Discovery of Benzothiazole Scaffold-Based DNA Gyrase B Inhibitors von Gjorgjieva, Marina, Tomašič, Tihomir, Barančokova, Michaela, Katsamakas, Sotirios, Ilaš, Janez, Tammela, Päivi, Peterlin Mašič, Lucija, Kikelj, Danijel

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Overcoming challenges of HERG potassium channel liability through rational design: Eag1 inhibitors for cancer treatment von Toplak, Žan, Hendrickx, Louise A., Abdelaziz, Reham, Shi, Xiaoyi, Peigneur, Steve, Tomašič, Tihomir, Tytgat, Jan, Peterlin‐Mašič, Lucija, Pardo, Luis A.

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Discovery of 4,5,6,7-Tetrahydrobenzo[1,2‑d]thiazoles as Novel DNA Gyrase Inhibitors Targeting the ATP-Binding Site von Tomašič, Tihomir, Katsamakas, Sotirios, Hodnik, Žiga, Ilaš, Janez, Brvar, Matjaž, Solmajer, Tom, Montalvão, Sofia, Tammela, Päivi, Banjanac, Mihailo, Ergović, Gabrijela, Anderluh, Marko, Mašič, Lucija Peterlin, Kikelj, Danijel

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Computer-aided structure-based optimization of 4,5,6,7-tetrahydrobenzo[]thiazole-2,6-diamine derivatives as DNA gyrase B inhibitors von Gutierrez, Lucas J, Vettorazzi, Marcela, Dernovšek, Jaka, Durcik, Martina, Maši, Lucija Peterlin, Tomaši, Tihomir, Enriz, Ricardo D

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Benzothiazole DNA gyrase inhibitors and their conjugates with siderophore mimics: design, synthesis and evaluation von Durcik, Martina, Cruz, Cristina D, Scorciapino, Mariano Andrea, Ilaš, Janez, Tammela, Päivi, Ceccarelli, Matteo, Maši, Lucija Peterlin, Tomaši, Tihomir

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Rational design of balanced dual-targeting antibiotics with limited resistance von Nyerges, Akos, Tomašič, Tihomir, Durcik, Martina, Revesz, Tamas, Szili, Petra, Draskovits, Gabor, Bogar, Ferenc, Skok, Žiga, Zidar, Nace, Ilaš, Janez, Zega, Anamarija, Kikelj, Danijel, Daruka, Lejla, Kintses, Balint, Vasarhelyi, Balint, Foldesi, Imre, Kata, Diána, Welin, Martin, Kimbung, Raymond, Focht, Dorota, Mašič, Lucija Peterlin, Pal, Csaba

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N‑Phenyl-4,5-dibromopyrrolamides and N‑Phenylindolamides as ATP Competitive DNA Gyrase B Inhibitors: Design, Synthesis, and Evaluation von Zidar, Nace, Macut, Helena, Tomašič, Tihomir, Brvar, Matjaž, Montalvão, Sofia, Tammela, Päivi, Solmajer, Tom, Peterlin Mašič, Lucija, Ilaš, Janez, Kikelj, Danijel

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New N -phenylpyrrolamide inhibitors of DNA gyrase with improved antibacterial activity von Cotman, Andrej Emanuel, Fulgheri, Federica, Piga, Martina, Peršolja, Peter, Tiz, Davide Benedetto, Skok, Žiga, Durcik, Martina, Sterle, Maša, Dernovšek, Jaka, Cruz, Cristina D, Tammela, Päivi, Szili, Petra Éva, Daruka, Lejla, Pál, Csaba, Zega, Anamarija, Mašič, Lucija Peterlin, Ilaš, Janez, Tomašič, Tihomir, Kikelj, Danijel, Zidar, Nace

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Bioactivation of bisphenol A and its analogs (BPF, BPAF, BPZ and DMBPA) in human liver microsomes von Schmidt, Jan, Kotnik, Petra, Trontelj, Jurij, Knez, Željko, Mašič, Lucija Peterlin

