DNA minor groove binders as potential antitumor and antimicrobial agents von Baraldi, Pier Giovanni, Bovero, Andrea, Fruttarolo, Francesca, Preti, Delia, Tabrizi, Mojgan Aghazadeh, Pavani, Maria Giovanna, Romagnoli, Romeo

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Synthesis and Biological Evaluation of 2- and 3-Aminobenzo[b]thiophene Derivatives as Antimitotic Agents and Inhibitors of Tubulin Polymerization von Romagnoli, Romeo, Baraldi, Pier Giovanni, Carrion, Maria Dora, Cara, Carlota Lopez, Preti, Delia, Fruttarolo, Francesca, Pavani, Maria Giovanna, Tabrizi, Mojgan Aghazadeh, Tolomeo, Manlio, Grimaudo, Stefania, Di Cristina, Antonella, Balzarini, Jan, Hadfield, John A, Brancale, Andrea, Hamel, Ernest

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Synthesis and Biological Evaluation of 2-Amino-3-(3‘,4‘,5‘-trimethoxybenzoyl)-5-aryl Thiophenes as a New Class of Potent Antitubulin Agents von Romagnoli, Romeo, Baraldi, Pier Giovanni, Pavani, Maria Giovanna, Tabrizi, Mojgan Aghazadeh, Preti, Delia, Fruttarolo, Francesca, Piccagli, Laura, Jung, M. Katherine, Hamel, Ernest, Borgatti, Monica, Gambari, Roberto

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Synthesis and Biological Evaluation of 2-(3‘,4‘,5‘-Trimethoxybenzoyl)-3-Amino 5-Aryl Thiophenes as a New Class of Tubulin Inhibitors von Romagnoli, Romeo, Baraldi, Pier Giovanni, Remusat, Vincent, Carrion, Maria Dora, Cara, Carlota Lopez, Preti, Delia, Fruttarolo, Francesca, Pavani, Maria Giovanna, Tabrizi, Mojgan Aghazadeh, Tolomeo, Manlio, Grimaudo, Stefania, Balzarini, Jan, Jordan, Mary Ann, Hamel, Ernest

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Synthesis and biological effects of a new series of 2-amino-3-benzoylthiophenes as allosteric enhancers of A1-adenosine receptor von BARALDI, P. G, ZAID, A. N, LAMPRONTI, I, FRUTTAROLO, F, PAVANI, M. G, TABRIZI, M. A, SHRYOCK, J. C, LEUNG, E, ROMAGNOLI, R

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Hybrid molecules based on distamycin A as potential antitumor agents von Baraldi, Pier Giovanni, Zaid, Abdel Naser, Preti, Delia, Fruttarolo, Francesca, Tabrizi, Mojgan Aghazadeh, Iaconinoto, Antonietta, Pavani, Maria Giovanna, Carrion, Maria Dora, Cara, Carlota Lopez, Romagnoli, Romeo

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Benzoyl and cinnamoyl nitrogen mustard derivatives of benzoheterocyclic analogues of the tallimustine: Synthesis and antitumour activity von BARALDI, Pier Giovanni, ROMAGNOLI, Romeo, PAVANI, Maria Giovanna, NUNEZ, Maria Del, BINGHAM, John P, HARTLEY, John A

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Novel Combretastatin Analogues Endowed with Antitumor Activity von Simoni, Daniele, Romagnoli, Romeo, Baruchello, Riccardo, Rondanin, Riccardo, Rizzi, Michele, Pavani, Maria Giovanna, Alloatti, Domenico, Giannini, Giuseppe, Marcellini, Marcella, Riccioni, Teresa, Castorina, Massimo, Guglielmi, Mario B, Bucci, Federica, Carminati, Paolo, Pisano, Claudio

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Antimicrobial and antitumor activity of n-heteroimmine-1,2,3-dithiazoles and their transformation in triazolo-, imidazo-, and pyrazolopirimidines von Baraldi, Pier Giovanni, Pavani, Maria Giovanna, Nuñez, Maria del Carmen, Brigidi, Patrizia, Vitali, Beatrice, Gambari, Roberto, Romagnoli, Romeo

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Design, Synthesis, DNA Binding, and Biological Evaluation of Water-Soluble Hybrid Molecules Containing Two Pyrazole Analogues of the Alkylating Cyclopropylpyrroloindole (CPI) Subun... von Baraldi, Pier Giovanni, Balboni, Gianfrano, Pavani, Maria Giovanna, Spalluto, Giampiero, Tabrizi, Mojgan Aghazadeh, Clercq, Erik De, Balzarini, Jan, Bando, Toshikazu, Sugiyama, Hiroshi, Romagnoli, Romeo

