Molecular Structures of Human Factor Xa Complexed with Ketopiperazine Inhibitors:  Preference for a Neutral Group in the S1 Pocket von Maignan, Sébastien, Guilloteau, Jean-Pierre, Choi-Sledeski, Yong Mi, Becker, Michael R, Ewing, William R, Pauls, Henry W, Spada, Alfred P, Mikol, Vincent

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A Convenient Synthesis of Heteroaryl Benzoic Acids via Suzuki Reaction von Gong, Yong, Pauls, Henry W.

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Crystal Structures of Human Factor Xa Complexed with Potent Inhibitors von Maignan, Sébastien, Guilloteau, Jean-Pierre, Pouzieux, Stéphanie, Choi-Sledeski, Yong Mi, Becker, Michael R, Klein, Scott I, Ewing, William R, Pauls, Henry W, Spada, Alfred P, Mikol, Vincent

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Optimization of the β-Aminoester class of factor Xa inhibitors. part 2: Identification of FXV673 as a potent and selective inhibitor with excellent In vivo anticoagulant activity von Guertin, Kevin R, Gardner, Charles J, Klein, Scott I, Zulli, Allison L, Czekaj, Mark, Gong, Yong, Spada, Alfred P, Cheney, Daniel L, Maignan, Sebastian, Guilloteau, Jean-Pierre, Brown, Karen D, Colussi, Dennis J, Chu, Valeria, Heran, Christopher L, Morgan, Suzanne R, Bentley, Ross G, Dunwiddie, Christopher T, Leadley, Robert J, Pauls, Henry W

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Pharmacological Characterization of a Novel Factor Xa Inhibitor, FXV673 von Chu, Valeria, Brown, Karen, Colussi, Dennis, Gao, Jingbo, Bostwick, Jeffery, Kasiewski, Charles, Bentley, Ross, Morgan, Susan, Guertin, Kevin, Pauls, Henry W, Gong, Yong, Zulli, Alison, Perrone, Mark H, Dunwiddie, Christopher T, Leadley, Robert J

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Optimization of the β-Aminoester class of factor Xa inhibitors. part 1: P 4 and side-Chain modifications for improved In vitro potency von Czekaj, Mark, Klein, Scott I, Guertin, Kevin R, Gardner, Charles J, Zulli, Allison L, Pauls, Henry W, Spada, Alfred P, Cheney, Daniel L, Brown, Karen D, Colussi, Dennis J, Chu, Valeria, Leadley, Robert J, Dunwiddie, Christopher T

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Solid-phase parallel synthesis of azarene pyrrolidinones as factor Xa inhibitors von Gong, Y, Becker, M, Choi-Sledeski, Y M, Davis, R S, Salvino, J M, Chu, V, Brown, K D, Pauls, H W

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Aminoisoquinolines: Design and synthesis of an orally active benzamidine isostere for the inhibition of factor XA von Choi-Sledeski, Y.M., Becker, M.R., Green, D.M., Davis, R., Ewing, W.R., Mason, H.J., Ly, C., Spada, A., Liang, G., Cheney, D., Barton, J., Chu, V., Brown, K., Colussi, D., Bentley, R., Leadley, R., Dunwiddie, C., Pauls, H.W.

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In Vitro Characterization of a Novel Factor Xa Inhibitor, RPR 130737 von Chu, Valeria, Brown, Karen, Colussi, Dennis, Choi, Yong-Mi, Green, Dan, Pauls, Henry W, Spada, Alfred P, Perrone, Mark H, Leadley, Robert J, Dunwiddie, Christopher T

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Synthesis, SAR and in vivo activity of novel thienopyridine sulfonamide pyrrolidinones as factor Xa inhibitors von Becker, Michael R., Ewing, William R., Davis, Roderick S., Pauls, Henry W., Ly, Cuong, Li, Aiwen, Mason, Helen J., Choi-Sledeski, Yong Mi, Spada, Alfred P., Chu, Valeria, Brown, Karen D., Colussi, Dennis J., Leadley, Robert J., Bentley, Ross, Bostwick, Jeff, Kasiewski, Charles, Morgan, Suzanne

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Amido-(propyl and allyl)-hydroxybenzamidines : Development of achiral inhibitors of factor Xa von YONG GONG, PAULS, H. W, SPADA, A. P, CZEKAJ, M, GUYAN LIANG, CHU, V, COLUSSI, D. J, BROWN, K. D, JINGBO GAO

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New inhibitors of cysteine proteinases. Peptidyl acyloxymethyl ketones and the quiescent nucleofuge strategy von Smith, Roger A, Copp, Leslie J, Coles, Peter J, Pauls, Henry W, Robinson, Valerie J, Spencer, Robin W, Heard, Stephen B, Krantz, Allen

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A novel synthesis of methyl .alpha.-L-garosaminide which illustrates a stereocontrolled approach to the cis-hydroxyamino moiety of amino sugars von Pauls, Henry W, Fraser-Reid, Bert

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An efficient synthesis of ristosamine utilizing the allylic hydroxyl of a hex-2-enopyranoside von Pauls, Henry W, Fraser-Reid, Bert

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C-13 NMR CHARACTERIZATION OF THE PAPAIN ADDUCT FORMED BY PEPTIDYL ACYLOXYMETHYL, ARYLOXYMETHYL, AND CHLOROMETHYL KETONE IRREVERSIBLE INHIBITORS von ROBINSON, VJ, PAULS, HW, COLES, PJ, SMITH, RA, KRANTZ, A

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Characterization of the bisphosphonate recognition site on hydroxyapatite using radioligand binding techniques with [14C]citric acid von JARVIS, M. F, BURNS, C. J, PAULS, H. W, ASSAL, A, KIM, J. S, CHENEY, D. L, YOUSSEFYEH, R. D

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Simple One-Pot Synthesis of 2-Acylmethylidene-3-methylthiazolines von Pauls, Henry W., Krantz, Allen

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2-(Peptidamido)-cyclobutanones: A novel strategy for the inhibition of serine elastases von Pauls, Henry W., Cheng, Bill, Reid, Lorne S.

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Chiral building blocks for amphotericin B von Liang, David, Pauls, Henry W, Fraser-Reid, Bert, Georges, Michael, Mubarak, Azeez M, Jarosz, Slawomir

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A short, efficient route to a protected daunosamine from L-rhamnose von Pauls, Henry W., Fraser-Reid, Bert

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