore curcuminoids against novel SARS-CoV-2 target... von Shanmugarajan, Dhivya, Kumar, B. R. Prashantha, Suresh, B

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Enantioselective Separation and Pharmacokinetics of a Chiral 1,4‐Dihydropyrimidine Derivative in Rats: A Combined Chromatography and Docking Approach von Sri, Chiriki Devi, Faizan, Syed, Chandra, Muttavarapu Rohit, Kumar, B. R. Prashantha, Gurupadayya, B. M.

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Novel Biginelli dihydropyrimidines with potential anticancer activity: A parallel synthesis and CoMSIA study von Prashantha Kumar, B.R., Sankar, Gopu, Nasir Baig, R.B., Chandrashekaran, Srinivasan

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Thiazolidinediones as antidiabetic agents: A critical review von Nanjan, M.J., Mohammed, Manal, Prashantha Kumar, B.R., Chandrasekar, M.J.N.

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Development of novel thiazolidine-2,4-dione derivatives as PPAR-γ agonists through design, synthesis, computational docking, MD simulation, and comprehensive in vitro and in vivo e... von Gowdru Srinivasa, Mahendra, B C, Revanasiddappa, Prabhu, Ashwini, Rani, Vinitha, Ghate, Sudeep D, Kumar B R, Prashantha

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Discovery of Novel Myristic Acid Derivatives as N-Myristoyltransferase Inhibitors: Design, Synthesis, Analysis, Computational Studies and Antifungal Activity von Javid, Saleem, Ather, Hissana, Hani, Umme, Siddiqua, Ayesha, Asif Ansari, Shaik Mohammad, Shanmugarajan, Dhivya, Yogish Kumar, Honnavalli, Arivuselvam, Rajaguru, Purohit, Madhusudan N, Kumar, B R Prashantha

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Predicting anti-HIV activity of 1,3,4-thiazolidinone derivatives: 3D-QSAR approach von Ravichandran, V., Prashantha Kumar, B.R., Sankar, S., Agrawal, R.K.

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Minutes of PPAR-γ agonism and neuroprotection von Prashantha Kumar, B.R., Kumar, Ashwini Prem, Jose, Jincy A., Prabitha, P., Yuvaraj, S., Chipurupalli, Sandhya, Jeyarani, Victoria, Manisha, Chennu, Banerjee, Sayani, Jeyabalan, Jeyaram Bharathi, Mohankumar, Suresh Kumar, Dhanabal, S.P., Justin, Antony

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Novel glitazones as PPARγ agonists: molecular design, synthesis, glucose uptake activity and 3D QSAR studies von Mandal, Subhankar P., Garg, Aakriti, Prabitha, P., Wadhwani, Ashish D., Adhikary, Laxmi, Kumar, B. R. Prashantha

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Novel dual PPARα/γ agonists protect against liver steatosis and improve insulin sensitivity while avoiding side effects von Guru, Bhavimani, Tamrakar, Akhilesh K., Manjula, S.N., Prashantha Kumar, B.R.

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Anticancer potential of novel symmetrical and asymmetrical dihydropyridines against breast cancer via EGFR inhibition: molecular design, synthesis, analysis and screening von Faizan, Syed, Talath, Sirajunisa, Wali, Adil Farooq, Hani, Umme, Haider, Nazima, Mandal, Subhankar P, Kumar, B R Prashantha

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Isolation, Identification, and Antibacterial Properties of Prodigiosin, a Bioactive Product Produced by a New Serratia marcescens JSSCPM1 Strain: Exploring the Biosynthetic Gene Cl... von Arivuselvam, Rajaguru, Dera, Ayed A., Parween Ali, Syed, Alraey, Yasser, Saif, Ahmed, Hani, Umme, Arumugam Ramakrishnan, Sivaa, Azeeze, Mohamed Sheik Tharik Abdul, Rajeshkumar, Raman, Susil, Aishwarya, Harindranath, Haritha, Kumar, B. R. Prashantha

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A promising in silico protocol to develop novel PPARγ antagonists as potential anticancer agents: Design, synthesis and experimental validation via PPARγ protein activity and compe... von Sivamani, Yuvaraj, Shanmugarajan, Dhivya, Durai Ananda Kumar, T., Faizan, Syed, Channappa, Bhavya, Naishima, Namburu Lalitha, Prashantha Kumar, B.R.

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Novel PPAR-γ agonists as potential neuroprotective agents against Alzheimer's disease: rational design, synthesis , in silico evaluation, PPAR-γ binding assay and transactivation a... von D, Priya, Hani, Umme, Haider, Nazima, Talath, Sirajunisa, Shanmugarajan, Dhivya, P, Prabitha, P, Archana, Prashantha Kumar, B R

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Design, parallel synthesis of Biginelli 1,4-dihydropyrimidines using PTSA as a catalyst, evaluation of anticancer activity and structure activity relationships via 3D QSAR studies von Faizan, Syed, Prashantha Kumar, B.R., Lalitha Naishima, Namburu, Ashok, T., Justin, Antony, Vijay Kumar, Merugumolu, Bistuvalli Chandrashekarappa, Revanasiddappa, Manjunathaiah Raghavendra, Nulgumnalli, Kabadi, Pradeep, Adhikary, Laxmi

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Structure-based design and synthesis of new 4-methylcoumarin-based lignans as pro-inflammatory cytokines (TNF-α, IL-6 and IL-1β) inhibitors von Santhosh Kumar, S., Sajeli Begum, Ahil, Hira, Kirti, Niazi, Sarfaraj, Prashantha Kumar, B.R., Araya, Hiroshi, Fujimoto, Yoshinori

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Rational Design, Synthesis, and In Vitro Neuroprotective Evaluation of Novel Glitazones for PGC-1α Activation via PPAR-γ: a New Therapeutic Strategy for Neurodegenerative Disorders... von Justin, Antony, Mandal, Subhankar, Prabitha, P., Dhivya, S., Yuvaraj, S., Kabadi, Pradeep, Sekhar, Satheesh John, Sandhya, C. H., Wadhwani, Ashish D., Divakar, Selvaraj, Bharathi, Jeyabalan Jeyaram, Durai, Priya, Prashantha Kumar, B. R.

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Design, synthesis and glucose uptake activity of some novel glitazones von Kar, Koyel, Krithika, Uma, Mithuna, Basu, Prabhuddha, Santhosh Kumar, S., Reji, Anu, Prashantha Kumar, B.R.

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Biphenyl-based small molecule inhibitors: Novel cancer immunotherapeutic agents targeting PD-1/PD-L1 interaction von Sasmal, Pujan, Kumar Babasahib, Sajeev, Prashantha Kumar, B.R., Manjunathaiah Raghavendra, Nulgumnalli

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