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Synthesis, Antiproliferative Effect, and Topoisomerase II Inhibitory Activity of 3‑Methyl-2-phenyl‑1H‑indoles von Zidar, Nace, Secci, Daniela, Tomašič, Tihomir, Mašič, Lucija Peterlin, Kikelj, Danijel, Passarella, Daniele, Argaez, Aida Nelly Garcia, Hyeraci, Mariafrancesca, Dalla Via, Lisa

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Discovery of Novel 5-Benzylidenerhodanine and 5-Benzylidenethiazolidine-2,4-dione Inhibitors of MurD Ligase von Zidar, Nace, Tomašić, Tihomir, Šink, Roman, Rupnik, Veronika, Kovač, Andreja, Turk, Samo, Patin, Delphine, Blanot, Didier, Contreras Martel, Carlos, Dessen, Andréa, Müller Premru, Manica, Zega, Anamarija, Gobec, Stanislav, Peterlin Mašič, Lucija, Kikelj, Danijel

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Structure-Activity Relationships of Benzothiazole-Based Hsp90 C-Terminal-Domain Inhibitors von Dernovšek, Jaka, Zajec, Živa, Durcik, Martina, Mašič, Lucija Peterlin, Gobec, Martina, Zidar, Nace, Tomašič, Tihomir

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Exploring the Chemical Space of Benzothiazole-Based DNA Gyrase B Inhibitors von Skok, Žiga, Barančoková, Michaela, Benek, Ondřej, Cruz, Cristina Durante, Tammela, Päivi, Tomašič, Tihomir, Zidar, Nace, Mašič, Lucija Peterlin, Zega, Anamarija, Stevenson, Clare E. M, Mundy, Julia E. A, Lawson, David M, Maxwell, Anthony, Kikelj, Danijel, Ilaš, Janez

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Structure-Function Studies of Sponge-Derived Compounds on the Cardiac CaV3.1 Channel von Depuydt, Anne-Sophie, Patel, Piyush A., Toplak, Žan, Bhat, Chinmaya, Voráčová, Manuela, Eteläinen, Irene, Vitulano, Fiammetta, Bruun, Tanja, Lempinen, Antti, Hribernik, Nives, Mäki-Lohiluoma, Eero, Hendrickx, Louise, Pinheiro-Junior, Ernesto Lopes, Tomašič, Tihomir, Mašič, Lucija Peterlin, Yli-Kauhaluoma, Jari, Kiuru, Paula, Tytgat, Jan, Peigneur, Steve

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Efflux pump inhibitors of clinically relevant multidrug resistant bacteria von Lamut, Andraž, Peterlin Mašič, Lucija, Kikelj, Danijel, Tomašič, Tihomir

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Bioactivation Potential of Thiophene-Containing Drugs von Gramec, Darja, Peterlin Mašič, Lucija, Sollner Dolenc, Marija

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Enhancing Antibacterial Efficacy: Combining Novel Bacterial Topoisomerase Inhibitors with Efflux Pump Inhibitors and Other Agents Against Gram-Negative Bacteria von Zorman, Maša, Kokot, Maja, Zdovc, Irena, Senerovic, Lidija, Mandic, Mina, Zidar, Nace, Cotman, Andrej Emanuel, Durcik, Martina, Peterlin Mašič, Lucija, Minovski, Nikola, Anderluh, Marko, Hrast Rambaher, Martina

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Bisphenol A and its analogs: Do their metabolites have endocrine activity? von GramecSkledar, Darja, Peterlin Mašič, Lucija

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Design of New Potent and Selective Thiophene-Based KV1.3 Inhibitors and Their Potential for Anticancer Activity von Gubič, Špela, Hendrickx, Louise, Shi, Xiaoyi, Toplak, Žan, Možina, Štefan, Theemsche, Kenny, Pinheiro-Junior, Ernesto, Peigneur, Steve, Labro, Alain, Pardo, Luis, Tytgat, Jan, Tomašič, Tihomir, Mašič, Lucija

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Antimicrobial activity of the marine alkaloids, clathrodin and oroidin, and their synthetic analogues von Zidar, Nace, Montalvão, Sofia, Hodnik, Žiga, Nawrot, Dorota A, Žula, Aleš, Ilaš, Janez, Kikelj, Danijel, Tammela, Päivi, Mašič, Lucija Peterlin

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