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Synthesis of 2-amino-3-heteroaroylthiophenes and evaluation of their activity as potential allosteric enhancers at the human A 1 receptor von Baraldi, Pier Giovanni, Pavani, Maria Giovanna, Shryock, John C., Moorman, Allan R., Iannotta, Valeria, Borea, Pier Andrea, Romagnoli, Romeo

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Synthesis and Biological Effects of Novel 2-Amino-3-naphthoylthiophenes as Allosteric Enhancers of the A1 Adenosine Receptor von Baraldi, Pier Giovanni, Romagnoli, Romeo, Pavani, Maria Giovanna, del Carmen Nuñez, Maria, Tabrizi, Mojgan Aghazadeh, Shryock, John C, Leung, Edward, Moorman, Allan R, Uluoglu, Canan, Iannotta, Valeria, Merighi, Stefania, Borea, Pier Andrea

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Synthesis and biological characterization of [3H] (2-amino-4,5,6,7-tetrahydrobenzo[b]thiophen-3-yl)-(4-chlorophenyl)-methanone, the first radiolabelled adenosine A1 allosteric enha... von BARALDI, Pier Giovanni, PAVANI, Maria Giovanna, LEUNG, Edward, MOORMAN, Allan R, VARANI, Katia, VINCENZI, Fabrizio, BOREA, Pier Andrea, ROMAGNOLI, Romeo

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Synthesis and cellular pharmacology studies of a series of 2-amino-3-aroyl-4-substituted thiophene derivatives von Romagnoli, Romeo, Baraldi, Pier Giovanni, Pavani, Maria Giovanna, Cruz-Lopez, Olga, Hamel, Ernest, Balzarini, Jan, Brognara, Eleonora, Zuccato, Cristina, Gambari, Roberto

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Synthesis, radiolabeling, and preliminary biological evaluation of [ 3H]-1-[( S)- N, O-bis-(isoquinolinesulfonyl)- N-methyl-tyrosyl]-4-( o-tolyl)-piperazine, a potent antagonist ra... von Romagnoli, Romeo, Baraldi, Pier Giovanni, Pavani, Maria Giovanna, Tabrizi, Mojgan Aghazadeh, Moorman, Allan R., Di Virgilio, Francesco, Cattabriga, Elena, Pancaldi, Cecilia, Gessi, Stefania, Borea, Pier Andrea

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Synthesis and biological characterization of [ super(3)H] (2-amino-4,5,6,7- tetrahydrobenzo[b]thiophen-3-yl)-(4-chlorophenyl)-methanone, the first radiolabelled adenosine A sub(1)... von Baraldi, Pier Giovanni, Pavani, Maria Giovanna, Leung, Edward, Moorman, Allan R, Varani, Katia, Vincenzi, Fabrizio, Borea, Pier Andrea, Romagnoli, Romeo

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Synthesis and biological characterization of [ 3H] (2-amino-4,5,6,7-tetrahydrobenzo[ b]thiophen-3-yl)-(4-chlorophenyl)-methanone, the first radiolabelled adenosine A 1 allosteric e... von Baraldi, Pier Giovanni, Pavani, Maria Giovanna, Leung, Edward, Moorman, Allan R., Varani, Katia, Vincenzi, Fabrizio, Borea, Pier Andrea, Romagnoli, Romeo

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Allosteric modulators for the A1-adenosine receptor von Baraldi, Pier Giovanni, Moorman, Allan R, Tabrizi, Mojgan Aghazadeh, Pavani, MariaGiovanna, Romagnoli, Romeo

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Synthesis of 2-amino-3-heteroaroylthiophenes and evaluation of their activity as potential allosteric enhancers at the human A1 receptor von BARALDI, Pier Giovanni, PAVANI, Maria Giovanna, SHRYOCK, John C, MOORMAN, Allan R, IANNOTTA, Valeria, BOREA, Pier Andrea, ROMAGNOLI, Romeo

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Synthesis, radiolabeling, and preliminary biological evaluation of [3H]-1-[(S)-N, O-bis-(isoquinolinesulfonyl)-N-methyl-tyrosyl]-4-(o-tolyl)-piperaz ine, a potent antagonist radiol... von ROMAGNOLI, Romeo, BARALDI, Pier Giovanni, PAVANI, Maria Giovanna, TABRIZI, Mojgan Aghazadeh, MOORMAN, Allan R, DI VIRGILIO, Francesco, CATTABRIGA, Elena, PANCALDI, Cecilia, GESSI, Stefania, BOREA, Pier Andrea

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