The evolution of amidine-based brain penetrant BACE1 inhibitors von Oehlrich, Daniel, Prokopcova, Hana, Gijsen, Harrie J.M.

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Palladium(0)-Catalyzed, Copper(I)-Mediated Coupling of Boronic Acids with Cyclic Thioamides. Selective Carbon−Carbon Bond Formation for the Functionalization of Heterocycles von Prokopcová, Hana, Kappe, C. Oliver

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Liebeskind-Srogl C----C Cross-Coupling Reaction von Prokopcová, Hana, Kappe, C. Oliver

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Desulfitative Carbon-Carbon Cross-Coupling of Thioamide Fragments with Boronic Acids von Prokopcová, Hana, Kappe, C. Oliver

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Structural Basis for Inhibition of Eg5 by Dihydropyrimidines: Stereoselectivity of Antimitotic Inhibitors Enastron, Dimethylenastron and Fluorastrol von Kaan, Hung Yi Kristal, Ulaganathan, Venkatasubramanian, Rath, Oliver, Prokopcová, Hana, Dallinger, Doris, Kappe, C. Oliver, Kozielski, Frank

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Structure-Activity Relationships and Molecular Docking of Novel Dihydropyrimidine-Based Mitotic Eg5 Inhibitors von Prokopcová, Hana, Dallinger, Doris, Uray, Georg, Kaan, Hung Yi Kristal, Ulaganathan, Venkatasubramanian, Kozielski, Frank, Laggner, Christian, Kappe, C. Oliver

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Synthesis of 5-Aroyldihydropyrimidinones via Liebeskind-Srogl Thiol Ester-Boronic Acid Cross-Couplings von Prokopcová, Hana, Pisani, Leonardo, Kappe, C. Oliver

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4-Cyano-6,7-dimethoxycarbostyrils with Solvent- and pH-Independent High Fluorescence Quantum Yields and Emission Maxima von Ahvale, Appasaheb B., Prokopcová, Hana, Šefčovičová, Jana, Steinschifter, Waltraud, Täubl, Anna E., Uray, Georg, Stadlbauer, Wolfgang

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Copper-Catalyzed C----C Coupling of Thiol Esters and Boronic Acids under Aerobic Conditions von Prokopcová, Hana, Kappe, C. Oliver

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Ruthenium‐Catalyzed Reductive Arylation of N‐(2‐Pyridinyl)amides with Isopropanol and Arylboronate Esters von Ronson, Thomas O., Renders, Evelien, Van Steijvoort, Ben F., Wang, Xubin, Wybon, Clarence C. D., Prokopcová, Hana, Meerpoel, Lieven, Maes, Bert U. W.

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The Role of the Alcohol and Carboxylic Acid in Directed Ruthenium-Catalyzed C(sp3)H α-Alkylation of Cyclic Amines von Bergman, Sheba D., Storr, Thomas E., Prokopcová, Hana, Aelvoet, Karel, Diels, Gaston, Meerpoel, Lieven, Maes, Bert U. W.

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A Bayesian Approach to Kinetic Modeling of Accelerated Stability Studies and Shelf Life Determination von Chau, Joris, Altan, Stan, Burggraeve, Anneleen, Coppenolle, Hans, Kifle, Yimer Wasihun, Prokopcova, Hana, Van Daele, Timothy, Sterckx, Hans

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1,4-Oxazine β‑Secretase 1 (BACE1) Inhibitors: From Hit Generation to Orally Bioavailable Brain Penetrant Leads von Rombouts, Frederik J. R, Tresadern, Gary, Delgado, Oscar, Martínez-Lamenca, Carolina, Van Gool, Michiel, García-Molina, Aránzazu, Alonso de Diego, Sergio A, Oehlrich, Daniel, Prokopcova, Hana, Alonso, José Manuel, Austin, Nigel, Borghys, Herman, Van Brandt, Sven, Surkyn, Michel, De Cleyn, Michel, Vos, Ann, Alexander, Richard, Macdonald, Gregor, Moechars, Dieder, Gijsen, Harrie, Trabanco, Andrés A

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Optimization of 1,4-Oxazine β‑Secretase 1 (BACE1) Inhibitors Toward a Clinical Candidate von Gijsen, Harrie J. M, Alonso de Diego, Sergio A, De Cleyn, Michel, García-Molina, Aránzazu, Macdonald, Gregor J, Martínez-Lamenca, Carolina, Oehlrich, Daniel, Prokopcova, Hana, Rombouts, Frederik J. R, Surkyn, Michel, Trabanco, Andrés A, Van Brandt, Sven, Van den Bossche, Dries, Van Gool, Michiel, Austin, Nigel, Borghys, Herman, Dhuyvetter, Deborah, Moechars, Diederik

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Microwave-assisted one-pot diboration/Suzuki cross-couplings. A rapid route to tetrasubstituted alkenes von Prokopcová, Hana, Ramírez, Jesús, Fernández, Elena, Kappe, C. Oliver

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Evaluation of a Series of β‑Secretase 1 Inhibitors Containing Novel Heteroaryl-Fused-Piperazine Amidine Warheads von Oehlrich, Daniel, Peschiulli, Aldo, Tresadern, Gary, Van Gool, Michiel, Vega, Juan Antonio, De Lucas, Ana Isabel, Alonso de Diego, Sergio A, Prokopcova, Hana, Austin, Nigel, Van Brandt, Sven, Surkyn, Michel, De Cleyn, Michel, Vos, Ann, Rombouts, Frederik J. R, Macdonald, Gregor, Moechars, Dieder, Gijsen, Harrie J. M, Trabanco, Andrés A

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Correction to Optimization of 1,4-Oxazine β‑Secretase 1 (BACE1) Inhibitors Toward a Clinical Candidate von Gijsen, Harrie J. M, Alonso de Diego, Sergio A, De Cleyn, Michel, García-Molina, Aránzazu, Macdonald, Gregor J, Martinez-Lamenca, Carolina, Oehlrich, Daniel, Prokopcova, Hana, Rombouts, Frederik J. R, Surkyn, Michel, Trabanco, Andrés A, Van Brandt, Sven, Van den Bossche, Dries, Van Gool, Michiel, Austin, Nigel, Borghys, Herman, Dhuyvetter, Deborah, Urmaliya, Vijay, Teisman, Ard, Moechars, Diederik

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The Role of the Alcohol and Carboxylic Acid in Directed Ruthenium-Catalyzed C(sp3)H [alpha]-Alkylation of Cyclic Amines von Bergman, Sheba D, Storr, Thomas E, Prokopcova, Hana, Aelvoet, Karel, Diels, Gaston, Meerpoel, Lieven, Maes, Bert U W

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C-2 Arylation of Piperidines through Directed Transition-Metal-Catalyzed sp3 CH Activation von Prokopcova, Hana, Bergman, Sheba D, Aelvoet, Karel, Smout, Veerle, Herrebout, Wouter, VanderVeken, Benjamin, Meerpoel, Lieven, Maes, Bert U W

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C-2 Arylation of Piperidines through Directed Transition-Metal-Catalyzed sp3 CH Activation von Prokopcová, Hana, Bergman, Sheba D., Aelvoet, Karel, Smout, Veerle, Herrebout, Wouter, Van der Veken, Benjamin, Meerpoel, Lieven, Maes, Bert U. W.

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