The mTORC1/4E-BP1 axis represents a critical signaling node during fibrogenesis von Woodcock, Hannah V., Eley, Jessica D., Guillotin, Delphine, Platé, Manuela, Nanthakumar, Carmel B., Martufi, Matteo, Peace, Simon, Joberty, Gerard, Poeckel, Daniel, Good, Robert B., Taylor, Adam R., Zinn, Nico, Redding, Matthew, Forty, Ellen J., Hynds, Robert E., Swanton, Charles, Karsdal, Morten, Maher, Toby M., Fisher, Andrew, Bergamini, Giovanna, Marshall, Richard P., Blanchard, Andy D., Mercer, Paul F., Chambers, Rachel C.

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The developability of heteroaromatic and heteroaliphatic rings - do some have a better pedigree as potential drug molecules than others? von Ritchie, Timothy J, Macdonald, Simon J. F, Peace, Simon, Pickett, Stephen D, Luscombe, Christopher N

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Author Correction: The mTORC1/4E-BP1 axis represents a critical signaling node during fibrogenesis von Woodcock, Hannah V., Eley, Jessica D., Guillotin, Delphine, Platé, Manuela, Nanthakumar, Carmel B., Martufi, Matteo, Peace, Simon, Joberty, Gerard, Poeckel, Daniel, Good, Robert B., Taylor, Adam R., Zinn, Nico, Redding, Matthew, Forty, Ellen J., Hynds, Robert E., Swanton, Charles, Karsdal, Morten, Maher, Toby M., Fisher, Andrew, Bergamini, Giovanna, Marshall, Richard P., Blanchard, Andy D., Mercer, Paul F., Chambers, Rachel C.

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A high-throughput MALDI-TOF MS biochemical screen for small molecule inhibitors of the antigen aminopeptidase ERAP1 von Müller, Leonie, Burton, Amy K, Tayler, Chloe L, Rowedder, James E, Hutchinson, Jonathan P, Peace, Simon, Quayle, Julie M, Leveridge, Melanie V, Annan, Roland S, Trost, Matthias, Peltier-Heap, Rachel E, Dueñas, Maria Emilia

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Three Groups Good, Four Groups Bad? Atropisomerism in ortho-Substituted Diaryl Ethers von Betson, Mark S., Clayden, Jonathan, Worrall, Christopher P., Peace, Simon

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UV‐Induced 1,3,4‐Oxadiazole Formation from 5‐Substituted Tetrazoles and Carboxylic Acids in Flow von Green, Luke, Livingstone, Keith, Bertrand, Sophie, Peace, Simon, Jamieson, Craig

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The discovery of GSK221149A: A potent and selective oxytocin antagonist von Liddle, John, Allen, Michael J., Borthwick, Alan D., Brooks, David P., Davies, David E., Edwards, Richard M., Exall, Anne M., Hamlett, Chris, Irving, Wendy R., Mason, Andrew M., McCafferty, Gerald P., Nerozzi, Fabrizio, Peace, Simon, Philp, Joanne, Pollard, Derek, Pullen, Mark A., Shabbir, Shaila S., Sollis, Steve L., Westfall, Timothy D., Woollard, Pat M., Wu, Charlene, Hickey, Deirdre M.B.

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Synthesis of the B-ring of FR182877. Investigation of the reactions of 6-fumaryl 1,3,8-nonatrienes von Clarke, Paul A., Davie, Rebecca L., Peace, Simon

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Discovery of 3‑Oxabicyclo[4.1.0]heptane, a Non-nitrogen Containing Morpholine Isostere, and Its Application in Novel Inhibitors of the PI3K-AKT-mTOR Pathway von Hobbs, Heather, Bravi, Gianpaolo, Campbell, Ian, Convery, Maire, Davies, Hannah, Inglis, Graham, Pal, Sandeep, Peace, Simon, Redmond, Joanna, Summers, Declan

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The Nitro-Mannich Reaction and Its Application to the Stereoselective Synthesis of 1,2-Diamines von Adams, Harry, Anderson, James C, Peace, Simon, Pennell, Andrew M. K

