Palladium(II)‐Catalyzed Site‐Selective C(sp3)−H Alkynylation of Oligopeptides: A Linchpin Approach for Oligopeptide–Drug Conjugation von Liu, Tao, Qiao, Jennifer X., Poss, Michael A., Yu, Jin‐Quan

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Decarboxylative Peptide Macrocyclization through Photoredox Catalysis von McCarver, Stefan J., Qiao, Jennifer X., Carpenter, Joseph, Borzilleri, Robert M., Poss, Michael A., Eastgate, Martin D., Miller, Michael M., MacMillan, David W. C.

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Inhibition of influenza virus replication via small molecules that induce the formation of higher-order nucleoprotein oligomers von Gerritz, Samuel W, Cianci, Christopher, Kim, Sean, Pearce, Bradley C, Deminie, Carol, Discotto, Linda, McAuliffe, Brian, Minassian, Beatrice F, Shi, Shuhao, Zhu, Shirong, Zhai, Weixu, Pendri, Annapurna, Li, Guo, Poss, Michael A, Edavettal, Suzanne, McDonnell, Patricia A, Lewis, Hal A, Maskos, Klaus, Mörtl, Mario, Kiefersauer, Reiner, Steinbacher, Stefan, Baldwin, Eric T, Metzler, William, Bryson, James, Healy, Matthew D, Philip, Thomas, Zoeckler, Mary, Schartman, Richard, Sinz, Michael, Leyva-Grado, Victor H, Hoffmann, Hans-Heinrich, Langley, David R, Meanwell, Nicholas A, Krystal, Mark

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Formation of α-chiral centers by asymmetric β-C(sp3)-H arylation, alkenylation, and alkynylation von Wu, Qing-Feng, Shen, Peng-Xiang, He, Jian, Wang, Xiao-Bing, Zhang, Forrest, Shao, Qian, Zhu, Ru-Yi, Mapelli, Claudio, Qiao, Jennifer X, Poss, Michael A, Yu, Jin-Quan

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Ligand-Enabled β‑C(sp3)–H Olefination of Free Carboxylic Acids von Zhuang, Zhe, Yu, Chang-Bin, Chen, Gang, Wu, Qing-Feng, Hsiao, Yi, Joe, Candice L, Qiao, Jennifer X, Poss, Michael A, Yu, Jin-Quan

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Ligand-Enabled β‑C–H Arylation of α‑Amino Acids Using a Simple and Practical Auxiliary von Chen, Gang, Shigenari, Toshihiko, Jain, Pankaj, Zhang, Zhipeng, Jin, Zhong, He, Jian, Li, Suhua, Mapelli, Claudio, Miller, Michael M, Poss, Michael A, Scola, Paul M, Yeung, Kap-Sun, Yu, Jin-Quan

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Ligand Enabled Pd(II)-Catalyzed γ‑C(sp3)–H Lactamization of Native Amides von Liu, Shuang, Zhuang, Zhe, Qiao, Jennifer X, Yeung, Kap-Sun, Su, Shun, Cherney, Emily C, Ruan, Zheming, Ewing, William R, Poss, Michael A, Yu, Jin-Quan

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A Selection of Macrocyclic Peptides That Bind STING From an mRNA‐Display Library With Split Degenerate Codons von Lin, Chi‐Wang, Harner, Mary J., Douglas, Andrew E., Lafont, Virginie, Yu, Fei, Lee, Ving G., Poss, Michael A., Swain, Joanna F., Wright, Martin, Lipovšek, Daša

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Exploration of macrocyclic peptide binders to the extracellular CRD domain of human receptor tyrosine kinase-like orphan receptor 1 (ROR1) von Qiao, Jennifer X., Witmer, Mark R., Lee, Ving, Wang, Tammy C., Reid, Patrick C., Arioka, Yuki, Farr, Glen, Hill-Drzewi, Melissa, Schweizer, Liang, Yamniuk, Aaron, Cheng, Lin, Abramczyk, Bozena, Corbett, Martin, Calambur, Deepa, Szapiel, Nicolas, Ryseck, Rolf, Ponath, Paul, Poss, Michael A., Carter, Percy

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CITU: A Peptide and Decarboxylative Coupling Reagent von deGruyter, Justine N., Malins, Lara R., Wimmer, Laurin, Clay, Khalyd J., Lopez-Ogalla, Javier, Qin, Tian, Cornella, Josep, Liu, Zhiqing, Che, Guanda, Bao, Denghui, Stevens, Jason M., Qiao, Jennifer X., Allen, Martin P., Poss, Michael A., Baran, Phil S.

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Long-Acting Tumor-Activated Prodrug of a TGFβR Inhibitor von Zhang, Yong, Parrish, Karen E, Tortolani, David R, Poss, Michael A, Huang, Audris, Wan, Honghe, Purandare, Ashok V, Donnell, Andrew F, Kempson, James, Hou, Xiaoping, Pawluczyk, Joseph, Yip, Shiuhang, Luk, Emily, Raghavan, Nimmi, Swanson, Jesse, Smalley, James, Murtaza, Anwar, Yang, Zheng, Augustine-Rauch, Karen, Lombardo, Louis J, Borzilleri, Robert

