Three Mechanistically Distinct Kinase Assays Compared: Measurement of Intrinsic ATPase Activity Identified the Most Comprehensive Set of ITK Inhibitors von Kashem, Mohammed A., Nelson, Richard M., Yingling, Jeffrey D., Pullen, Steven S., Prokopowicz, III, Anthony S., Jones, Jessi Wildeson, Wolak, John P., Rogers, George R., Morelock, Maurice M., Snow, Roger J., Homon, Carol Ann, Jakes, Scott

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Discovery of potent and selective PKC-θ inhibitors von Cywin, Charles L., Dahmann, Georg, Prokopowicz, Anthony S., Young, Erick R.R., Magolda, Ronald L., Cardozo, Mario G., Cogan, Derek A., DiSalvo, Darren, Ginn, John D., Kashem, Mohammed A., Wolak, John P., Homon, Carol A., Farrell, Thomas M., Grbic, Heather, Hu, Hanbo, Kaplita, Paul V., Liu, Lisa H., Spero, Denice M., Jeanfavre, Deborah D., O’Shea, Kathy M., White, Della M., Woska, Joseph R., Brown, Maryanne L.

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Discovery of 2-Phenylamino-imidazo[4,5-h]isoquinolin-9-ones:  A New Class of Inhibitors of Lck Kinase von Snow, Roger J, Cardozo, Mario G, Morwick, Tina M, Busacca, Carl A, Dong, Yong, Eckner, Robert J, Jacober, Stephen, Jakes, Scott, Kapadia, Suresh, Lukas, Susan, Panzenbeck, Maret, Peet, Gregory W, Peterson, Jeffrey D, Prokopowicz, Anthony S, Sellati, Rosemarie, Tolbert, Robert M, Tschantz, Matt A, Moss, Neil

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Optimization of 2-Phenylaminoimidazo[4,5-h]isoquinolin-9-ones:  Orally Active Inhibitors of lck Kinase von Goldberg, Daniel R, Butz, Tanja, Cardozo, Mario G, Eckner, Robert J, Hammach, Abdelhakim, Huang, Jessica, Jakes, Scott, Kapadia, Suresh, Kashem, Mohammed, Lukas, Susan, Morwick, Tina M, Panzenbeck, Maret, Patel, Usha, Pav, Susan, Peet, Gregory W, Peterson, Jeffrey D, Prokopowicz, Anthony S, Snow, Roger J, Sellati, Rosemarie, Takahashi, Hidenori, Tan, Jonathan, Tschantz, Matt A, Wang, Xiao-Jun, Wang, Yong, Wolak, John, Xiong, Pla, Moss, Neil

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4-Trifloxy-9-SEM-β-Carboline:  Preparation and Synthetic Utility von Busacca, Carl A, Eriksson, Magnus C, Dong, Yong, Prokopowicz, Anthony S, Salvagno, Annette M, Tschantz, Matt A

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Isoquinolinone synthesis by SNAr reaction: a versatile route to imidazo[4,5-h]isoquinolin-9-ones von Snow, Roger J., Butz, Tanja, Hammach, Abdelhakim, Kapadia, Suresh, Morwick, Tina M., Prokopowicz, Anthony S., Takahashi, Hidenori, Tan, Jonathan D., Tschantz, Matt A., Wang, Xiao-Jun

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Isoquinolinone synthesis by S NAr reaction: a versatile route to imidazo[4,5- h]isoquinolin-9-ones von Snow, Roger J., Butz, Tanja, Hammach, Abdelhakim, Kapadia, Suresh, Morwick, Tina M., Prokopowicz, Anthony S., Takahashi, Hidenori, Tan, Jonathan D., Tschantz, Matt A., Wang, Xiao-Jun

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Rho kinase inhibitors von Liu, Weimin, Wu, Frank, Bosanac, Todd, Shih, Cheng-Kon, Young, Erick Richard, Ginn, John David, Turner, Michael Robert, Prokopowicz, Anthony S, Hickey, Eugene Richard, Schlyer, Sabine K, Snow, Roger John, Kirrane, Jr., Thomas Martin

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Addition reactions of cyclic s-trans-enaminones with Grignard reagents von Shawe, Thomas T., Hansen, Darren B., Peet, Kelly Ann, Prokopowicz, Anthony S., Robinson, Patrice M., Cannon, Annatina, Dougherty, Kathleen E., Ross, Andrew A., Landino, Linda M.