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Correction to Discovery of 3‑Oxabicyclo[4.1.0]heptane, a Non-nitrogen Containing Morpholine Isostere, and Its Application in Novel Inhibitors of the PI3K-AKT-mTOR Pathway von Hobbs, Heather, Bravi, Gianpaolo, Campbell, Ian, Convery, Maire, Davies, Hannah, Inglis, Graham, Pal, Sandeep, Peace, Simon, Redmond, Joanna, Summers, Declan

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Increasing small molecule drug developability in sub-optimal chemical space von Ritchie, Timothy J., Macdonald, Simon J. F., Peace, Simon, Pickett, Stephen D., Luscombe, Christopher N.

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Evolution of a Novel, Orally Bioavailable Series of PI3Kδ Inhibitors from an Inhaled Lead for the Treatment of Respiratory Disease von Amour, Augustin, Barton, Nick, Cooper, Anthony W. J, Inglis, Graham, Jamieson, Craig, Luscombe, Christopher N, Morrell, Josie, Peace, Simon, Perez, David, Rowland, Paul, Tame, Chris, Uddin, Sorif, Vitulli, Giovanni, Wellaway, Natalie

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Discovery of Potent, Efficient, and Selective Inhibitors of Phosphoinositide 3‑Kinase δ through a Deconstruction and Regrowth Approach von Barton, Nick, Convery, Máire, Cooper, Anthony W. J, Down, Kenneth, Hamblin, J. Nicole, Inglis, Graham, Peace, Simon, Rowedder, James, Rowland, Paul, Taylor, Jonathan A, Wellaway, Natalie

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Identification of a sulfonamide series of CCR2 antagonists von Peace, Simon, Philp, Joanne, Brooks, Carl, Piercy, Val, Moores, Kitty, Smethurst, Chris, Watson, Steve, Gaines, Simon, Zippoli, Mara, Mookherjee, Claudette, Ife, Robert

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Pyridyl-2,5-Diketopiperazines as Potent, Selective, and Orally Bioavailable Oxytocin Antagonists: Synthesis, Pharmacokinetics, and In Vivo Potency von Borthwick, Alan D, Liddle, John, Davies, Dave E, Exall, Anne M, Hamlett, Christopher, Hickey, Deirdre M, Mason, Andrew M, Smith, Ian E. D, Nerozzi, Fabrizio, Peace, Simon, Pollard, Derek, Sollis, Steve L, Allen, Michael J, Woollard, Patrick M, Pullen, Mark A, Westfall, Timothy D, Stanislaus, Dinesh J

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Correction to Evolution of a Novel, Orally Bioavailable Series of PI3Kδ Inhibitors from an Inhaled Lead for the Treatment of Respiratory Disease von Amour, Augustin, Barton, Nick, Cooper, Anthony W. J, Inglis, Graham, Jamieson, Craig, Luscombe, Christopher N, Morrell, Josie, Peace, Simon, Perez, David, Rowland, Paul, Tame, Christopher J, Uddin, Sorif, Vitulli, Giovanni, Wellaway, Natalie

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Correction to Evolution of a Novel, Orally Bioavailable Series of PI3Kδ Inhibitors from an Inhaled Lead for the Treatment of Respiratory Disease von Amour, Augustin, Barton, Nick, Cooper, Anthony W. J, Inglis, Graham, Jamieson, Craig, Luscombe, Christopher N, Morrell, Josie, Peace, Simon, Perez, David, Rowland, Paul, Tame, Christopher J, Uddin, Sorif, Vitulli, Giovanni, Wellaway, Natalie

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Three Groups Good, Four Groups Bad? Atropisomerism in ortho-Substituted Diaryl Ethers von Betson, Mark S., Clayden, Jonathan, Worrall, Christopher P., Peace, Simon

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Increasing small molecule drug developability in sub-optimal chemical spaceElectronic supplementary information (ESI) available: Tables containing (a) the average values of all the... von Ritchie, Timothy J, Macdonald, Simon J. F, Peace, Simon, Pickett, Stephen D, Luscombe, Christopher N

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