Induction of hepatitis A virus-neutralizing antibody by a virus-specific synthetic peptide von EMINI, E. A, HUGHES, J. V, PERLOW, D. S, BOGER, J

Volltext

Nonpeptide oxytocin antagonists: Analogs of L-371,257 with improved potency von Williams, Peter D., Bock, Mark G., Evans, Ben E., Freidinger, Roger M., Gallicchio, Steven N., Guidotti, Maribeth T., Jacobson, Marlene A., Kuo, Michelle S., Levy, Michelle R., Lis, Edward V., Michelson, Stuart R., Pawluczyk, Joseph M., Perlow, Debra S., Pettibone, Douglas J., Quigley, Amy G., Reiss, Duane R., Salvatore, Christopher, Stauffer, Kenneth J., Woyden, Carla J.

Volltext

Renin inhibitors. Syntheses of subnanomolar, competitive, transition-state analog inhibitors containing a novel analog of statine von Boger, Joshua, Payne, Linda S, Perlow, Debra S, Lohr, Nancy S, Poe, Martin, Blaine, Edward H, Ulm, Edgar H, Schorn, Terry W, LaMont, Bruce I

Volltext

Nonpeptide oxytocin antagonists: Potent, orally bioavailable analogs of L-371,257 containing A 1- R-(pyridyl)ethyl ether terminus von Kuo, Michelle S., Bock, Mark G., Freidinger, Roger M., Guidotti, Maribeth T., Lis, Edward V., Pawluczyk, Joseph M., Perlow, Debra S., Pettibone, Douglas J., Quigley, Amy G., Reiss, Duane R., Williams, Peter D., Woyden, Carla J.

Volltext

Development of a novel class of cyclic hexapeptide oxytocin antagonists based on a natural product von Williams, Peter D, Bock, Mark G, Tung, Roger D, Garsky, Victor M, Perlow, Debra S, Erb, Jill M, Lundell, G. F, Gould, Norman P, Whitter, Willie L

Volltext

Conformationally constrained tachykinin analogs which are selective ligands for the eledoisin binding site von Cascieri, M A, Chicchi, G G, Freidinger, R M, Colton, C D, Perlow, D S, Williams, B, Curtis, N R, McKnight, A T, Maguire, J J, Veber, D F

Volltext

A super active cyclic hexapeptide analog of somatostatin von Veber, Daniel F., Saperstein, Richard, Nutt, Ruth F., Freidinger, Roger M., Brady, Stephen F., Curley, Paul, Perlow, Debra S., Paleveda, William J., Colton, C.Dylion, Zacchei, Anthony G., Tocco, Dominick J., Hoff, Dale R., Vandlen, Richard L., Gerich, John E., Hall, Larry, Mandarino, Lawrence, Cordes, Eugene H., Anderson, Paul S., Hirschmann, Ralph

Volltext

The selectivity of statine-based inhibitors against various human aspartic proteinases von Jupp, R A, Dunn, B M, Jacobs, J W, Vlasuk, G, Arcuri, K E, Veber, D F, Perlow, D S, Payne, L S, Boger, J, de Laszlo, S

Volltext

Angiotensin-converting enzyme inhibitors: synthesis and biological activity of acyl tripeptide analogues of enalapril von GREENLEE, W. J, ALLIBONE, P. L, PERLOW, D. S, PATCHETT, A. A, ULM, E. H, VASSIL, T. C

Volltext

Use of N-Fmoc amino acid chlorides and activated 2-(fluorenylmethoxy)-5(4H)-oxazolones in solid-phase peptide synthesis. Efficient syntheses of highly N-alkylated cyclic hexapeptid... von Perlow, Debra S, Erb, Jill M, Gould, Norman P, Tung, Roger D, Freidinger, Roger M, Williams, Peter D, Veber, Daniel F

Volltext

Protected lactam-bridged dipeptides for use as conformational constraints in peptides von Freidinger, Roger M, Perlow, Debra Schwenk, Veber, Daniel F

Volltext

Bioactive Conformation of Luteinizing Hormone-Releasing Hormone: Evidence from a Conformationally Constrained Analog von Freidinger, Roger M., Veber, Daniel F., Perlow, Debra Schwenk, Brooks, Jerry R., Saperstein, Richard

Volltext

Conformational modifications of cyclic hexapeptide somatostatin analogs von Freidinger, Roger M., Perlow, Debra Schwenk, Randall, William C., Saperstein, Richard, Arison, Byron H., Veber, Daniel F.

