Conformational Plasticity of the 2A Proteinase from Enterovirus 71 von Cai, Qixu, Yameen, Muhammad, Liu, Weihua, Gao, Zhenting, Li, Yaozong, Peng, Xuanjia, Cai, Yaxian, Wu, Caiming, Zheng, Qian, Li, Jian, Lin, Tianwei

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A general approach to access 5,6-dihydroindolo-naphthyridine ring system von He, Shuwen, Li, Peng, Dai, Xing, Liu, Hong, Lai, Zhong, Xiao, Dong, McComas, Casey C., Du, Chunyan, Liu, Yuehui, Yin, Jingjun, Dang, Qun, Zorn, Nicolas, Peng, Xuanjia, Nargund, Ravi P., Palani, Anandan

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Solution-Phase DNA-Compatible Pictet-Spengler Reaction Aided by Machine Learning Building Block Filtering von Li, Ke, Liu, Xiaohong, Liu, Sixiu, An, Yulong, Shen, Yanfang, Sun, Qingxia, Shi, Xiaodong, Su, Wenji, Cui, Weiren, Duan, Zhiqiang, Kuai, Letian, Yang, Hongfang, Satz, Alexander L., Chen, Kaixian, Jiang, Hualiang, Zheng, Mingyue, Peng, Xuanjia, Lu, Xiaojie

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Selections and screenings of DNA-encoded chemical libraries against enzyme and cellular targets von Satz, Alexander L., Kuai, Letian, Peng, Xuanjia

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Synthesis of 1,2-Amino Alcohols by Photoredox-Mediated Decarboxylative Coupling of α‑Amino Acids and DNA-Conjugated Carbonyls von Wen, Huanan, Ge, Rui, Qu, Yi, Sun, Jialin, Shi, Xiaodong, Cui, Weiren, Yan, Hao, Zhang, Qi, An, Yulong, Su, Wenji, Yang, Hongfang, Kuai, Letian, Satz, Alexander L, Peng, Xuanjia

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A Strategy for the Synthesis of Sulfonamides on DNA von Liu, Wei, Deng, Wei, Sun, Saisai, Yu, Chunyan, Su, Xubo, Wu, Aliang, Yuan, Youlang, Ma, Zhonglin, Li, Ke, Yang, Hongfang, Peng, Xuanjia, Dietrich, Justin

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Palladium-mediated Suzuki-Miyaura Cross-Coupling Reaction of Potassium Boc-protected aminomethyltrifluoroborate with DNA-Conjugated aryl bromides for DNA-Encoded chemical library s... von Qu, Yi, Liu, Sixiu, Wen, Huanan, Xu, Yanfen, An, Yulong, Li, Ke, Ni, Mengyuan, Shen, Yanfang, Shi, Xiaodong, Su, Wenji, Cui, Weiren, Kuai, Letian, Satz, Alexander L., Yang, Hongfang, Lu, Xiaojie, Peng, Xuanjia

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Copper-Mediated DNA-Compatible One-Pot Click Reactions of Alkynes with Aryl Borates and TMS-N 3 von Qu, Yi, Wen, Huanan, Ge, Rui, Xu, Yanfen, Gao, Hong, Shi, Xiaodong, Wang, Jiangong, Cui, Weiren, Su, Wenji, Yang, Hongfang, Kuai, Letian, Satz, Alexander L, Peng, Xuanjia

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DNA Compatible Intermolecular Wittig Olefination for the Construction of α, β‑Unsaturated Carbonyl Compounds von An, Yu-Long, Li, Ke, Shen, Yanfang, Hong, Zibing, Chen, Linlin, Hu, Yujing, Zhou, Lichun, Wang, Disha, Shi, Xiaodong, Liu, Shien, Su, Wenji, Cui, Weiren, Kuai, Letian, Yang, Hongfang, Peng, Xuanjia

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Copper-Mediated DNA-Compatible One-Pot Click Reactions of Alkynes with Aryl Borates and TMS-N3 von Qu, Yi, Wen, Huanan, Ge, Rui, Xu, Yanfen, Gao, Hong, Shi, Xiaodong, Wang, Jiangong, Cui, Weiren, Su, Wenji, Yang, Hongfang, Kuai, Letian, Satz, Alexander L, Peng, Xuanjia

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DNA-Compatible Copper-Catalyzed Oxidative Amidation of Aldehydes with Non-Nucleophilic Arylamines von Li, Ke, Qu, Yi, An, Yulong, Breinlinger, Eric, Webster, Matthew P, Wen, Huanan, Ding, Duanchen, Zhao, Meng, Shi, Xiaodong, Wang, Jiangong, Su, Wenji, Cui, Weiren, Satz, Alexander L, Yang, Hongfang, Kuai, Letian, Little, Andrew, Peng, Xuanjia

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Discovery of selective, orally bioavailable, N-linked arylsulfonamide Nav1.7 inhibitors with pain efficacy in mice von Roecker, Anthony J., Egbertson, Melissa, Jones, Kristen L.G., Gomez, Robert, Kraus, Richard L., Li, Yuxing, Koser, Amy Jo, Urban, Mark O., Klein, Rebecca, Clements, Michelle, Panigel, Jacqueline, Daley, Christopher, Wang, Jixin, Finger, Eleftheria N., Majercak, John, Santarelli, Vincent, Gregan, Irene, Cato, Matthew, Filzen, Tracey, Jovanovska, Aneta, Wang, Ying-Hong, Wang, Deping, Joyce, Leo A., Sherer, Edward C., Peng, Xuanjia, Wang, Xiu, Sun, Haiyan, Coleman, Paul J., Houghton, Andrea K., Layton, Mark E.

