Selective inhibitors of JAK1 targeting an isoform-restricted allosteric cysteine von Kavanagh, Madeline E., Horning, Benjamin D., Khattri, Roli, Roy, Nilotpal, Lu, Justine P., Whitby, Landon R., Ye, Elva, Brannon, Jaclyn C., Parker, Albert, Chick, Joel M., Eissler, Christie L., Wong, Ashley J., Rodriguez, Joe L., Rodiles, Socorro, Masuda, Kim, Teijaro, John R., Simon, Gabriel M., Patricelli, Matthew P., Cravatt, Benjamin F.

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Characterization of a selective inhibitor of the Parkinson's disease kinase LRRK2 von Alessi, Dario R, Gray, Nathanael S, Deng, Xianming, Dzamko, Nicolas, Prescott, Alan, Davies, Paul, Liu, Qingsong, Yang, Qingkai, Lee, Jiing-Dwan, Patricelli, Matthew P, Nomanbhoy, Tyzoon K

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Functional Interplay between Caspase Cleavage and Phosphorylation Sculpts the Apoptotic Proteome von Dix, Melissa M., Simon, Gabriel M., Wang, Chu, Okerberg, Eric, Patricelli, Matthew P., Cravatt, Benjamin F.

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Functional Interrogation of the Kinome Using Nucleotide Acyl Phosphates von Patricelli, Matthew P, Szardenings, A. Katrin, Liyanage, Marek, Nomanbhoy, Tyzoon K, Wu, Min, Weissig, Helge, Aban, Arwin, Chun, Doris, Tanner, Stephen, Kozarich, John W

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Reversible inhibitor of p97, DBeQ, impairs both ubiquitin-dependent and autophagic protein clearance pathways von Chou, Tsui-Fen, Brown, Steve J., Minond, Dmitriy, Nordin, Brian E., Li, Kelin, Jones, Amanda C., Chase, Peter, Porubsky, Patrick R., Stoltz, Brian M., Schoenen, Frank J., Patricelli, Matthew P., Hodder, Peter, Rosen, Hugh, Deshaies, Raymond J., King, Randy

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Supersensitivity to Anandamide and Enhanced Endogenous Cannabinoid Signaling in Mice Lacking Fatty Acid Amide Hydrolase von Cravatt, Benjamin F., Demarest, Kristin, Patricelli, Matthew P., Bracey, Michael H., Giang, Dan K., Martin, Billy R., Lichtman, Aron H.

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Characterization of Torin2, an ATP-Competitive Inhibitor of mTOR, ATM, and ATR von QINGSONG LIU, CHUNXIAO XU, ERCAN, Dalia, NIEPEL, Mario, THOREEN, Carson C, KANG, Seong A, PATRICELLI, Matthew P, YUCHUAN WANG, TUPPER, Tanya, ALTABEF, Abigail, KAWAMURA, Hidemasa, HELD, Kathryn D, KIRUBAKARAN, Sivapriya, CHOU, Danny M, ELLEDGE, Stephen J, JANNE, Pasi A, WONG, Kwok-Kin, SABATINI, David M, GRAY, Nathanael S, XIN ZHANG, HUR, Wooyoung, YAN LIU, KWIATKOWSKI, Nicholas P, JINHUA WANG, WESTOVER, Kenneth D, PENG GAO

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Fragment-based covalent ligand discovery von Lu, Wenchao, Kostic, Milka, Zhang, Tinghu, Che, Jianwei, Patricelli, Matthew P, Jones, Lyn H, Chouchani, Edward T, Gray, Nathanael S

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Pharmacological Inhibition of BMK1 Suppresses Tumor Growth through Promyelocytic Leukemia Protein von Yang, Qingkai, Deng, Xianming, Lu, Bingwen, Cameron, Michael, Fearns, Colleen, Patricelli, Matthew P., Yates, John R., Gray, Nathanael S., Lee, Jiing-Dwan

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Activity-Based Protein Profiling: The Serine Hydrolases von Liu, Yongsheng, Patricelli, Matthew P., Cravatt, Benjamin F.

