Phosphoramidates and phosphonamidates (ProTides) with antiviral activity von Slusarczyk, Magdalena, Serpi, Michaela, Pertusati, Fabrizio

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Polyfluorinated groups in medicinal chemistry von Bassetto, Marcella, Ferla, Salvatore, Pertusati, Fabrizio

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Synthesis of 2‐Acetamido‐1,3,4‐Tri‐O‐Acetyl‐2‐Deoxy‐D‐Mannopyranose ‐6‐Phosphate Prodrugs as Potential Therapeutic Agents von Pertusati, Fabrizio, Morewood, James

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Phosphonoamidate prodrugs of C5-substituted pyrimidine acyclic nucleosides for antiviral therapy von Pertusati, Fabrizio, Serafini, Sara, Albadry, Najmiyah, Snoeck, Robert, Andrei, Graciela

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Design and synthesis of novel bicalutamide and enzalutamide derivatives as antiproliferative agents for the treatment of prostate cancer von Bassetto, Marcella, Ferla, Salvatore, Pertusati, Fabrizio, Kandil, Sahar, Westwell, Andrew D., Brancale, Andrea, McGuigan, Christopher

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λ5‑Phosphorus-Containing α‑Diazo Compounds: A Valuable Tool for Accessing Phosphorus-Functionalized Molecules von Marinozzi, Maura, Pertusati, Fabrizio, Serpi, Michaela

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[Delta]5-Phosphorus-Containing [alpha]-Diazo Compounds: A Valuable Tool for Accessing Phosphorus-Functionalized Molecules von Marinozzi, Maura, Pertusati, Fabrizio, Serpi, Michaela

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A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents... von Pertusati, Fabrizio, Ferla, Salvatore, Bassetto, Marcella, Brancale, Andrea, Khandil, Sahar, Westwell, Andrew D., McGuigan, Christopher

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Drug repurposing: phosphate prodrugs of anticancer and antiviral FDA-approved nucleosides as novel antimicrobials von Pertusati, Fabrizio, Pileggi, Elisa, Richards, Jennifer, Wootton, Mandy, Van Leemputte, Thijs, Persoons, Leentje, De Coster, David, Villanueva, Xabier, Daelemans, Dirk, Steenackers, Hans, McGuigan, Christopher, Serpi, Michaela

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Synthesis, molecular docking and antibacterial activity of an oxadiazole-based lipoteichoic acid inhibitor and its metabolites von Serpi, Michaela, Pertusati, Fabrizio, Morozzi, Chiara, Novelli, Giulia, Giannantonio, Daniele, Duggan, Katrina, Vittorio, Serena, Fallis, Ian A., De Luca, Laura, Williams, David

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Medicinal Chemistry of Nucleoside Phosphonate Prodrugs for Antiviral Therapy von Pertusat, Fabrizio, Serpi, Michaela, McGuigan, Christopher

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Targeting GNE Myopathy: A Dual Prodrug Approach for the Delivery of N‑Acetylmannosamine 6‑Phosphate von Morozzi, Chiara, Sedláková, Jana, Serpi, Michaela, Avigliano, Marialuce, Carbajo, Rosangela, Sandoval, Lucia, Valles-Ayoub, Yadira, Crutcher, Patrick, Thomas, Stephen, Pertusati, Fabrizio

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Kinase-independent phosphoramidate S1P1 receptor agonist benzyl ether derivatives von James, Edward, Pertusati, Fabrizio, Brancale, Andrea, McGuigan, Chris

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Phosphonoamidate prodrugs of C5-substituted pyrimidine acyclic nucleosides for antiviral therapy von Pertusati, Fabrizio, Serafini, Sara, Albadry, Najmiyah, Snoeck, Robert, Andrei, Graciela

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Expedient synthesis and biological evaluation of alkenyl acyclic nucleoside phosphonate prodrugs von Pileggi, Elisa, Serpi, Michaela, Andrei, Graciela, Schols, Dominique, Snoeck, Robert, Pertusati, Fabrizio

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Preparation of Pyrimidine Alkenyl Acyclic Nucleoside Phosphonoamidates von Pileggi, Elisa, Serpi, Michaela, Pertusati, Fabrizio

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Rational design and synthesis of novel anti-prostate cancer agents bearing a 3,5-bis-trifluoromethylphenyl moiety von Ferla, Salvatore, Bassetto, Marcella, Pertusati, Fabrizio, Kandil, Sahar, Westwell, Andrew D., Brancale, Andrea, McGuigan, Christopher

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PMPA and PMEA prodrugs for the treatment of HIV infections and human papillomavirus (HPV) associated neoplasia and cancer von Pertusati, Fabrizio, Hinsinger, Karen, Flynn, Áine Sinéad, Powell, Ned, Tristram, Amanda, Balzarini, Jan, McGuigan, Christopher

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Design, synthesis and biological evaluation of phosphorodiamidate prodrugs of antiviral and anticancer nucleosides von McGuigan, Christopher, Bourdin, Claire, Derudas, Marco, Hamon, Nadège, Hinsinger, Karen, Kandil, Sahar, Madela, Karolina, Meneghesso, Silvia, Pertusati, Fabrizio, Serpi, Michaela, Slusarczyk, Magdalena, Chamberlain, Stanley, Kolykhalov, Alexander, Vernachio, John, Vanpouille, Christophe, Introini, Andrea, Margolis, Leonid, Balzarini, Jan

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Synthesis of 2-Chirally Substituted 3,3′-Biquinazoline-4,4′-diones von Pertusati, Fabrizio, Coogan, Michael P.

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