Crystal Structures of Human Factor Xa Complexed with Potent Inhibitors von Maignan, Sébastien, Guilloteau, Jean-Pierre, Pouzieux, Stéphanie, Choi-Sledeski, Yong Mi, Becker, Michael R, Klein, Scott I, Ewing, William R, Pauls, Henry W, Spada, Alfred P, Mikol, Vincent

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Developments in Applied Artificial Intelligence: 16th International Conference on Industrial and Engineering Applications of Artificial Intelligence and Expert Systems, IEA/AIE 200... von Chung, Paul W. H, Hinde, Chris, Ali, Moonis

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Aminoisoquinolines: Design and synthesis of an orally active benzamidine isostere for the inhibition of factor XA von Choi-Sledeski, Y.M., Becker, M.R., Green, D.M., Davis, R., Ewing, W.R., Mason, H.J., Ly, C., Spada, A., Liang, G., Cheney, D., Barton, J., Chu, V., Brown, K., Colussi, D., Bentley, R., Leadley, R., Dunwiddie, C., Pauls, H.W.

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Pharmacological Characterization of a Novel Factor Xa Inhibitor, FXV673 von Chu, Valeria, Brown, Karen, Colussi, Dennis, Gao, Jingbo, Bostwick, Jeffery, Kasiewski, Charles, Bentley, Ross, Morgan, Susan, Guertin, Kevin, Pauls, Henry W, Gong, Yong, Zulli, Alison, Perrone, Mark H, Dunwiddie, Christopher T, Leadley, Robert J

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In Vitro Characterization of a Novel Factor Xa Inhibitor, RPR 130737 von Chu, Valeria, Brown, Karen, Colussi, Dennis, Choi, Yong-Mi, Green, Dan, Pauls, Henry W, Spada, Alfred P, Perrone, Mark H, Leadley, Robert J, Dunwiddie, Christopher T

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Synthesis, SAR and in vivo activity of novel thienopyridine sulfonamide pyrrolidinones as factor Xa inhibitors von Becker, Michael R., Ewing, William R., Davis, Roderick S., Pauls, Henry W., Ly, Cuong, Li, Aiwen, Mason, Helen J., Choi-Sledeski, Yong Mi, Spada, Alfred P., Chu, Valeria, Brown, Karen D., Colussi, Dennis J., Leadley, Robert J., Bentley, Ross, Bostwick, Jeff, Kasiewski, Charles, Morgan, Suzanne

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Amido-(propyl and allyl)-hydroxybenzamidines : Development of achiral inhibitors of factor Xa von YONG GONG, PAULS, H. W, SPADA, A. P, CZEKAJ, M, GUYAN LIANG, CHU, V, COLUSSI, D. J, BROWN, K. D, JINGBO GAO

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Characterization of the bisphosphonate recognition site on hydroxyapatite using radioligand binding techniques with [14C]citric acid von JARVIS, M. F, BURNS, C. J, PAULS, H. W, ASSAL, A, KIM, J. S, CHENEY, D. L, YOUSSEFYEH, R. D

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Solid-phase parallel synthesis of azarene pyrrolidinones as factor Xa inhibitors von Gong, Y, Becker, M, Choi-Sledeski, Y M, Davis, R S, Salvino, J M, Chu, V, Brown, K D, Pauls, H W

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Chiral building blocks for amphotericin B von Liang, David, Pauls, Henry W, Fraser-Reid, Bert, Georges, Michael, Mubarak, Azeez M, Jarosz, Slawomir

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Molecular Structures of Human Factor Xa Complexed with Ketopiperazine Inhibitors:  Preference for a Neutral Group in the S1 Pocket von Maignan, Sébastien, Guilloteau, Jean-Pierre, Choi-Sledeski, Yong Mi, Becker, Michael R, Ewing, William R, Pauls, Henry W, Spada, Alfred P, Mikol, Vincent

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New inhibitors of cysteine proteinases. Peptidyl acyloxymethyl ketones and the quiescent nucleofuge strategy von Smith, Roger A, Copp, Leslie J, Coles, Peter J, Pauls, Henry W, Robinson, Valerie J, Spencer, Robin W, Heard, Stephen B, Krantz, Allen

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A Convenient Synthesis of Heteroaryl Benzoic Acids via Suzuki Reaction von Gong, Yong, Pauls, Henry W.

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Design and Structure−Activity Relationships of Potent and Selective Inhibitors of Blood Coagulation Factor Xa von Ewing, William R, Becker, Michael R, Manetta, Vincent E, Davis, Roderick S, Pauls, Henry W, Mason, Helen, Choi-Sledeski, Yong Mi, Green, Daniel, Cha, Don, Spada, Alfred P, Cheney, Daniel L, Mason, Jonathan S, Maignan, Sebastien, Guilloteau, Jean-Pierre, Brown, Karen, Colussi, Dennis, Bentley, Ross, Bostwick, Jeff, Kasiewski, Charles J, Morgan, Suzanne R, Leadley, Robert J, Dunwiddie, Christopher T, Perrone, Mark H, Chu, Valeria

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Simple One-Pot Synthesis of 2-Acylmethylidene-3-methylthiazolines von Pauls, Henry W., Krantz, Allen

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IRREVERSIBLE INHIBITION OF TRANSGLUTAMINASES BY SULFONIUM METHYLKETONES - OPTIMIZATION OF SPECIFICITY AND POTENCY WITH OMEGA-AMINOACYL SPACERS von PLIURA, DH, BONAVENTURA, BJ, PAULS, HW, KILLACKEY, JF, KRANTZ, A

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2-(Peptidamido)-cyclobutanones: A novel strategy for the inhibition of serine elastases von Pauls, Henry W., Cheng, Bill, Reid, Lorne S.

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Theory and Algorithm for Rule Base Refinement von Zhuge, Hai, Sun, Yunchuan, Guo, Weiyu

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Design and Implementation of Personality of Humanoids in Human Humanoid Non-verbal Interaction von Okuno, Hiroshi G., Nakadai, Kazuhiro, Kitano, Hiroaki

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Preserving Diversity in Particle Swarm Optimisation von Hendtlass, Tim

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