Update on melatonin receptors: IUPHAR Review 20 von Jockers, Ralf, Delagrange, Philippe, Dubocovich, Margarita L., Markus, Regina P., Renault, Nicolas, Tosini, Gianluca, Cecon, Erika, Zlotos, Darius P.

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International Union of Basic and Clinical Pharmacology. LXXV. Nomenclature, classification, and pharmacology of G protein-coupled melatonin receptors von Dubocovich, Margarita L, Delagrange, Philippe, Krause, Diana N, Sugden, David, Cardinali, Daniel P, Olcese, James

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Negative regulation of melatonin secretion by melatonin receptors in ovine pinealocytes von Lepinay, Julie, Taragnat, Catherine, Dubois, Jean-Philippe, Chesneau, Didier, Jockers, Ralf, Delagrange, Philippe, Bozon, Veronique

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Mathematical modeling of the microtubule detyrosination/tyrosination cycle for cell-based drug screening design von Grignard, Jeremy, Lamamy, Véronique, Vermersch, Eva, Delagrange, Philippe, Stephan, Jean-Philippe, Dorval, Thierry, Fages, François

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GPR50-Ctail cleavage and nuclear translocation: a new signal transduction mode for G protein-coupled receptors von Ahmad, Raise, Lahuna, Olivier, Sidibe, Anissa, Daulat, Avais, Zhang, Qiang, Luka, Marine, Guillaume, Jean-Luc, Gallet, Sarah, Guillonneau, François, Hamroune, Juliette, Polo, Sophie, Prévot, Vincent, Delagrange, Philippe, Dam, Julie, Jockers, Ralf

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Convergence of Melatonin and Serotonin (5-HT) Signaling at MT2/5-HT2C Receptor Heteromers von Kamal, Maud, Gbahou, Florence, Guillaume, Jean-Luc, Daulat, Avais M., Benleulmi-Chaachoua, Abla, Luka, Marine, Chen, Patty, Kalbasi Anaraki, Dina, Baroncini, Marc, Mannoury la Cour, Clotilde, Millan, Mark J., Prevot, Vincent, Delagrange, Philippe, Jockers, Ralf

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Importance of the second extracellular loop for melatonin MT1 receptor function and absence of melatonin binding in GPR50 von Clement, Nathalie, Renault, Nicolas, Guillaume, Jean‐Luc, Cecon, Erika, Journé, Anne‐Sophie, Laurent, Xavier, Tadagaki, Kenjiro, Cogé, Francis, Gohier, Arnaud, Delagrange, Philippe, Chavatte, Philippe, Jockers, Ralf

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The orphan GPR50 receptor specifically inhibits MT1 melatonin receptor function through heterodimerization von Levoye, Angélique, Dam, Julie, Ayoub, Mohammed A, Guillaume, Jean-Luc, Couturier, Cyril, Delagrange, Philippe, Jockers, Ralf

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Molecular tools to study melatonin pathways and actions von Boutin, Jean A, Audinot, Valérie, Ferry, Gilles, Delagrange, Philippe

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Daily variation in the electrophysiological activity of mouse medial habenula neurones von Sakhi, Kanwal, Belle, Mino D. C., Gossan, Nicole, Delagrange, Philippe, Piggins, Hugh D.

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The orphan GPR50 receptor promotes constitutive TGFβ receptor signaling and protects against cancer development von Wojciech, Stefanie, Ahmad, Raise, Belaid-Choucair, Zakia, Journé, Anne-Sophie, Gallet, Sarah, Dam, Julie, Daulat, Avais, Ndiaye-Lobry, Delphine, Lahuna, Olivier, Karamitri, Angeliki, Guillaume, Jean-Luc, Do Cruzeiro, Marcio, Guillonneau, François, Saade, Anastasia, Clément, Nathalie, Courivaud, Thomas, Kaabi, Nawel, Tadagaki, Kenjiro, Delagrange, Philippe, Prévot, Vincent, Hermine, Olivier, Prunier, Céline, Jockers, Ralf

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Protein interactome mining defines melatonin MT1 receptors as integral component of presynaptic protein complexes of neurons von Benleulmi-Chaachoua, Abla, Chen, Lina, Sokolina, Kate, Wong, Victoria, Jurisica, Igor, Emerit, Michel Boris, Darmon, Michèle, Espin, Almudena, Stagljar, Igor, Tafelmeyer, Petra, Zamponi, Gerald W., Delagrange, Philippe, Maurice, Pascal, Jockers, Ralf

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Preferential Formation of MT1/MT2 Melatonin Receptor Heterodimers with Distinct Ligand Interaction Properties Compared with MT2 Homodimers von Ayoub, Mohammed A, Levoye, Angélique, Delagrange, Philippe, Jockers, Ralf

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X‐ray structural studies of quinone reductase 2 nanomolar range inhibitors von Pegan, Scott D., Sturdy, Megan, Ferry, Gilles, Delagrange, Philippe, Boutin, Jean A., Mesecar, Andrew D.

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Recombinant human melatonin receptor MT1 isolated in mixed detergents shows pharmacology similar to that in mammalian cell membranes von Logez, Christel, Berger, Sylvie, Legros, Céline, Banères, Jean-Louis, Cohen, William, Delagrange, Philippe, Nosjean, Olivier, Boutin, Jean A, Ferry, Gilles, Simonin, Frédéric, Wagner, Renaud

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Hamster Melatonin Receptors: Cloning and Binding Characterization of MT1 and Attempt to Clone MT2 von Gautier, Célia, Dufour, Emilie, Dupré, Clémence, Lizzo, Giulia, Caignard, Sarah, Riest-Fery, Isabelle, Brasseur, Chantal, Legros, Céline, Delagrange, Philippe, Nosjean, Olivier, Simonneaux, Valérie, Boutin, Jean, Guenin, Sophie-Pénélope

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Expression of the orphan GPR50 protein in rodent and human dorsomedial hypothalamus, tanycytes and median eminence von Sidibe, Anissa, Mullier, Amandine, Chen, Patty, Baroncini, Marc, Boutin, Jean A., Delagrange, Philippe, Prevot, Vincent, Jockers, Ralf

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Purification and Identification of G Protein-coupled Receptor Protein Complexes under Native Conditions von Daulat, Avais M., Maurice, Pascal, Froment, Carine, Guillaume, Jean-Luc, Broussard, Cédric, Monsarrat, Bernard, Delagrange, Philippe, Jockers, Ralf

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Functional Expression of MT2 (Mel1b) Melatonin Receptors in Human PAZ6 Adipocytes von Brydon, Lena, Petit, Laurence, Delagrange, Philippe, Strosberg, A. Donny, Jockers, Ralf

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Novel conformationally constrained analogues of agomelatine as new melatoninergic ligands von Rami, Marouan, Landagaray, Elodie, Ettaoussi, Mohamed, Boukhalfa, Koussayla, Caignard, Daniel-Henri, Delagrange, Philippe, Berthelot, Pascal, Yous, Saïd

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