Small-molecule inhibitors of human mitochondrial DNA transcription von Bonekamp, Nina A., Peter, Bradley, Hillen, Hauke S., Felser, Andrea, Bergbrede, Tim, Choidas, Axel, Horn, Moritz, Unger, Anke, Di Lucrezia, Raffaella, Atanassov, Ilian, Li, Xinping, Koch, Uwe, Menninger, Sascha, Boros, Joanna, Habenberger, Peter, Giavalisco, Patrick, Cramer, Patrick, Denzel, Martin S., Nussbaumer, Peter, Klebl, Bert, Falkenberg, Maria, Gustafsson, Claes M., Larsson, Nils-Göran

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An Efficient Proteomics Method to Identify the Cellular Targets of Protein Kinase Inhibitors von Godl, Klaus, Wissing, Josef, Kurtenbach, Alexander, Habenberger, Peter, Blencke, Stephanie, Gutbrod, Heidrun, Salassidis, Kostadinos, Stein-Gerlach, Matthias, Missio, Andrea, Cotten, Matt, Daub, Henrik

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Systematic Kinase Inhibitor Profiling Identifies CDK9 as a Synthetic Lethal Target in NUT Midline Carcinoma von Brägelmann, Johannes, Dammert, Marcel A., Dietlein, Felix, Heuckmann, Johannes M., Choidas, Axel, Böhm, Stefanie, Richters, André, Basu, Debjit, Tischler, Verena, Lorenz, Carina, Habenberger, Peter, Fang, Zhizhou, Ortiz-Cuaran, Sandra, Leenders, Frauke, Eickhoff, Jan, Koch, Uwe, Getlik, Matthäus, Termathe, Martin, Sallouh, Muhammad, Greff, Zoltán, Varga, Zoltán, Balke-Want, Hyatt, French, Christopher A., Peifer, Martin, Reinhardt, H. Christian, Örfi, László, Kéri, György, Ansén, Sascha, Heukamp, Lukas C., Büttner, Reinhard, Rauh, Daniel, Klebl, Bert M., Thomas, Roman K., Sos, Martin L.

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Anti-leukemic effect of CDK9 inhibition in T-cell prolymphocytic leukemia von Johansson, Patricia, Dierichs, Laura, Klein-Hitpass, Ludger, Bergmann, Anke K., Möllmann, Michael, Menninger, Sascha, Habenberger, Peter, Klebl, Bert, Siveke, Jens T., Dührsen, Ulrich, Choidas, Axel, Dürig, Jan

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Identification of SRPK1 and SRPK2 as the Major Cellular Protein Kinases Phosphorylating Hepatitis B Virus Core Protein von Daub, Henrik, Blencke, Stephanie, Habenberger, Peter, Kurtenbach, Alexander, Dennenmoser, Julia, Wissing, Josef, Ullrich, Axel, Cotten, Matt

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Chemical Proteomic Analysis Reveals Alternative Modes of Action for Pyrido[2,3-d]pyrimidine Kinase Inhibitors von Wissing, Josef, Godl, Klaus, Brehmer, Dirk, Blencke, Stephanie, Weber, Martina, Habenberger, Peter, Stein-Gerlach, Matthias, Missio, Andrea, Cotten, Matt, Müller, Stefan, Daub, Henrik

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White Paper: Mimetics of Class 2 Tumor Suppressor Proteins as Novel Drug Candidates for Personalized Cancer Therapy von Dahl, Edgar, Villwock, Sophia, Habenberger, Peter, Choidas, Axel, Rose, Michael, Klebl, Bert M

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Negishi Cross‐Coupling in the Preparation of Benzyl Substituted Pyrrolopyrimidine Based CSF1R Inhibitors von Aarhus, Thomas I, Teksum, Vilde, Unger, Anke, Habenberger, Peter, Wolf, Alexander, Eickhoff, Jan, Klebl, Bert, Wolowczyk, Camilla, Bjørkøy, Geir, Sundby, Eirik, Hoff, Bård H

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Pyrrolopyrimidine based CSF1R inhibitors: Attempted departure from Flatland von Bjørnstad, Frithjof, Havik, Simen, Aarhus, Thomas Ihle, Mahdi, Iktedar, Unger, Anke, Habenberger, Peter, Degenhart, Carsten, Eickhoff, Jan, Klebl, Bert M., Sundby, Eirik, Hoff, Bård Helge

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Negishi Cross‐Coupling in the Preparation of Benzyl Substituted Pyrrolo[2,3‐d]pyrimidine Based CSF1R Inhibitors von Aarhus, Thomas I., Teksum, Vilde, Unger, Anke, Habenberger, Peter, Wolf, Alexander, Eickhoff, Jan, Klebl, Bert, Wolowczyk, Camilla, Bjørkøy, Geir, Sundby, Eirik, Hoff, Bård H.

