Entropy–Entropy Compensation between the Protein, Ligand, and Solvent Degrees of Freedom Fine-Tunes Affinity in Ligand Binding to Galectin-3C von Wallerstein, Johan, Ekberg, Vilhelm, Ignjatović, Majda Misini, Kumar, Rohit, Caldararu, Octav, Peterson, Kristoffer, Wernersson, Sven, Brath, Ulrika, Leffler, Hakon, Oksanen, Esko, Logan, Derek T., Nilsson, Ulf J., Ryde, Ulf, Akke, Mikael

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Determining the Affinity and Kinetics of Small Molecule Inhibitors of Galectin-1 Using Surface Plasmon Resonance von Kim, Henry, Kretz, Louis, Ronin, Céline, Starck, Christina, Roper, James A, Kahl-Knutson, Barbro, Peterson, Kristoffer, Leffler, Hakon, Nilsson, Ulf J, Pedersen, Anders, Zetterberg, Fredrik R, Slack, Robert J

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Discovery and Optimization of the First Highly Effective and Orally Available Galectin‑3 Inhibitors for Treatment of Fibrotic Disease von Zetterberg, Fredrik R., MacKinnon, Alison, Brimert, Thomas, Gravelle, Lise, Johnsson, Richard E., Kahl-Knutson, Barbro, Leffler, Hakon, Nilsson, Ulf J., Pedersen, Anders, Peterson, Kristoffer, Roper, James A., Schambye, Hans, Slack, Robert J., Tantawi, Susan

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Discovery of Selective and Orally Available Galectin‑1 Inhibitors von Zetterberg, Fredrik R., Diehl, Carl, Håkansson, Maria, Kahl-Knutson, Barbro, Leffler, Hakon, Nilsson, Ulf J., Peterson, Kristoffer, Roper, James A., Slack, Robert J.

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Systematic Tuning of Fluoro-galectin‑3 Interactions Provides Thiodigalactoside Derivatives with Single-Digit nM Affinity and High Selectivity von Peterson, Kristoffer, Kumar, Rohit, Stenström, Olof, Verma, Priya, Verma, Prashant R, Håkansson, Maria, Kahl-Knutsson, Barbro, Zetterberg, Fredrik, Leffler, Hakon, Akke, Mikael, Logan, Derek T, Nilsson, Ulf J

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Monosaccharide Derivatives with Low‐Nanomolar Lectin Affinity and High Selectivity Based on Combined Fluorine–Amide, Phenyl–Arginine, Sulfur–π, and Halogen Bond Interactions... von Zetterberg, Fredrik R., Peterson, Kristoffer, Johnsson, Richard E., Brimert, Thomas, Håkansson, Maria, Logan, Derek T., Leffler, Hakon, Nilsson, Ulf J.

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Surface guided electron FLASH radiotherapy for canine cancer patients von Mannerberg, Annika, Konradsson, Elise, Kügele, Malin, Edvardsson, Anneli, Kadhim, Mustafa, Ceberg, Crister, Peterson, Kristoffer, Thomasson, Hanna‐Maria, Arendt, Maja L., Børresen, Betina, Jensen, Kristine Bastholm, Ceberg, Sofie

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Galectin‑9 Signaling Drives Breast Cancer Invasion through Extracellular Matrix von Pally, Dharma, Banerjee, Mallar, Hussain, Shahid, Kumar, Rekha V., Petersson, Alexandra, Rosendal, Ebba, Gunnarsson, Ludvig, Peterson, Kristoffer, Leffler, Hakon, Nilsson, Ulf J., Bhat, Ramray

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Discovery of the Selective and Orally Available Galectin‑1 Inhibitor GB1908 as a Potential Treatment for Lung Cancer von Zetterberg, Fredrik R., Peterson, Kristoffer, Nilsson, Ulf J., Andréasson Dahlgren, Kajsa, Diehl, Carl, Holyer, Ian, Håkansson, Maria, Khabut, Areej, Kahl-Knutson, Barbro, Leffler, Hakon, MacKinnon, Alison C., Roper, James A., Slack, Robert J., Zarrizi, Reihaneh, Pedersen, Anders

