Enantioselective Total Synthesis of (−)-Minovincine in Nine Chemical Steps: An Approach to Ketone Activation in Cascade Catalysis von Laforteza, Brian N., Pickworth, Mark, MacMillan, David W. C.

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A Practical Flow Reactor for Continuous Organic Photochemistry von Hook, Benjamin D. A, Dohle, Wolfgang, Hirst, Paul R, Pickworth, Mark, Berry, Malcolm B, Booker-Milburn, Kevin I

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Asymmetric Decarboxylative Allylation of Oxindoles von Franckevičius, Vilius, Cuthbertson, James D, Pickworth, Mark, Pugh, David S, Taylor, Richard J. K

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Helix Persistence and Breakdown in Oligoureas of Metaphenylenediamine: Apparent Diastereotopicity as a Spectroscopic Marker of Helix Length in Solution von Clayden, Jonathan, Lemiègre, Loïc, Morris, Gareth A, Pickworth, Mark, Snape, Timothy J, Jones, Lyn H

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Relaying stereochemistry through aromatic ureas: 1,9 and 1,15 remote stereocontrol von Clayden, Jonathan, Pickworth, Mark, Jones, Lyn H

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Conformation and stereodynamics of 2,2'-disubstituted N,N'-diaryl ureas von Clayden, Jonathan, Lemiègre, Loïc, Pickworth, Mark, Jones, Lyn

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Slow interconversion of enantiomeric conformers or atropisomers of anilide and urea derivatives of 2-substituted anilines von Adler, Thomas, Bonjoch, Josep, Clayden, Jonathan, Font-Bardía, Mercè, Pickworth, Mark, Solans, Xavier, Solé, Daniel, Vallverdú, Lluís

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From structure to clinic: Design of a muscarinic M1 receptor agonist with potential to treatment of Alzheimer's disease von Brown, Alastair J H, Bradley, Sophie J, Marshall, Fiona H, Brown, Giles A, Bennett, Kirstie A, Brown, Jason, Cansfield, Julie E, Cross, David M, de Graaf, Chris, Hudson, Brian D, Dwomoh, Louis, Dias, João M, Errey, James C, Hurrell, Edward, Liptrot, Jan, Mattedi, Giulio, Molloy, Colin, Nathan, Pradeep J, Okrasa, Krzysztof, Osborne, Greg, Patel, Jayesh C, Pickworth, Mark, Robertson, Nathan, Shahabi, Shahram, Bundgaard, Christoffer, Phillips, Keith, Broad, Lisa M, Goonawardena, Anushka V, Morairty, Stephen R, Browning, Michael, Perini, Francesca, Dawson, Gerard R, Deakin, John F W, Smith, Robert T, Sexton, Patrick M, Warneck, Julie, Vinson, Mary, Tasker, Tim, Tehan, Benjamin G, Teobald, Barry, Christopoulos, Arthur, Langmead, Christopher J, Jazayeri, Ali, Cooke, Robert M, Rucktooa, Prakash, Congreve, Miles S, Weir, Malcolm, Tobin, Andrew B

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Structure-Based Drug Discovery of N‑((R)‑3-(7-Methyl‑1H‑indazol-5-yl)-1-oxo-1-(((S)‑1-oxo-3-(piperidin-4-yl)-1-(4-(pyridin-4-yl)piperazin-1-yl)propan-2-yl)amino)propan-2-yl)-2′-oxo... von Bucknell, Sarah J, Ator, Mark A, Brown, Alastair J. H, Brown, Jason, Cansfield, Andrew D, Cansfield, Julie E, Christopher, John A, Congreve, Miles, Cseke, Gabriella, Deflorian, Francesca, Jones, Christopher R, Mason, Jonathan S, O’Brien, M. Alistair, Ott, Gregory R, Pickworth, Mark, Southall, Stacey M

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From structure to clinic: Design of a muscarinic M1 receptor agonist with the potential to treat Alzheimer’s disease von Brown, Alastair J.H., Bradley, Sophie J., Marshall, Fiona H., Brown, Giles A., Bennett, Kirstie A., Brown, Jason, Cansfield, Julie E., Cross, David M., de Graaf, Chris, Hudson, Brian D., Dwomoh, Louis, Dias, João M., Errey, James C., Hurrell, Edward, Liptrot, Jan, Mattedi, Giulio, Molloy, Colin, Nathan, Pradeep J., Okrasa, Krzysztof, Osborne, Greg, Patel, Jayesh C., Pickworth, Mark, Robertson, Nathan, Shahabi, Shahram, Bundgaard, Christoffer, Phillips, Keith, Broad, Lisa M., Goonawardena, Anushka V., Morairty, Stephen R., Browning, Michael, Perini, Francesca, Dawson, Gerard R., Deakin, John F.W., Smith, Robert T., Sexton, Patrick M., Warneck, Julie, Vinson, Mary, Tasker, Tim, Tehan, Benjamin G., Teobald, Barry, Christopoulos, Arthur, Langmead, Christopher J., Jazayeri, Ali, Cooke, Robert M., Rucktooa, Prakash, Congreve, Miles S., Weir, Malcolm, Tobin, Andrew B.

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Ring-Selective Functionalization of N,N ‘-Diarylureas by Regioselective N-Alkylation and Directed Ortho Metalation von Clayden, Jonathan, Turner, Hazel, Pickworth, Mark, Adler, Thomas

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Synthesis of enantiomerically enriched isotopically-labelled anilines by (−)-sparteine directed lithiation von Clayden, Jonathan, Lemiègre, Loïc, Pickworth, Mark

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Achieving conformational control over C-C, C-N and C-O bonds in biaryls, N,N'-diarylureas and diaryl ethers: advantages of a relay axis von Betson, Mark S, Bracegirdle, Ann, Clayden, Jonathan, Helliwell, Madeleine, Lund, Andrew, Pickworth, Mark, Snape, Timothy J, Worrall, Christopher P

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Enantioselective Total Synthesis of (−)-Minovincine in Nine Chemical Steps: An Approach to Ketone Activation in Cascade Catalysis von Laforteza, Brian N., Pickworth, Mark, MacMillan, David W. C.

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CRYSTALLINE FORMS AND SALTS OF A MUSCARINIC RECEPTOR AGONIST von PICKWORTH, Mark, MCGEE, Paul, BROWN, Giles Albert, CANSFIELD, Julie

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MUSCARINIC RECEPTOR AGONISTS von PICKWORTH, Mark, MCGEE, Paul, BROWN, Giles Albert, CANSFIELD, Julie

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Muscarinic agonists von Tehan, Benjamin Gerald, Teobald, Barry John, Cansfield, Julie, Brown, Giles Albert, Pickworth, Mark

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MUSCARINIC AGONISTS von PICKWORTH, Mark, BROWN, Giles Albert, CONGREVE, Miles Stuart, TEHAN, Benjamin Gerald

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MUSCARINIC AGONISTS von PICKWORTH, Mark, BROWN, Giles Albert, CONGREVE, Miles Stuart, TEHAN, Benjamin Gerald

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QUINOLINONE AND BENZOXAZINE DERIVATIVES AS MUSCARINIC M1 AND/OR M4 RECEPTOR AGONISTS von PICKWORTH, Mark, BROWN, Giles Albert, CONGREVE, Miles Stuart, TEHAN, Benjamin Gerald

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