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RHO KINASE INHIBITORS von BOSANAC, Todd, KIRRANE, Thomas, Martin, YOUNG, Erick, Richard, SHIH, Cheng-kon, SCHLYER, Sabine, K, LIU, Weimin, TURNER, Michael, Robert, HICKEY, Eugene, Richard, SNOW, Roger, John, PROKOPOWICZ, Anthony, S, WU, Frank, GINN, John, David

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RHO KINASE INHIBITORS von Liu, Weimin, Wu, Frank, Bosanac, Todd, Shih, Cheng-Kon, Young, Erick Richard, Kirrane, JR., Thomas Martin, Ginn, John David, Turner, Michael Robert, Prokopowicz, Anthony S, Hickey, Eugene Richard, Schlyer, Sabine K, Snow, Roger John

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FLUORESCENT PROBES FOR USE IN PROTEIN KINASE INHIBITOR BINDING ASSAY von JAKES, SCOTT, BROWN, MARTHA PRISCILLA, JONES, JESSI WILDESON, LABADIA, MARK E, PROKOPOWICZ, ANTHONY S

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RHO KINASE INHIBITORS von Kirrane, JR. Thomas Martin, Wu Frank, Young Erick Richard, Ginn John David, Turner Michael Robert, Bosanac Todd, Snow Roger John, Prokopowicz Anthony S, Shih Cheng-Kon, Schlyer Sabine K, Liu Weimin, Hickey Eugene Richard

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RHO KINASE INHIBITORS von WU FRANK, HICKEY EUGENE RICHARD, PROKOPOWICZ ANTHONY S, SHIH CHENG-KON, BOSANAC TODD, YOUNG ERICK RICHARD, KIRRANE, JR. THOMAS MARTIN, GINN JOHN DAVID, LIU WEIMIN, SCHLYER SABINE K, SNOW ROGER JOHN, TURNER MICHAEL ROBERT

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PYRAZINE COMPOUNDS, THEIR USE AND METHODS OF PREPARATION von MORWICK, TINA, MARIE, MAO, WANG, PROKOPOWICZ, ANTHONY, S

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RHO KINASE INHIBITORS von WU FRANK, HICKEY EUGENE RICHARD, PROKOPOWICZ ANTHONY S, SHIH CHENG-KON, BOSANAC TODD, YOUNG ERICK RICHARD, KIRRANE, JR. THOMAS MARTIN, GINN JOHN DAVID, LIU WEIMIN, SCHLYER SABINE K, SNOW ROGER JOHN, TURNER MICHAEL ROBERT

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RHO KINASE INHIBITORS von LIU, WEIMIN, BOSANAC, TODD, KIRRANE, THOMAS MARTIN, SHIH, CHENG-KON, SNOW, ROGER JOHN, YOUNG, ERICK RICHARD, WU, FRANK, HICKEY, EUGENE RICHARD, GINN, JOHN DAVID, PROKOPOWICZ, ANTHONY S, SCHLYER, SABINE K, TURNER, MICHAEL ROBERT

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PYRAZINE COMPOUNDS, THEIR USE AND METHODS OF PREPARATION von MORWICK, TINA, MARIE, MAO, WANG, PROKOPOWICZ, ANTHONY, S

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PYRAZINE COMPOUNDS, THEIR USE AND METHODS OF PREPARATION von MORWICK, TINA MARIE, MAO, WANG, PROKOPOWICZ, ANTHONY S

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Isoquinolinone Rho kinase inhibitors von WU FRANK, HICKEY EUGENE RICHARD, PROKOPOWICZ ANTHONY S, SHIH CHENG-KON, BOSANAC TODD, YOUNG ERICK RICHARD, KIRRANE, JR. THOMAS MARTIN, GINN JOHN DAVID, LIU WEIMIN, SCHLYER SABINE K, SNOW ROGER JOHN, TURNER MICHAEL ROBERT

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