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Design, synthesis, and biological evaluation of anti-EV71 agents von Li, Peng, Yang, Bailing, Hao, Fei, Wang, Ping, He, Haiying, Huang, Lei, Zhang, Xuan, Zhang, Shengbin, Peng, Xuanjia, Yin, Ke, Hu, Jiao, Chen, Xinsheng, Gu, Zhengxian, Wang, Li, Shen, Liang, Hu, Guoping, Li, Ning, Li, Jian, Chen, Shuhui, Xiao, Wei, Wang, Zhenzhong, Guo, Qingming, Chang, Xiujuan, Zhang, Lanjun, Cai, Qixu, Lin, Tianwei

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Fragment-wise design of inhibitors to 3C proteinase from enterovirus 71 von Wu, Caiming, Zhang, Lanjun, Li, Peng, Cai, Qixu, Peng, Xuanjia, Yin, Ke, Chen, Xinsheng, Ren, Haixia, Zhong, Shilin, Weng, Yuwei, Guan, Yi, Chen, Shuhui, Wu, Jinzhun, Li, Jian, Lin, Tianwei

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Development of a New Structural Class of Broadly Acting HCV Non‐Nucleoside Inhibitors Leading to the Discovery of MK‐8876 von McComas, Casey C., Palani, Anandan, Chang, Wei, Holloway, M. Katharine, Lesburg, Charles A., Li, Peng, Liverton, Nigel, Meinke, Peter T., Olsen, David B., Peng, Xuanjia, Soll, Richard M., Ummat, Ajay, Wu, Jie, Wu, Jin, Zorn, Nicolas, Ludmerer, Steven W.

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Discovery of Arylsulfonamide Nav1.7 Inhibitors: IVIVC, MPO Methods, and Optimization of Selectivity Profile von Roecker, Anthony J, Layton, Mark E, Pero, Joseph E, Kelly, Michael J, Greshock, Thomas J, Kraus, Richard L, Li, Yuxing, Klein, Rebecca, Clements, Michelle, Daley, Christopher, Jovanovska, Aneta, Ballard, Jeanine E, Wang, Deping, Zhao, Fuqiang, Brunskill, Andrew P. J, Peng, Xuanjia, Wang, Xiu, Sun, Haiyan, Houghton, Andrea K, Burgey, Christopher S

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Tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of left-hand-side moiety (Part-2) von Singh, Sheo B, Kaelin, David E, Wu, Jin, Miesel, Lynn, Tan, Christopher M, Black, Todd, Nargund, Ravi, Meinke, Peter T, Olsen, David B, Lagrutta, Armando, Lu, Jun, Patel, Sangita, Rickert, Keith W, Smith, Robert F, Soisson, Stephen, Sherer, Edward, Joyce, Leo A, Wei, Changqing, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Takano, Hisashi, Shibasaki, Mitsuhito, Yajima, Masanobu, Nishimura, Akinori, Shibata, Takeshi, Fukuda, Yasumichi

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Hydroxy tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of RHS moiety (Part-3) von Singh, Sheo B., Kaelin, David E., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Gill, Charles, Black, Todd, Nargund, Ravi, Meinke, Peter T., Olsen, David B., Lagrutta, Armando, Wei, Changqing, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Takeuchi, Tomoko, Shibue, Taku, Ohata, Kohei, Takano, Hisashi, Ban, Shizuka, Nishimura, Akinori, Fukuda, Yasumichi

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Structure activity relationship of pyridoxazinone substituted RHS analogs of oxabicyclooctane-linked 1,5-naphthyridinyl novel bacterial topoisomerase inhibitors as broad-spectrum a... von Singh, Sheo B., Kaelin, David E., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Meinke, Peter T., Olsen, David B., Lagrutta, Armando, Wei, Changqing, Liao, Yonggang, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Yajima, Masanobu, Shibue, Taku, Shibata, Takeshi, Ohata, Kohei, Nishimura, Akinori, Fukuda, Yasumichi

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Discovery of Arylsulfonamide Na v 1.7 Inhibitors: IVIVC, MPO Methods, and Optimization of Selectivity Profile von Roecker, Anthony J, Layton, Mark E, Pero, Joseph E, Kelly, 3rd, Michael J, Greshock, Thomas J, Kraus, Richard L, Li, Yuxing, Klein, Rebecca, Clements, Michelle, Daley, Christopher, Jovanovska, Aneta, Ballard, Jeanine E, Wang, Deping, Zhao, Fuqiang, Brunskill, Andrew P J, Peng, Xuanjia, Wang, Xiu, Sun, Haiyan, Houghton, Andrea K, Burgey, Christopher S

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