Thienothiopyran-2-sulfonamides: novel topically active carbonic anhydrase inhibitors for the treatment of glaucoma von Baldwin, John J, Ponticello, Gerald S, Anderson, Paul S, Christy, Marcia E, Murcko, Mark A, Randall, William C, Schwam, Harvey, Sugrue, Michael F, Gautheron, Pierre

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Identification and SAR for a selective, nonpeptidyl thrombin inhibitor von Naylor-Olsen, Adel M., Ponticello, Gerald S., Lewis, S.Dale, Mulichak, Anne M., Chen, Zhonguo, Habecker, Charles N., Phillips, Brian T., Sanders, William M., Tucker, Thomas J., Shafer, Jules A., Vacca, Joseph P.

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Thienothiopyran-2-sulfonamides: a novel class of water-soluble carbonic anhydrase inhibitors von Ponticello, Gerald S, Freedman, Mark B, Habecker, Charles N, Lyle, Paulette A, Schwam, Harvey, Varga, Sandor L, Christy, Marcia E, Randall, William C, Baldwin, John J

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A comparison of L-671,152 and MK-927, two topically effective ocular hypotensive carbonic anhydrase inhibitors, in experimental animals von Sugrue, M. F., Mallorga, P., Schwam, H., Baldwin, J. J., Ponticello, G. S.

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On the use of the O-methylmandelate ester for establishment of absolute configuration of secondary alcohols von Trost, Barry M, Belletire, John L, Godleski, Stephen, McDougal, Patrick G, Balkovec, James M, Baldwin, John J, Christy, Marcia E, Ponticello, Gerald S, Varga, Sandor L, Springer, James P

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Positions of His‐64 and a bound water in human carbonic anhydrase II upon binding three structurally related inhibitors von Smith, Graham M., Alexander, Richard S, Christianson, David W., Mckeever, Brian M., Ponticello, Gerald S., Springer, James P., Randall, William C., Baldwin, John J., Habecker, Charles N.

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MK-927: A Topically Active Ocular Hypotensive Carbonic Anhydrase Inhibitor von SUGRUE, M.F., GAUTHERON, P., GROVE, J., MALLORGA, P., VIADER, M.P., SCHWAM, H., BALDWIN, J.J., CHRISTY, M.E., PONTICELLO, G.S.

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L-653,328: an ocular hypotensive agent with modest beta receptor blocking activity von Sugrue, MF, Gautheron, P, Grove, J, Mallorga, P, Viader, MP, Baldwin, JJ, Ponticello, GS, Varga, SL

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A short radiosynthesis of 6-[C3H3]-dorzolamide at very high specific activity and optical purity von Eng, W.-s., Burns, H. D., Ponticello, G. S., Selnick, H. G.

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2-Pyridylimidazoles as inhibitors of xanthine oxidase von Baldwin, J. J, Lumma, P. K, Novello, F. C, Ponticello, G. S, Sprague, J. M, Duggan, D. E

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beta.-Adrenergic blocking agents with acute antihypertensive activity von Baldwin, J. J, Engelhardt, E. L, Hirschmann, R, Lundell, G. F, Ponticello, G. S, Ludden, C. T, Sweet, C. S, Scriabine, A, Share, N. N, Hall, R

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A novel naphthyridinone synthesis via enamine cyclization von Baldwin, J. J, Mensler, K, Ponticello, G. S

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An approach to peripheral vasodilator-.beta.-adrenergic blocking agents von Baldwin, J. J, Hirschmann, R, Lumma, P. K, Lumma, W. C, Ponticello, G. S, Sweet, C. S, Scriabine, A

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Preparative methods for ergoline synthons: Uhle's ketone and the C-homo analog von Ponticello, G. S, Baldwin, J. J, Lumma, P. K, McClure, D. E

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Preclinical studies on L-671,152, a topically effective ocular hypotensive carbonic anhydrase inhibitor von Sugrue, M F, Mallorga, P, Schwam, H, Baldwin, J J, Ponticello, G S

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The synthesis of dihydrothieno[2,3-b]thiophenes by a metal-halogen exchange initiated intramolecular acylation von Selnick, Harold G., Radzilowski, Ellen M., Ponticello, Gerald S.

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An unusual dimer of 2-mercaptothiophene von Ponticello, Gerald S, Habecker, Charles N, Varga, Sandor L, Pitzenberger, Steven M

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Utilization of .alpha.,.beta.-unsaturated acids as Michael acceptors for the synthesis of thieno[2,3-b]thiopyrans von Ponticello, Gerald S, Freedman, Mark B, Habecker, Charles N, Holloway, M. Katharine, Amato, Joseph S, Conn, Robin S, Baldwin, John J

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Heterocyclic analogs of the antihypertensive .beta.-adrenergic blocking agent (S)-2-[3-(tert-butylamino)-2-hydroxypropoxy]-3-cyanopyridine von Baldwin, John J, Engelhardt, Edward L, Hirschmann, Ralph, Ponticello, Gerald S, Atkinson, Joseph G, Wasson, Burton K, Sweet, Charles S, Scriabine, Alexander

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Beta 1-selective adrenoceptor antagonists: examples of the 2-[4-[3-(substituted amino)-2-hydroxypropoxy]phenyl]imidazole class. 2 von Baldwin, J J, Christy, M E, Denny, G H, Habecker, C N, Freedman, M B, Lyle, P A, Ponticello, G S, Varga, S L, Gross, D M, Sweet, C S

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