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Targeting KRAS Mutant Cancers with a Covalent G12C-Specific Inhibitor von Janes, Matthew R., Zhang, Jingchuan, Li, Lian-Sheng, Hansen, Rasmus, Peters, Ulf, Guo, Xin, Chen, Yuching, Babbar, Anjali, Firdaus, Sarah J., Darjania, Levan, Feng, Jun, Chen, Jeffrey H., Li, Shuangwei, Li, Shisheng, Long, Yun O., Thach, Carol, Liu, Yuan, Zarieh, Ata, Ely, Tess, Kucharski, Jeff M., Kessler, Linda V., Wu, Tao, Yu, Ke, Wang, Yi, Yao, Yvonne, Deng, Xiaohu, Zarrinkar, Patrick P., Brehmer, Dirk, Dhanak, Dashyant, Lorenzi, Matthew V., Hu-Lowe, Dana, Patricelli, Matthew P., Ren, Pingda, Liu, Yi

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Pathophysiological significance and therapeutic targeting of germinal center kinase in diffuse large B-cell lymphoma von Matthews, Julie Marie, Bhatt, Shruti, Patricelli, Matthew P., Nomanbhoy, Tyzoon K., Jiang, Xiaoyu, Natkunam, Yasodha, Gentles, Andrew J., Martinez, Ezequiel, Zhu, Daxing, Chapman, Jennifer Rose, Cortizas, Elena, Shyam, Ragini, Chinichian, Shideh, Advani, Ranjana, Tan, Li, Zhang, Jianming, Choi, Hwan Geun, Tibshirani, Robert, Buhrlage, Sara J., Gratzinger, Dita, Verdun, Ramiro, Gray, Nathanael S., Lossos, Izidore S.

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Selective Inhibition of Oncogenic KRAS Output with Small Molecules Targeting the Inactive State von Patricelli, Matthew P, Janes, Matthew R, Li, Lian-Sheng, Hansen, Rasmus, Peters, Ulf, Kessler, Linda V, Chen, Yuching, Kucharski, Jeff M, Feng, Jun, Ely, Tess, Chen, Jeffrey H, Firdaus, Sarah J, Babbar, Anjali, Ren, Pingda, Liu, Yi

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Profiling Protein Kinases and Other ATP Binding Proteins in Arabidopsis Using Acyl-ATP Probes von Villamor, Joji Grace, Kaschani, Farnusch, Colby, Tom, Oeljeklaus, Julian, Zhao, David, Kaiser, Markus, Patricelli, Matthew P., van der Hoorn, Renier A.L.

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Direct visualization of serine hydrolase activities in complex proteomes using fluorescent active site-directed probes von Patricelli, Matthew P., Giang, Dan K., Stamp, Lisa M., Burbaum, Jonathan J.

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Identification of a Tumor Specific, Active-Site Mutation in Casein Kinase 1α by Chemical Proteomics von Okerberg, Eric S, Hainley, Anna, Brown, Heidi, Aban, Arwin, Alemayehu, Senait, Shih, Ann, Wu, Jane, Patricelli, Matthew P, Kozarich, John W, Nomanbhoy, Tyzoon, Rosenblum, Jonathan S

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Correction: Identification of a Tumor Specific, Active-Site Mutation in Casein Kinase 1α by Chemical Proteomics von Okerberg, Eric S, Hainley, Anna, Brown, Heidi, Aban, Arwin, Alemayehu, Senait, Shih, Ann, Wu, Jane, Patricelli, Matthew P, Kozarich, John W, Nomanbhoy, Tyzoon, Rosenblum, Jonathan S

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Mapping Enzyme Active Sites in Complex Proteomes von Adam, Gregory C, Burbaum, Jonathan, Kozarich, John W, Patricelli, Matthew P, Cravatt, Benjamin F

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Exceptionally Potent Inhibitors of Fatty Acid Amide Hydrolase: The Enzyme Responsible for Degradation of Endogenous Oleamide and Anandamide von Boger, Dale L., Sato, Haruhiko, Lerner, Aaron E., Hedrick, Michael P., Fecik, Robert A., Miyauchi, Hiroshi, Wilkie, Gordon D., Austin, Bryce J., Patricelli, Matthew P., Cravatt, Benjamin F.

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High-Resolution Functional Proteomics by Active-Site Peptide Profiling von Okerberg, Eric S., Wu, Jiangyue, Zhang, Baohong, Samii, Babak, Blackford, Kelly, Winn, David T., Shreder, Kevin R., Burbaum, Jonathan J., Patricelli, Matthew P., Stubbe, JoAnne

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