Volltext

A potent cyclic hexapeptide analogue of somatostatin von Veber, Daniel F, Freidinger, Roger M, Perlow, Debra Schwenk, Paleveda, William J, Holly, Frederick W, Strachan, Robert G, Nutt, Ruth F, Arison, Byron H, Homnick, Carl, Randall, William C, Glitzer, Monroe S, Saperstein, Richard, Hirschmann, Ralph

Volltext

A series of 5-(5,6)-dihydrouracil substituted 8-hydroxy-[1,6]naphthyridine-7-carboxylic acid 4-fluorobenzylamide inhibitors of HIV-1 integrase and viral replication in cells von Embrey, Mark W., Wai, John S., Funk, Timothy W., Homnick, Carl F., Perlow, Debbie S., Young, Steven D., Vacca, Joseph P., Hazuda, Daria J., Felock, Peter J., Stillmock, Kara A., Witmer, Marc V., Moyer, Gregory, Schleif, William A., Gabryelski, Lori J., Jin, Lixia, Chen, I-Wu, Ellis, Joan D., Wong, Bradley K., Lin, Jiunn H., Leonard, Yvonne M., Tsou, Nancy N., Zhuang, Linghang

Volltext

Renin inhibitors containing conformationally restricted P1-P1' dipeptide mimetics von Williams, Peter D, Perlow, Debra S, Payne, Linda S, Holloway, M. Katherine, Siegl, Peter K. S, Schorn, Terry W, Lynch, Robert J, Doyle, John J, Strouse, John F

Volltext

Nanomolar-affinity, non-peptide oxytocin receptor antagonists von Evans, Ben E, Lundell, George F, Gilbert, Kevin F, Bock, Mark G, Rittle, Kenneth E, Carroll, Leigh Anne, Williams, Peter D, Pawluczyk, Joseph M, Leighton, James L

Volltext

Conformationally constrained o-tolylpiperazine camphorsulfonamide oxytocin antagonists. Structural modifications that provide high receptor affinity and suggest a bioactive conform... von Williams, Peter D., Ball, Richard G., Clineschmidt, Bradley V., Culberson, J.Chris, Erb, Jill M., Freidinger, Roger M., Pawluczyk, Joseph M., Perlow, Debra S., Pettibone, Douglas J., Veber, Daniel F.

Volltext

Synthesis of 9-fluorenylmethyloxycarbonyl-protected N-alkyl amino acids by reduction of oxazolidinones von Freidinger, Roger M, Hinkle, Jeffery S, Perlow, Debra S

Volltext

1-7,7-Dimethyl-2(S)-(2(S)-amino-4-(methylsulfonyl)butyramido)bicyclo[2.2.1]-heptan-1(S)-ylmethylsulfonyl-4-(2-methylphenyl)piperazine (L-368,899) : an orally bioavailable, non-pept... von WILLIAMS, P. D, ANDERSON, P. S, FITZPATRICK, S. L, FREIDINGER, R. M, KAUFMAN, M. J, LUNDELL, G. F, MURPHY, J. S, PAWLUCZYK, J. M, PERLOW, D. S, PETTIBONE, D. J, PITZENBERGER, S. M, THOMPSON, K. L, BALL, R. G, VEBER, D. F, BOCK, M. G, CARROLL, L.-A, SHUET-HING LEE CHIU, CLINESCHMIDT, B. V, CULBERSON, J. C, ERB, J. M, EVANS, B. E

Volltext