A potent and orally active HIV-1 integrase inhibitor von Egbertson, Melissa S., Moritz, H. Marie, Melamed, Jeffrey Y., Han, Wei, Perlow, Debra S., Kuo, Michelle S., Embrey, Mark, Vacca, Joseph P., Zrada, Matthew M., Cortes, Amanda R., Wallace, Audrey, Leonard, Yvonne, Hazuda, Daria J., Miller, Michael D., Felock, Peter J., Stillmock, Kara A., Witmer, Marc V., Schleif, William, Gabryelski, Lori J., Moyer, Gregory, Ellis, Joan D., Jin, Lixia, Xu, Wei, Braun, Matthew P., Kassahun, Kellem, Tsou, Nancy N., Young, Steven D.

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Renin inhibitors. Syntheses of subnanomolar, competitive, transition-state analog inhibitors containing a novel analog of statine von Boger, Joshua, Payne, Linda S, Perlow, Debra S, Lohr, Nancy S, Poe, Martin, Blaine, Edward H, Ulm, Edgar H, Schorn, Terry W, LaMont, Bruce I

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Synthesis of 9-fluorenylmethyloxycarbonyl-protected N-alkyl amino acids by reduction of oxazolidinones von Freidinger, Roger M, Hinkle, Jeffery S, Perlow, Debra S

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Use of N-Fmoc amino acid chlorides and activated 2-(fluorenylmethoxy)-5(4H)-oxazolones in solid-phase peptide synthesis. Efficient syntheses of highly N-alkylated cyclic hexapeptid... von Perlow, Debra S, Erb, Jill M, Gould, Norman P, Tung, Roger D, Freidinger, Roger M, Williams, Peter D, Veber, Daniel F

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Development of a novel class of cyclic hexapeptide oxytocin antagonists based on a natural product von Williams, Peter D, Bock, Mark G, Tung, Roger D, Garsky, Victor M, Perlow, Debra S, Erb, Jill M, Lundell, G. F, Gould, Norman P, Whitter, Willie L

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Renin inhibitors containing conformationally restricted P1-P1' dipeptide mimetics von Williams, Peter D, Perlow, Debra S, Payne, Linda S, Holloway, M. Katherine, Siegl, Peter K. S, Schorn, Terry W, Lynch, Robert J, Doyle, John J, Strouse, John F

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A super active cyclic hexapeptide analog of somatostatin von Veber, Daniel F., Saperstein, Richard, Nutt, Ruth F., Freidinger, Roger M., Brady, Stephen F., Curley, Paul, Perlow, Debra S., Paleveda, William J., Colton, C.Dylion, Zacchei, Anthony G., Tocco, Dominick J., Hoff, Dale R., Vandlen, Richard L., Gerich, John E., Hall, Larry, Mandarino, Lawrence, Cordes, Eugene H., Anderson, Paul S., Hirschmann, Ralph

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Angiotensin-converting enzyme inhibitors: synthesis and biological activity of acyltripeptide analogs of enalapril von Greenlee, William J, Allibone, Patricia L, Perlow, Debra S, Patchett, Arthur A, Ulm, Edgar H, Vassil, Theodore C

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1-(((7,7-Dimethyl-2(S)-(2(S)-amino-4-(methylsulfonyl)butyramido)bicyclo[2.2.1]heptan-1(S)-yl)methyl)sulfonyl)-4-(2-methylphenyl)piperazine (L-368,899): An Orally Bioavailable, Non-... von Williams, Peter D, Anderson, Paul S, Ball, Richard G, Bock, Mark G, Carroll, LeighAnne, Chiu, Shuet-Hing Lee, Clineschmidt, Bradley V, Culberson, J. Chris, Erb, Jill M

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Nonpeptide oxytocin antagonists: Analogs of L-371,257 with improved potency von Williams, Peter D., Bock, Mark G., Evans, Ben E., Freidinger, Roger M., Gallicchio, Steven N., Guidotti, Maribeth T., Jacobson, Marlene A., Kuo, Michelle S., Levy, Michelle R., Lis, Edward V., Michelson, Stuart R., Pawluczyk, Joseph M., Perlow, Debra S., Pettibone, Douglas J., Quigley, Amy G., Reiss, Duane R., Salvatore, Christopher, Stauffer, Kenneth J., Woyden, Carla J.

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Nonpeptide oxytocin antagonists: Potent, orally bioavailable analogs of L-371,257 containing A 1- R-(pyridyl)ethyl ether terminus von Kuo, Michelle S., Bock, Mark G., Freidinger, Roger M., Guidotti, Maribeth T., Lis, Edward V., Pawluczyk, Joseph M., Perlow, Debra S., Pettibone, Douglas J., Quigley, Amy G., Reiss, Duane R., Williams, Peter D., Woyden, Carla J.

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Conformationally constrained o-tolylpiperazine camphorsulfonamide oxytocin antagonists. Structural modifications that provide high receptor affinity and suggest a bioactive conform... von Williams, Peter D., Ball, Richard G., Clineschmidt, Bradley V., Culberson, J.Chris, Erb, Jill M., Freidinger, Roger M., Pawluczyk, Joseph M., Perlow, Debra S., Pettibone, Douglas J., Veber, Daniel F.

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Nanomolar-affinity, non-peptide oxytocin receptor antagonists von Evans, Ben E, Lundell, George F, Gilbert, Kevin F, Bock, Mark G, Rittle, Kenneth E, Carroll, Leigh Anne, Williams, Peter D, Pawluczyk, Joseph M, Leighton, James L

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Practical Synthesis of 4-Fluoro-2-(methylthio)benzylamine (V) and the Corresponding Sulfone (X) and Sulfonamide (XVI) von Perlow, Debra S., Kuo, Michelle S., Moritz, H. Marie, Wai, John S., Egbertson, Melissa S.

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ChemInform Abstract: Synthesis of Protected Lactam-Bridged Dipeptides von Perlow, Debra S., Freidinger, Roger M.

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Angiotensin-converting enzyme inhibitors: synthesis and biological activity of acyl tripeptide analogues of enalapril von GREENLEE, W. J, ALLIBONE, P. L, PERLOW, D. S, PATCHETT, A. A, ULM, E. H, VASSIL, T. C

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HIV Integrase inhibitors von HAN, WEI, EGBERTSON, MELISSA, PERLOW, DEBRA S, RUZEK, ROWENA D, ZHUANG, LINGHANG, WAI, JOHN S, OBLIGADO, VANESSA E

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HIV integrase inhibitors von ETTE MATTHEW M.,WILLIAMS PETER D.,PYE PHILIP J.,ANGELAUD REMY,ASKIN DAVID, HAN WEI,EGBERTSON MELISSA,WAI JOHN S.,ZHUANG LINGHANG,RUZEK ROWENA D.,PERLOW DEBRA S.,ISAACS RICHARD C. A.,CAMERON MARK,FOSTER BRUCE S.,DOLLING ULF H.,HOERRNER R. SCOTT,OBLIGADO VANESSA E.,NEILSON LOU

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HIV integrase inhibitors von HAN, WEI, EGBERTSON, MELISSA, PERLOW, DEBRA S, RUZEK, ROWENA D, ZHUANG, LINGHANG, WAI, JOHN S, OBLIGADO, VANESSA E

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HIV INTEGRASE INHIBITORS von PERLOW,DEBRA,S, OBLIGADO,VANESSA,E, WAI,JOHN,S, ZHUANG,LINGHANG, RUZEK,ROWENA,D, HAN,WEI, EGBERTSON,MELISSA

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