Emerging technologies for metabolite generation and structural diversification von Cusack, Kevin P., Koolman, Hannes F., Lange, Udo E.W., Peltier, Hillary M., Piel, Isabel, Vasudevan, Anil

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One-Pot Asymmetric Synthesis of Either Diastereomer of tert-Butanesulfinyl-protected Amines from Ketones von Tanuwidjaja, Jessica, Peltier, Hillary M, Ellman, Jonathan A

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The Total Synthesis of Tubulysin D von Peltier, Hillary M, McMahon, Jeffrey P, Patterson, Andrew W, Ellman, Jonathan A

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Discovery of (R)-(3-fluoropyrrolidin-1-yl)(6-((5-(trifluoromethyl)pyridin-2-yl)oxy)quinolin-2-yl)methanone (ABBV-318) and analogs as small molecule Nav1.7/ Nav1.8 blockers for the... von Patel, Meena V., Peltier, Hillary M., Matulenko, Mark A., Koenig, John R., C. Scanio, Marc J., Gum, Rebecca J., El-Kouhen, Odile F., Fricano, Meagan M., Lundgaard, Greta L., Neelands, Torben, Zhang, Xu-Feng, Zhan, Cenchen, Pai, Madhavi, Ghoreishi-Haack, Nayereh, Hudzik, Thomas, Gintant, Gary, Martin, Ruth, McGaraughty, Steve, Xu, Jun, Bow, Daniel, Kalvass, John C., Kym, Philip R., DeGoey, David A., Kort, Michael E.

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Pharmacological characterization of 1-(5-chloro-6-(trifluoromethoxy)-1H-benzoimidazol-2-yl)-1H-pyrazole-4-carboxylic acid (JNJ-42041935), a potent and selective hypoxia-inducible f... von Barrett, Terrance D, Palomino, Heather L, Brondstetter, Theresa I, Kanelakis, Kimon C, Wu, Xiaodong, Haug, Peter V, Yan, Wen, Young, Andrew, Hua, Hong, Hart, Juliet C, Tran, Da-Thao, Venkatesan, Hariharan, Rosen, Mark D, Peltier, Hillary M, Sepassi, Kia, Rizzolio, Michele C, Bembenek, Scott D, Mirzadegan, Tara, Rabinowitz, Michael H, Shankley, Nigel P

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Design, Synthesis, and Biological Properties of Highly Potent Tubulysin D Analogues von Patterson, Andrew W., Peltier, Hillary M., Sasse, Florenz, Ellman, Jonathan A.

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Expedient Synthesis of N-Methyl Tubulysin Analogues with High Cytotoxicity von Patterson, Andrew W, Peltier, Hillary M, Ellman, Jonathan A

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Results from a Phase 1b/2 Study of Ibrutinib Combination Therapy in Advanced Urothelial Carcinoma von Mar, Nataliya, Zakharia, Yousef, Falcon, Alejandro, Morales-Barrera, Rafael, Mellado, Begona, Duran, Ignacio, Oh, Do-Youn, Williamson, Stephen K, Gajate, Pablo, Arkenau, Hendrik-Tobias, Jones, Robert J, Teo, Min Yuen, Turan, Tolga, McLaughlin, Robert T, Peltier, Hillary M, Chong, Elizabeth, Atluri, Harisha, Dean, James P, Castellano, Daniel

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N-Sulfinyl Metalloenamine Conjugate Additions:  Asymmetric Synthesis of Piperidines von Peltier, Hillary M, Ellman, Jonathan A

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Beyond Traditional Structure-Based Drug Design: The Role of Iron Complexation, Strain, and Water in the Binding of Inhibitors for Hypoxia-Inducible Factor Prolyl Hydroxylase 2 von Bembenek, Scott D, Venkatesan, Hariharan, Peltier, Hillary M, Rosen, Mark D, Barrett, Terrance D, Kanelakis, Kimon C, Palomino, Heather L, Brondstetter, Theresa I, Mirzadegan, Taraneh, Rabinowitz, Michael H

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Catalytic Enantioselective Sulfinyl Transfer Using Cinchona Alkaloid Catalysts von Peltier, Hillary M, Evans, Jared W, Ellman, Jonathan A

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One-Pot Microwave-Promoted Synthesis of Nitriles from Aldehydes via tert-Butanesulfinyl Imines von Tanuwidjaja, Jessica, Peltier, Hillary M., Lewis, Jared C., Schenkel, Laurie B., Ellman, Jonathan A.