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Discovery of Aminothiazole Inhibitors of Cyclin-Dependent Kinase 2:  Synthesis, X-ray Crystallographic Analysis, and Biological Activities von Kim, Kyoung Soon, Kimball, S. David, Misra, Raj N, Rawlins, David B, Hunt, John T, Xiao, Hai-Yun, Lu, Songfeng, Qian, Ligang, Han, Wen-Ching, Shan, Weifang, Mitt, Toomas, Cai, Zhen-Wei, Poss, Michael A, Zhu, Hong, Sack, John S, Tokarski, John S, Chang, Chieh Ying, Pavletich, Nikola, Kamath, Amrita, Humphreys, William G, Marathe, Punit, Bursuker, Isia, Kellar, Kristen A, Roongta, Urvashi, Batorsky, Roberta, Mulheron, Janet G, Bol, David, Fairchild, Craig R, Lee, Francis Y, Webster, Kevin R

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Core exploration in optimization of chemokine receptor CCR4 antagonists von Purandare, Ashok V., Wan, Honghe, Somerville, John E., Burke, Christine, Vaccaro, Wayne, Yang, XiaoXia, McIntyre, Kim W., Poss, Michael A.

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Synthesis of Fmoc-Protected Arylphenylalanines (Bip Derivatives) via Nonaqueous Suzuki-Miyaura Cross-Coupling Reactions von Qiao, Jennifer X, Fraunhoffer, Kenneth J, Hsiao, Yi, Li, Yi-Xin, Wang, Chunlei, Wang, Tammy C, Poss, Michael A

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Identification of 2‑Pyridinylindole-Based Dual Antagonists of Toll-like Receptors 7 and 8 (TLR7/8) von Sreekantha, Ratna Kumar, Mussari, Christopher P., Dodd, Dharmpal S., Pasunoori, Laxman, Hegde, Subramanya, Posy, Shana L., Critton, David, Ruepp, Stefan, Subramanian, Murali, Salter-Cid, Luisa M., Tagore, Debarati Mazumder, Sarodaya, Sanket, Dudhgaonkar, Shailesh, Poss, Michael A., Schieven, Gary L., Carter, Percy H., Macor, John E., Dyckman, Alaric J.

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Decarboxylative Peptide Macrocyclization through Photoredox Catalysis von McCarver, Stefan J., Qiao, Jennifer X., Carpenter, Joseph, Borzilleri, Robert M., Poss, Michael A., Eastgate, Martin D., Miller, Michael M., MacMillan, David W. C.

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Identification of a Potent, Selective, and Efficacious Phosphatidylinositol 3‑Kinase δ (PI3Kδ) Inhibitor for the Treatment of Immunological Disorders von Liu, Qingjie, Shi, Qing, Marcoux, David, Batt, Douglas G, Cornelius, Lyndon, Qin, Lan-Ying, Ruan, Zheming, Neels, James, Beaudoin-Bertrand, Myra, Srivastava, Anurag S, Li, Ling, Cherney, Robert J, Gong, Hua, Watterson, Scott H, Weigelt, Carolyn, Gillooly, Kathleen M, McIntyre, Kim W, Xie, Jenny H, Obermeier, Mary T, Fura, Aberra, Sleczka, Bogdan, Stefanski, Kevin, Fancher, R. M, Padmanabhan, Shweta, RP, Thatipamula, Kundu, Ipsit, Rajareddy, Kallem, Smith, Rodney, Hennan, James K, Xing, Dezhi, Fan, Jingsong, Levesque, Paul C, Ruan, Qian, Pitt, Sidney, Zhang, Rosemary, Pedicord, Donna, Pan, Jie, Yarde, Melissa, Lu, Hao, Lippy, Jonathan, Goldstine, Christine, Skala, Stacey, Rampulla, Richard A, Mathur, Arvind, Gupta, Anuradha, Arunachalam, Pirama Nayagam, Sack, John S, Muckelbauer, Jodi K, Cvijic, Mary Ellen, Salter-Cid, Luisa M, Bhide, Rajeev S, Poss, Michael A, Hynes, John, Carter, Percy H, Macor, John E, Ruepp, Stefan, Schieven, Gary L, Tino, Joseph A

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Discovery and SAR of pyrrolo[2,1-f][1,2,4]triazin-4-amines as potent and selective PI3Kδ inhibitors von Bhide, Rajeev S., Neels, James, Qin, Lan-Ying, Ruan, Zheming, Stachura, Sylwia, Weigelt, Carolyn, Sack, John S., Stefanski, Kevin, Gu, Xiaomei, Xie, Jenny H., Goldstine, Christine B., Skala, Stacey, Pedicord, Donna L., Ruepp, Stefan, Dhar, T.G. Murali, Carter, Percy H., Salter-Cid, Luisa M., Poss, Michael A., Davies, Paul

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Frontispiz: A Selection of Macrocyclic Peptides That Bind STING From an mRNA‐Display Library With Split Degenerate Codons von Lin, Chi‐Wang, Harner, Mary J., Douglas, Andrew E., Lafont, Virginie, Yu, Fei, Lee, Ving G., Poss, Michael A., Swain, Joanna F., Wright, Martin, Lipovšek, Daša

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The synthesis of novel heteroaryl-fused 7,8,9,10-tetrahydro-6H-azepino[1,2-a]indoles, 4-oxo-2,3-dihydro-1H-[1,4]diazepino[1,7-a]indoles and 1,2,4,5-tetrahydro-[1,4]oxazepino[4,5-a]... von Ding, Min, He, Feng, Poss, Michael A, Rigat, Karen L, Wang, Ying-Kai, Roberts, Susan B, Qiu, Dike, Fridell, Robert A, Gao, Min, Gentles, Robert G

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