Peptidyl Acyloxymethyl Ketones as Activity‐Based Probes for the Main Protease of SARS‐CoV‐2 von Plassche, Merel A. T., Barniol‐Xicota, Marta, Verhelst, Steven H. L.

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Rapid synthesis of internal peptidyl α-ketoamides by on resin oxidation for the construction of rhomboid protease inhibitors von Van Kersavond, Tim, Konopatzki, Raphael, van der Plassche, Merel A. T, Yang, Jian, Verhelst, Steven H. L

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Correction: Rapid synthesis of internal peptidyl α-ketoamides by on resin oxidation for the construction of rhomboid protease inhibitors von Van Kersavond, Tim, Konopatzki, Raphael, van der Plassche, Merel A. T, Yang, Jian, Verhelst, Steven H. L

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Rapid Solid-Phase Construction of Serine Hydrolase Probes Results in Selective Activity-Based Probes for Acyl Protein Thioesterases-1/2 von Vanhoutte, Roeland, van de Plassche, Merel A. T, Verhelst, Steven H. L

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Use of Non-Natural Amino Acids for the Design and Synthesis of a Selective, Cell-Permeable MALT1 Activity-Based Probe von van de Plassche, Merel A. T, O’Neill, Thomas J, Seeholzer, Thomas, Turk, Boris, Krappmann, Daniel, Verhelst, Steven H. L

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Facile Synthesis of Aminomethyl Phosphinate Esters as Serine Protease Inhibitors with Primed Site Interaction von Kahler, Jan Pascal, Lenders, Stijn, van de Plassche, Merel A. T, Verhelst, Steven H. L

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A Lysosome-Targeted Tetrazine for Organelle-Specific Click-to-Release Chemistry in Antigen Presenting Cells von Ligthart, Nina A.M., de Geus, Mark A.R., van de Plassche, Merel A.T., Torres García, Diana, Isendoorn, Marjolein M.E., Reinalda, Luuk, Ofman, Daniëlle, van Leeuwen, Tyrza, van Kasteren, Sander I.

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Front Cover: Peptidyl Acyloxymethyl Ketones as Activity‐Based Probes for the Main Protease of SARS‐CoV‐2 (ChemBioChem 23/2020) von Plassche, Merel A. T., Barniol‐Xicota, Marta, Verhelst, Steven H. L.

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Recent Advances in Activity-Based Protein Profiling of Proteases von Chakrabarty, Suravi, Kahler, Jan Pascal, van de Plassche, Merel A. T., Vanhoutte, Roeland, Verhelst, Steven H. L.

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Methyltetrazine as a small live-cell compatible bioorthogonal handle for imaging enzyme activities in situ von Torres-García, Diana, van de Plassche, Merel A. T., van Boven, Emma, van Leeuwen, Tyrza, Groenewold, Mirjam G. J., Sarris, Alexi J. C., Klein, Luuk, Overkleeft, Herman S., van Kasteren, Sander I.

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Methyltetrazine as a small live-cell compatible bioorthogonal handle for imaging enzyme activities von Torres-García, Diana, van de Plassche, Merel A. T, van Boven, Emma, van Leeuwen, Tyrza, Groenewold, Mirjam G. J, Sarris, Alexi J. C, Klein, Luuk, Overkleeft, Herman S, van Kasteren, Sander I

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Live‐Cell Imaging of Sterculic Acid—a Naturally Occurring 1,2‐Cyclopropene Fatty Acid—by Bioorthogonal Reaction with Turn‐On Tetrazine‐Fluorophore Conjugates von Bertheussen, Kristine, Plassche, Merel, Bakkum, Thomas, Gagestein, Berend, Ttofi, Iakovia, Sarris, Alexi J. C., Overkleeft, Herman S., Stelt, Mario, Kasteren, Sander I.

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Rapid Solid-Phase Construction of Serine Hydrolase Probes Results in Selective Activity-Based Probes for Acyl Protein Thioesterases-1/2 von Vanhoutte, Roeland, van de Plassche, Merel A.T, Verhelst, Steven H.L

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Live‐Cell Imaging of Sterculic Acid—a Naturally Occurring 1,2‐Cyclopropene Fatty Acid—by Bioorthogonal Reaction with Turn‐On Tetrazine‐Fluorophore Conjugates von Bertheussen, Kristine, Plassche, Merel, Bakkum, Thomas, Gagestein, Berend, Ttofi, Iakovia, Sarris, Alexi J. C., Overkleeft, Herman S., Stelt, Mario, Kasteren, Sander I.

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Peptidyl Acyloxymethyl Ketones as Activity-Based Probes for the Main Protease of SARS-CoV-2 von van de Plassche, Merel A.T, Barniol-Xicota, Marta, Verhelst, Steven H.L

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Rapid synthesis of internal peptidyl α-ketoamides by on resin oxidation for the construction of rhomboid protease inhibitors von Van Kersavond, Tim, Konopatzki, Raphael, van der Plassche, Merel A.T, Yang, Jian, Verhelst, Steven H.L

Volltext

Use of Non-Natural Amino Acids for the Design and Synthesis of a Selective, Cell-Permeable MALT1 Activity-Based Probe von van de Plassche, Merel A.T, O'Neill, Thomas J, Seeholzer, Thomas, Turk, Boris, Krappmann, Daniel, Verhelst, Steven H.L

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Recent Advances in Activity-Based Protein Profiling of Proteases von Chakrabarty, Suravi, Kahler, Jan Pascal, van de Plassche, Merel A.T, Vanhoutte, Roeland, Verhelst, Steven H.L

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Facile Synthesis of Aminomethyl Phosphinate Esters as Serine Protease Inhibitors with Primed Site Interaction von Kahler, Jan Pascal, Lenders, Stijn, van de Plassche, Merel A.T, Verhelst, Steven H.L

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4‑Oxo-β-lactams as Covalent Inhibitors of the Mitochondrial Intramembrane Protease PARL von Ji, Shanping, Bach, Kathrin, Miriyala, Vijay Madhav, Dohnálek, Jan, Riopedre-Fernandez, Miguel, Lepšík, Martin, van de Plassche, Merel, Vanhoutte, Roeland, Barniol-Xicota, Marta, Moreira, Rui, Strisovsky, Kvido, Verhelst, Steven H. L.

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