SST0001, a Chemically Modified Heparin, Inhibits Myeloma Growth and Angiogenesis via Disruption of the Heparanase/Syndecan-1 Axis von RITCHIE, Joseph P, RAMANI, Vishnu C, ZUNINO, Franco, VLODAVSKY, Israel, SANDERSON, Ralph D, YANG YANG, YONGSHENG REN, NAGGI, Annamaria, TORRI, Giangiacomo, CASU, Benito, PENCO, Sergio, PISANO, Claudio, CARMINATI, Paolo, TORTORETO, Monica

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Modulation of the Heparanase-inhibiting Activity of Heparin through Selective Desulfation, Graded N-Acetylation, and Glycol Splitting von Naggi, Annamaria, Casu, Benito, Perez, Marta, Torri, Giangiacomo, Cassinelli, Giuseppe, Penco, Sergio, Pisano, Claudio, Giannini, Giuseppe, Ishai-Michaeli, Rivka, Vlodavsky, Israel

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New macrocyclic analogs of the natural histone deacetylase inhibitor FK228; design, synthesis and preliminary biological evaluation von Ni, Minghong, Esposito, Emiliano, Raj, Victor Paul, Muzi, Laura, Zunino, Franco, Zuco, Valentina, Cominetti, Denis, Penco, Sergio, Dal Pozzo, Alma

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Natural and semisynthetic azaphilones as a new scaffold for Hsp90 inhibitors von Musso, Loana, Dallavalle, Sabrina, Merlini, Lucio, Bava, Adriana, Nasini, Gianluca, Penco, Sergio, Giannini, Giuseppe, Giommarelli, Chiara, De Cesare, Andrea, Zuco, Valentina, Vesci, Loredana, Pisano, Claudio, Dal Piaz, Fabrizio, De Tommasi, Nunziatina, Zunino, Franco

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Preclinical profile of antitumor activity of a novel hydrophilic camptothecin, ST1968 von Pisano, Claudio, De Cesare, Michelandrea, Beretta, Giovanni Luca, Zuco, Valentina, Pratesi, Graziella, Penco, Sergio, Vesci, Loredana, Foderà, Rosanna, Ferrara, Fabiana Fosca, Guglielmi, Mario Berardino, Carminati, Paolo, Dallavalle, Sabrina, Morini, Gabriella, Merlini, Lucio, Orlandi, Augusto, Zunino, Franco

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Short Heparin Sequences Spaced by Glycol-Split Uronate Residues Are Antagonists of Fibroblast Growth Factor 2 and Angiogenesis Inhibitors von Casu, Benito, Guerrini, Marco, Naggi, Annamaria, Perez, Marta, Torri, Giangiacomo, Ribatti, Domenico, Carminati, Paolo, Giannini, Giuseppe, Penco, Sergio, Pisano, Claudio, Belleri, Mirella, Rusnati, Marco, Presta, Marco

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Pattern of Antitumor Activity of a Novel Camptothecin, ST1481, in a Large Panel of Human Tumor Xenografts von PRATESI, Graziella, DE CESARE, Michelandrea, VESCI, Loredana, ZUNINO, Franco, CARENINI, Nives, PEREGO, Paola, RIGHETTI, Sabina C, CUCCO, Carla, MERLINI, Lucio, PISANO, Claudio, PENCO, Sergio, CARMINATI, Paolo

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7-Azaindole-1-carboxamides as a new class of PARP-1 inhibitors von Cincinelli, Raffaella, Musso, Loana, Merlini, Lucio, Giannini, Giuseppe, Vesci, Loredana, Milazzo, Ferdinando M., Carenini, Nives, Perego, Paola, Penco, Sergio, Artali, Roberto, Zunino, Franco, Pisano, Claudio, Dallavalle, Sabrina

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alpha.-Regioselectivity in palladium-catalyzed arylation of acyclic enol ethers von Cabri, Walter, Candiani, Ilaria, Bedeschi, Angelo, Penco, Sergio, Santi, Roberto

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Abstract 3096: Host antitumor immune response activated by Dual POLA1-HDAC11 inhibitors endowed with a large spectrum of antitumor activity von Pisano, Claudio, Merlini, Lucio, Penco, Sergio, Cincinelli, Raffaella, Darwiche, Nadine, Guglielmi, Mario B., Porta, Ilaria La, Pizzulo, Maddalena, Prosperi, Federica, Signorino, Giacomo, Colelli, Fabiana, Cardile, Francesco, Focareta, Laura, Fucci, Alessandra, D'Andrea, Egildo L., Riccio, Assunta, Dallavalle, Sabrina