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Synthesis and Development of Highly Selective Pyrrolo[2,3‑d]pyrimidine CSF1R Inhibitors Targeting the Autoinhibited Form von Aarhus, Thomas Ihle, Bjørnstad, Frithjof, Wolowczyk, Camilla, Larsen, Kristin Uhlving, Rognstad, Line, Leithaug, Trygve, Unger, Anke, Habenberger, Peter, Wolf, Alexander, Bjørkøy, Geir, Pridans, Clare, Eickhoff, Jan, Klebl, Bert, Hoff, Bård H., Sundby, Eirik

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Total Synthesis and Biological Evaluation of (−)-Englerin A and B: Synthesis of Analogues with Improved Activity Profile von Radtke, Lea, Willot, Matthieu, Sun, Hongyan, Ziegler, Slava, Sauerland, Stephanie, Strohmann, Carsten, Fröhlich, Roland, Habenberger, Peter, Waldmann, Herbert, Christmann, Mathias

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Discovery of a Novel Inhibitor of the Hedgehog Signaling Pathway through Cell‐based Compound Discovery and Target Prediction von Kremer, Lea, Schultz‐Fademrecht, Carsten, Baumann, Matthias, Habenberger, Peter, Choidas, Axel, Klebl, Bert, Kordes, Susanne, Schöler, Hans R., Sterneckert, Jared, Ziegler, Slava, Schneider, Gisbert, Waldmann, Herbert

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Identification of an (−)‐englerin A analogue, which antagonizes (−)‐englerin A at TRPC1/4/5 channels von Rubaiy, Hussein N, Seitz, Tobias, Hahn, Sven, Choidas, Axel, Habenberger, Peter, Klebl, Bert, Dinkel, Klaus, Nussbaumer, Peter, Waldmann, Herbert, Christmann, Mathias, Beech, David J

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SAMHD1 is recurrently mutated in T-cell prolymphocytic leukemia von Johansson, Patricia, Klein-Hitpass, Ludger, Choidas, Axel, Habenberger, Peter, Mahboubi, Bijan, Kim, Baek, Bergmann, Anke, Scholtysik, René, Brauser, Martina, Lollies, Anna, Siebert, Reiner, Zenz, Thorsten, Dührsen, Ulrich, Küppers, Ralf, Dürig, Jan

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CDK9 Inhibition with LDC526 Is an Effective Treatment for T-Cell Prolymphocytic Leukemia (T-PLL) in Vitro von Johansson, Patricia, Habenberger, Peter, Klein-Hitpass, Ludger, Duehrsen, Ulrich, Küppers, Ralf, Schultz-Fademrecht, Carsten, Choidas, Axel, Dürig, Jan

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Abstract 2823: Identification of highly selective inhibitors of cyclin-dependent kinase 12 von Choidas, Axel, Schultz-Fademrecht, Carsten, Degeenhardt, Carsten, Habenberger, Peter, Koch, Uwe, Eickhoff, Jan E., Greifenberg, Ann Kathrin, Nussbaumer, Peter, Geyer, Matthias, Klebl, Bert M.

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Abstract 1349: Systematic deconvolution of kinase inhibitor profiles identifies synthetic lethal targets in ERBB2-mutant and BRD4-NUT rearranged cancer von Braegelmann, Johannes, Habenberger, Peter, Dietlein, Felix, Heuckmann, Johannes M., Menninger, Sascha, Koch, Uwe, Choidas, Axel, Rauh, Daniel, Klebl, Bert, Sos, Martin L., Thomas, Roman K.

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Abstract 2997: Dynarrestin, a novel dynein inhibitor that does not block ciliogenesis von Baumann, Matthias, Höing, Susanne, Yeh, Ting-Yu, Martinez, Nancy, Habenberger, Peter, Kremer, Lea, Drexler, Hannes CA, Küchler, Philipp, Reinhardt, Peter, Choidas, Axel, Zischinsky, Mia-Lisa, Zischinsky, Gunther, Ketcham, Stephanie A., Wagner, Lydia, Nussbaumer, Peter, Ziegler, Slava, Klebl, Bert, Schroer, Trina, Schöler, Hans R., Waldmann, Herbert, Sterneckert, Jared L.

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Dynarrestin, a Novel Inhibitor of Cytoplasmic Dynein von Höing, Susanne, Yeh, Ting-Yu, Baumann, Matthias, Martinez, Nancy E., Habenberger, Peter, Kremer, Lea, Drexler, Hannes C.A., Küchler, Philipp, Reinhardt, Peter, Choidas, Axel, Zischinsky, Mia-Lisa, Zischinsky, Gunther, Nandini, Swaran, Ledray, Aaron P., Ketcham, Stephanie A., Reinhardt, Lydia, Abo-Rady, Masin, Glatza, Michael, King, Stephen J., Nussbaumer, Peter, Ziegler, Slava, Klebl, Bert, Schroer, Trina A., Schöler, Hans R., Waldmann, Herbert, Sterneckert, Jared

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