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P-422 Impact of early response and CXCR4 mutation status on progression-free survival with ibrutinib-based therapy in Waldenström macroglobulinemia: a post hoc analysis of the iNNO... von Castillo, Jorge, Sarosiek, Shayna, Branagan, Andrew, Bokun, Alex, Peltier, Hillary, Girardi, Vincent, Pacia, Michelle, Treon, Steven

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Benzimidazole-2-pyrazole HIF Prolyl 4-Hydroxylase Inhibitors as Oral Erythropoietin Secretagogues von Rosen, Mark D, Venkatesan, Hariharan, Peltier, Hillary M, Bembenek, Scott D, Kanelakis, Kimon C, Zhao, Lucy X, Leonard, Barry E, Hocutt, Frances M, Wu, Xiaodong, Palomino, Heather L, Brondstetter, Theresa I, Haugh, Peter V, Cagnon, Laurence, Yan, Wen, Liotta, Lisa A, Young, Andrew, Mirzadegan, Tara, Shankley, Nigel P, Barrett, Terrance D, Rabinowitz, Michael H

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Discovery of (R)-(3-fluoropyrrolidin-1-yl)(6-((5-(trifluoromethyl)pyridin-2-yl)oxy)quinolin-2-yl)methanone (ABBV-318) and analogs as small molecule Na v 1.7/ Nav1.8 blockers for th... von Patel, Meena V, Peltier, Hillary M, Matulenko, Mark A, Koenig, John R, C Scanio, Marc J, Gum, Rebecca J, El-Kouhen, Odile F, Fricano, Meagan M, Lundgaard, Greta L, Neelands, Torben, Zhang, Xu-Feng, Zhan, Cenchen, Pai, Madhavi, Ghoreishi-Haack, Nayereh, Hudzik, Thomas, Gintant, Gary, Martin, Ruth, McGaraughty, Steve, Xu, Jun, Bow, Daniel, Kalvass, John C, Kym, Philip R, DeGoey, David A, Kort, Michael E

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Pharmacological Characterization of 1-(5-Chloro-6-(trifluoromethoxy)-1 H -benzoimidazol-2-yl)-1 H -pyrazole-4-carboxylic Acid (JNJ-42041935), a Potent and Selective Hypoxia-Inducib... von Barrett, Terrance D., Palomino, Heather L., Brondstetter, Theresa I., Kanelakis, Kimon C., Wu, Xiaodong, Haug, Peter V., Yan, Wen, Young, Andrew, Hua, Hong, Hart, Juliet C., Tran, Da-Thao, Venkatesan, Hariharan, Rosen, Mark D., Peltier, Hillary M., Sepassi, Kia, Rizzolio, Michele C., Bembenek, Scott D., Mirzadegan, Tara, Rabinowitz, Michael H., Shankley, Nigel P.

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ChemInform Abstract: Emerging Technologies for Metabolite Generation and Structural Diversification von Cusack, Kevin P., Koolman, Hannes F., Lange, Udo E. W., Peltier, Hillary M., Piel, Isabel, Vasudevan, Anil

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Results from a Phase 1b/2 Study of Ibrutinib Combination Therapy in Advanced Urothelial Carcinoma von Mar, Nataliya, Zakharia, Yousef, Falcon, Alejandro, Morales-Barrera, Rafael, Mellado, Begoña, Duran, Ignacio, Oh, Do-Youn, Williamson, Stephen K, Gajate, Pablo, Arkenau, Hendrik-Tobias, Jones, Robert J, Teo, Min Yuen, Turan, Tolga, McLaughlin, Robert T, Peltier, Hillary M, Chong, Elizabeth, Atluri, Harisha, Dean, James P, Castellano, Daniel, Universitat Autònoma de Barcelona

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Benzoimidazoles as prolyl hydroxylase inhibitors von Venkatesan, Hariharan, Peltier, Hillary M, Phuong, Victor K, Rosen, Mark D, Tarantino, Kyle T, Hocutt, Frances Meredith, Rabinowitz, Michael H, Zhao, Lucy Xiumin, Leonard, Jr., Barry Eastman

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BENZOIMIDAZOLES AS PROLYL HYDROXYLASE INHIBITORS von LEONARD, BARRY EASTMAN, PHUONG, VICTOR K, VENKATESAN, HARIHARAN, PELTIER, HILLARY M, RABINOWITZ, MICHAEL H, ZHAO, LUCY XIUMIN, ROSEN, MARK D, HOCUTT, FRANCES MEREDITH, TARANTINO, KYLE T

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