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Abstract 4848: Preclinical antitumor activity of novel DNA polymerase 1 (POLA1) inhibitors von Pisano, Claudio, Merlini, Lucio, Penco, Sergio, Cincinelli, Raffaella, Darwiche, Nadine, Guglielmi, Mario B., Porta, Ilaria La, Signorino, Giacomo, Rubis, Gabriele De, Colelli, Fabiana, Cardile, Francesco, Fucci, Alessandra, D'Andrea, Egildo L., Dallavalle, Sabrina

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Design, synthesis, and evaluation of biphenyl-4-yl-acrylohydroxamic acid derivatives as histone deacetylase (HDAC) inhibitors von Dallavalle, Sabrina, Cincinelli, Raffaella, Nannei, Raffaella, Merlini, Lucio, Morini, Gabriella, Penco, Sergio, Pisano, Claudio, Vesci, Loredana, Barbarino, Marcella, Zuco, Valentina, De Cesare, Michelandrea, Zunino, Franco

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Abstract 4195: MIR002: a new POLA1 inhibitor endowed with a large spectrum of antitumor activity von Pisano, Claudio, Merlini, Lucio, Penco, Sergio, Cincinelli, Raffaella, Darwiche, Nadine, Guglielmi, Mario B., Esposito, Antonietta, Porta, Ilaria La, Signorino, Giacomo, Rubis, Gabriele De, Colelli, Fabiana, Cardile, Francesco, Fucci, Alessandra, D'Andrea, Egildo L., Dallavalle, Sabrina

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Conjugates of a Novel 7-Substituted Camptothecin with RGD-Peptides as αvβ3 Integrin Ligands: An Approach to Tumor-Targeted Therapy von Dal Pozzo, Alma, Esposito, Emiliano, Ni, Minghong, Muzi, Laura, Pisano, Claudio, Bucci, Federica, Vesci, Loredana, Castorina, Massimo, Penco, Sergio

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Heck reaction on anthraquinone derivatives: ligand, solvent and salt effects von Cabri, Walter, Candiani, Ilaria, DeBernardinis, Silvia, Francalanci, Franco, Penco, Sergio, Santo, Roberto

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Azetidinones as Zinc-Binding Groups to Design Selective HDAC8 Inhibitors von Galletti, Paola, Quintavalla, Arianna, Ventrici, Caterina, Giannini, Giuseppe, Cabri, Walter, Penco, Sergio, Gallo, Grazia, Vincenti, Silvia, Giacomini, Daria

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Synthesis, Modeling, and RET Protein Kinase Inhibitory Activity of 3- and 4-Substituted β-Carbolin-1-ones von Cincinelli, Raffaella, Cassinelli, Giuliana, Dallavalle, Sabrina, Lanzi, Cinzia, Merlini, Lucio, Botta, Maurizio, Tuccinardi, Tiziano, Martinelli, Adriano, Penco, Sergio, Zunino, Franco

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Isoxazolo(aza)naphthoquinones: A new class of cytotoxic Hsp90 inhibitors von Bargiotti, Alberto, Musso, Loana, Dallavalle, Sabrina, Merlini, Lucio, Gallo, Grazia, Ciacci, Andrea, Giannini, Giuseppe, Cabri, Walter, Penco, Sergio, Vesci, Loredana, Castorina, Massimo, Milazzo, Ferdinando Maria, Cervoni, Maria Luisa, Barbarino, Marcella, Pisano, Claudio, Giommarelli, Chiara, Zuco, Valentina, De Cesare, Michelandrea, Zunino, Franco

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Novel tumor-targeted RGD peptide–camptothecin conjugates: Synthesis and biological evaluation von Dal Pozzo, Alma, Ni, Ming-Hong, Esposito, Emiliano, Dallavalle, Sabrina, Musso, Loana, Bargiotti, Alberto, Pisano, Claudio, Vesci, Loredana, Bucci, Federica, Castorina, Massimo, Foderà, Rosanna, Giannini, Giuseppe, Aulicino, Concetta, Penco, Sergio

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A new group of oxime carbamates as reversible inhibitors of fatty acid amide hydrolase von Gattinoni, Sonia, Simone, Chiara De, Dallavalle, Sabrina, Fezza, Filomena, Nannei, Raffaella, Battista, Natalia, Minetti, Patrizia, Quattrociocchi, Gianandrea, Caprioli, Antonio, Borsini, Franco, Cabri, Walter, Penco, Sergio, Merlini, Lucio, Maccarrone, Mauro

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