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Galectin‐3 is an amplifier of the interleukin‐1β‐mediated inflammatory response in corneal keratinocytes von Uchino, Yuichi, Woodward, Ashley M., Mauris, Jérôme, Peterson, Kristoffer, Verma, Priya, Nilsson, Ulf J., Rajaiya, Jaya, Argüeso, Pablo

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Galectin-3: studying role of fluorine interaction to achieve high affinity and selectivity von Kumar, Rohit, Peterson, Kristoffer, Nilsson, Ulf, Logan, Derek

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Substituted polyfluoroaryl interactions with an arginine side chain in galectin-3 are governed by steric-, desolvation and electronic conjugation effects von Kumar, Rohit, Peterson, Kristoffer, Misini Ignjatović, Majda, Leffler, Hakon, Ryde, Ulf, Nilsson, Ulf J, Logan, Derek T

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Galectin-1 Induces the Production of Immune-Suppressive Cytokines in Human and Mouse T Cells von Herman, Kimberly D., Holyer, Ian, Humphries, Duncan C., Adamska, Anna, Roper, James A., Peterson, Kristoffer, Zetterberg, Fredrik R., Pedersen, Anders, MacKinnon, Alison C., Slack, Robert J.

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In Vivo Veritas: 18F‑Radiolabeled Glycomimetics Allow Insights into the Pharmacological Fate of Galectin‑3 Inhibitors von Bratteby, Klas, Torkelsson, Edvard, L’Estrade, Elina Tampio, Peterson, Kristoffer, Shalgunov, Vladimir, Xiong, Mengfei, Leffler, Hakon, Zetterberg, Fredrik R, Olsson, Tomas G, Gillings, Nic, Nilsson, Ulf J, Herth, Matthias M, Erlandsson, Maria

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Substituted polyfluoroaryl interactions with an arginine side chain in galectin-3 are governed by steric-, desolvation and electronic conjugation effectsElectronic supplementary in... von Kumar, Rohit, Peterson, Kristoffer, Misini Ignjatovi, Majda, Leffler, Hakon, Ryde, Ulf, Nilsson, Ulf J, Logan, Derek T

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Structure and Energetics of Ligand–Fluorine Interactions with Galectin‐3 Backbone and Side‐Chain Amides: Insight into Solvation Effects and Multipolar Interactions von Kumar, Rohit, Ignjatović, Majda Misini, Peterson, Kristoffer, Olsson, Martin, Leffler, Hakon, Ryde, Ulf, Nilsson, Ulf J., Logan, Derek T.

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Molecular basis for galectin-ligand interactions : Design, synthesis and analysis of ligands von Peterson, Kristoffer

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3-Substituted 1-Naphthamidomethyl-C-galactosyls Interact with Two Unique Sub-sites for High-Affinity and High-Selectivity Inhibition of Galectin-3 von Dahlqvist, Alexander, Mandal, Santanu, Peterson, Kristoffer, Håkansson, Maria, Logan, Derek T, Zetterberg, Fredrik R, Leffler, Hakon, Nilsson, Ulf J

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Aromatic heterocycle galectin-1 interactions for selective single-digit nM affinity ligands von Peterson, Kristoffer, Collins, Patrick M, Huang, Xiaoli, Kahl-Knutsson, Barbro, Essén, Sofia, Zetterberg, Fredrik R, Oredsson, Stina, Leffler, Hakon, Blanchard, Helen, Nilsson, Ulf J

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In Vivo Veritas : 18 F-Radiolabeled Glycomimetics Allow Insights into the Pharmacological Fate of Galectin-3 Inhibitors von Bratteby, Klas, Torkelsson, Edvard, L'Estrade, Elina Tampio, Peterson, Kristoffer, Shalgunov, Vladimir, Xiong, Mengfei, Leffler, Hakon, Zetterberg, Fredrik R, Olsson, Tomas G, Gillings, Nic, Nilsson, Ulf J, Herth, Matthias M, Erlandsson, Maria

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