Discovery of potent, selective 4-fluoroproline-based thrombin inhibitors with improved metabolic stability von Staas, Donnette D., Savage, Kelly L., Sherman, Vanessa L., Shimp, Heidi L., Lyle, Terry A., Tran, Lekhanh O., Wiscount, Catherine M., McMasters, Daniel R., Sanderson, Philip E.J., Williams, Peter D., Lucas, Bobby J., Krueger, Julie A., Dale Lewis, S., White, Rebecca B., Yu, Sean, Wong, Bradley K., Kochansky, Christopher J., Reza Anari, M., Yan, Youwei, Vacca, Joseph P.

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Metabolism-Directed Optimization of 3-Aminopyrazinone Acetamide Thrombin Inhibitors. Development of an Orally Bioavailable Series Containing P1 and P3 Pyridines von Burgey, Christopher S, Robinson, Kyle A, Lyle, Terry A, Sanderson, Philip E. J, Lewis, S. Dale, Lucas, Bobby J, Krueger, Julie A, Singh, Rominder, Miller-Stein, Cynthia, White, Rebecca B, Wong, Bradley, Lyle, Elizabeth A, Williams, Peter D, Coburn, Craig A, Dorsey, Bruce D, Barrow, James C, Stranieri, Maria T, Holahan, Marie A, Sitko, Gary R, Cook, Jacquelynn J, McMasters, Daniel R, McDonough, Colleen M, Sanders, William M, Wallace, Audrey A, Clayton, Franklin C, Bohn, Dennis, Leonard, Yvonne M, Detwiler, Theodore J, Lynch, Joseph J, Yan, Youwei, Chen, Zhongguo, Kuo, Lawrence, Gardell, Stephen J, Shafer, Jules A, Vacca, Joseph P

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Small, low nanomolar, noncovalent thrombin inhibitors lacking a group to fill the ‘Distal binding pocket’ von Sanderson, Philip E.J., Cutrona, Kellie J., Dyer, Dona L., Krueger, Julie A., Kuo, Lawrence C., Lewis, S.Dale, Lucas, Bobby J., Yan, Youwei

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Azaindoles: moderately basic P1 groups for enhancing the selectivity of thrombin inhibitors von Sanderson, Philip E.J., Stanton, Matthew G., Dorsey, Bruce D., Lyle, Terry A., McDonough, Colleen, Sanders, William M., Savage, Kelly L., Naylor-Olsen, Adel M., Krueger, Julie A., Lewis, S.Dale, Lucas, Bobby J., Lynch, Joseph J., Yan, Youwei

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Enantioselective complexation of simple amides by a C2 host molecule von Sanderson, Philip E. J, Kilburn, Jeremy D, Still, W. Clark

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The phenyldimethylsilyl group as a masked hydroxy group von Fleming, Ian, Henning, Rolf, Parker, David C., Plaut, Howard E., Sanderson, Philip E. J.

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3-Amino-4-sulfonylpyridinone acetamide and related pyridothiadiazine thrombin inhibitors von Sanderson, Philip E.J., Cutrona, Kellie J., Savage, Kelly L., Naylor-Olsen, Adel M., Bickel, Denise J., Bohn, Dennis L., Clayton, Franklin C., Krueger, Julie A., Lewis, S.Dale, Lucas, Bobby J., Lyle, Elizabeth A., Wallace, Audrey A., Welsh, Denice C., Yan, Youwei

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Small, noncovalent serine protease inhibitors von Sanderson, Philip E. J.

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Novel indole-3-sulfonamides as potent HIV non-nucleoside reverse transcriptase inhibitors (NNRTIs) von Zhao, Zhijian, Wolkenberg, Scott E., Lu, Meiqing, Munshi, Vandna, Moyer, Gregory, Feng, Meizhen, Carella, Anthony V., Ecto, Linda T., Gabryelski, Lori J., Lai, Ming-Tain, Prasad, Sridar G., Yan, Youwei, McGaughey, Georgia B., Miller, Michael D., Lindsley, Craig W., Hartman, George D., Vacca, Joseph P., Williams, Theresa M.

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Enantioselective complexation of the alanine dipeptide by a C2 host molecule von Liu, Ruiping, Sanderson, Philip E. J, Still, W. Clark

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Efficacious, Orally Bioavailable Thrombin Inhibitors Based on 3-Aminopyridinone or 3-Aminopyrazinone Acetamide Peptidomimetic Templates von Sanderson, Philip E. J, Lyle, Terry A, Cutrona, Kellie J, Dyer, Dona L, Dorsey, Bruce D, McDonough, Colleen M, Naylor-Olsen, Adel M, Chen, I-Wu, Chen, Zhongguo, Cook, Jacquelynn J, Cooper, Carolyn M, Gardell, Stephen J, Hare, Timothy R, Krueger, Julie A, Lewis, S. Dale, Lin, Jiunn H, Lucas, Bobby J, Lyle, Elizabeth A, Lynch, Joseph J, Stranieri, Maria T, Vastag, Kari, Yan, Youwei, Shafer, Jules A, Vacca, Joseph P

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Characterization of the Two-step Pathway for Inhibition of Thrombin by α-Ketoamide Transition State Analogs von Sidney D. Lewis, Bobby J. Lucas, Stephen F. Brady, John T. Sisko, Kellie J. Cutrona, Philip E. J. Sanderson, Roger M. Freidinger, Shi-Shan Mao, Stephen J. Gardell, Jules A. Shafer

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COMPUESTOS DERIVADOS DE NAFTIRIDINA SUSTITUIDOS, INHIBIDORES DE LA ACTIVIDAD DE AKT; COMPOSICIN FARMACEUTICA QUE COMPRENDE A DICHO COMPUESTO; Y USO DEL COMPUESTO PARA EL TRATAMIENT... von LAYTON, MARK E., RODZINAK, KEVIN J., SANDERSON, PHILIP E

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The Regiochemistry of the Protodesilylation of Some Cyclopropylmethylsilanes Derived from Allylsilanes von Fleming, Ian, Sanderson, Philip E. J., Terrett, Nicholas K.

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ChemInform Abstract: Small, Noncovalent Serine Protease Inhibitors von Sanderson, Philip E. J.

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3-Amino-4-sulfonylpyridinone Acetamide and Related Pyridothiadiazine Thrombin Inhibitors von Sanderson, Philip E. J., ., et al

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1,3-disubstituted heteroaryl nmda/nr2b antagonists von LAYTON MARK E.,RODZINAK KEVIN J.,KELLY MICHAEL J.III,SANDERSON PHILIP E

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Small, Low Nanomolar, Noncovalent Thrombin Inhibitors Lacking a Group to Fill the "Distal Binding Pocket" von Sanderson, Philip E. J., Cutrona, Kellie J., Dyer, Dona L., Krueger, Julie A., Kuo, Lawrence C., Lewis, S. Dale, Lucas, Bobby J., Yan, Youwei

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THROMBIN INHIBITORS von STAAS, DONNETTE, D, LYLE, TERRY, A, SANDERSON, PHILIP, E. J, WILLIAMS, PETER, D

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THROMBIN INHIBITORS von PHILIP, E. J. SANDERSON, TERRY, A. LYLE, DONNETTE, D. STAAS, PETER, D. WILLIAMS

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