Discovery of Orally Active Inhibitors of Brahma Homolog (BRM)/SMARCA2 ATPase Activity for the Treatment of Brahma Related Gene 1 (BRG1)/SMARCA4-Mutant Cancers von Papillon, Julien P. N, Nakajima, Katsumasa, Adair, Christopher D, Hempel, Jonathan, Jouk, Andriana O, Karki, Rajeshri G, Mathieu, