PLAG alleviates cisplatin-induced cachexia in lung cancer implanted mice von Kim, Guen Tae, Kim, Eun Young, Shin, Su-Hyun, Lee, Hyowon, Lee, Se Hee, Park, Kaapjoo, Sohn, Ki-Young, Yoon, Sun Young, Kim, Jae Wha

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Abstract 1447: Suppressive effect of PLAG on tumor progression and its synergistic therapeutic effect with ICI therapy through adenosine clearance von Kim, Guen Tae, Yoon, Sun Young, Park, Kaapjoo, Kim, Heesoo, Sohn, Ki-Young, Kim, Jae Wha

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Identification of YH-GKA, a novel benzamide glucokinase activator as therapeutic candidate for type 2 diabetes mellitus von Park, Kaapjoo

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The effect of mGlu5 receptor positive allosteric modulators on signaling molecules in brain slices von Liu, Feng, Zhang, Guoming, Hornby, Geoffrey, Vasylyev, Dmytro, Bowlby, Mark, Park, Kaapjoo, Gilbert, Adam, Marquis, Karen, Andree, Terrance H.

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Isolation and Identification of Eukaryotic Initiation Factor 4A as a Molecular Target for the Marine Natural Product Pateamine A von Low, Woon‐Kai, Dang, Yongjun, Schneider‐Poetsch, Tilman, Shi, Zonggao, Choi, Nam Song, Rzasa, Robert M., Shea, Helene A., Li, Shukun, Park, Kaapjoo, Ma, Gil, Romo, Daniel, Liu, Jun O.

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Synthesis of 3-Indolyl-2,5-dihydroxybenzoquinones von Pirrung, Michael C, Park, Kaapjoo, Li, Zhitao

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Discovery of thienothiazolocarboxamide analogues as novel anti-tubercular agent von Jin, Guanghai, Mi Kim, Young, Lee, Aram, Choi, Junghwan, Kang, Sunhee, Seo, Mooyoung, Jea Seo, Jeong, Lee, Sumi, Kang, Juhee, Kim, Jaeseung, Park, Sinyoung, Woo, Minjeong, Falcão, Virgínia Carla de Almeida, Lee, Honggun, Heo, Jinyeong, Shum, David, Park, Kaapjoo, Delorme, Vincent, Choi, Inhee

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Design and Synthesis of Acetylenyl Benzamide Derivatives as Novel Glucokinase Activators for the Treatment of T2DM von Park, Kaapjoo, Lee, Byoung Moon, Hyun, Kwan Hoon, Han, Taedong, Lee, Dong Hoon, Choi, Hyun Ho

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Signaling Effects of Demethylasterriquinone B1, a Selective Insulin Receptor Modulator von Webster, Nicholas J.G, Park, Kaapjoo, Pirrung, Michael C

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Discovery of 3-(4-methanesulfonylphenoxy)-N-[1-(2-methoxy-ethoxymethyl)-1H-pyrazol-3-yl]-5-(3-methylpyridin-2-yl)-benzamide as a novel glucokinase activator (GKA) for the treatment... von Park, Kaapjoo, Lee, Byoung Moon, Hyun, Kwan Hoon, Lee, Dong Hoon, Choi, Hyun Ho, Kim, Hyunmi, Chong, Wonee, Kim, Kyeong Bae, Nam, Su Youn

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Compound 19e, a Novel Glucokinase Activator, Protects against Cytokine-Induced Beta-Cell Apoptosis in INS-1 Cells von Oh, Yoon Sin, Seo, Eunhui, Park, Kaapjoo, Jun, Hee-Sook

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Discovery of a novel phenylethyl benzamide glucokinase activator for the treatment of type 2 diabetes mellitus von Park, Kaapjoo, Lee, Byoung Moon, Kim, Young Hwan, Han, Taedong, Yi, Wonhui, Lee, Dong Hoon, Choi, Hyun Ho, Chong, Wonee, Lee, Chun Ho

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Abstract 5478: EC-18 suppressed tumor growth and alleviated side effects caused by cisplatin in the HNSCC implantation model von KIM, Guentae, Kim, Eun Young, Shin, Su-Hyun, Lee, Hyowon, Yoon, Sun Young, Park, Kaapjoo, Sohn, Ki-young, Kim, Jae Wha

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Treatment with glucokinase activator, YH-GKA, increases cell proliferation and decreases glucotoxic apoptosis in INS-1 cells von Oh, Yoon Sin, Lee, Youn-Jung, Park, Kaapjoo, Choi, Hyun Ho, Yoo, Sangjong, Jun, Hee-Sook

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Novel benzofuran-3-one indole inhibitors of PI3 kinase-α and the mammalian target of rapamycin: Hit to lead studies von Bursavich, Matthew G., Brooijmans, Natasja, Feldberg, Lawrence, Hollander, Irwin, Kim, Stephen, Lombardi, Sabrina, Park, Kaapjoo, Mallon, Robert, Gilbert, Adam M.

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Discovery of selective metal-binding peptoids using 19F encoded combinatorial libraries von Pirrung, Michael C, Park, Kaapjoo

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Synthesis and activity of tryptophan sulfonamide derivatives as novel non-hydroxamate TNF-α converting enzyme (TACE) inhibitors von Park, Kaapjoo, Gopalsamy, Ariamala, Aplasca, Alexis, Ellingboe, John W., Xu, Weixin, Zhang, Yuhua, Levin, Jeremy I.

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Novel purine and pyrazolo[3,4- d]pyrimidine inhibitors of PI3 kinase-α: Hit to lead studies von Gilbert, Adam M., Nowak, Pawel, Brooijmans, Natasja, Bursavich, Matthew G., Dehnhardt, Christoph, Santos, Efren Delos, Feldberg, Larry R., Hollander, Irwin, Kim, Stephen, Lombardi, Sabrina, Park, Kaapjoo, Venkatesan, Aranapakam M., Mallon, Robert

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Inhibition of the Signal Transducer and Activator of Transcription-3 (STAT3) Signaling Pathway by 4-Oxo-1-Phenyl-1,4-Dihydroquinoline-3-Carboxylic Acid Esters von Xu, Jun, Cole, Derek C, Chang, Chao-Pei Betty, Ayyad, Ramzi, Asselin, Magda, Hao, Wenshan, Gibbons, James, Jelinsky, Scott A, Saraf, Kathryn A, Park, Kaapjoo

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Design and synthesis of 3,4-dihydro-1H-[1]-benzothieno[2,3-c]pyran and 3,4-dihydro-1H-pyrano[3,4-b]benzofuran derivatives as non-nucleoside inhibitors of HCV NS5B RNA dependent RNA... von Gopalsamy, Ariamala, Aplasca, Alexis, Ciszewski, Gregory, Park, Kaapjoo, Ellingboe, John W, Orlowski, Mark, Feld, Boris, Howe, Anita Y M

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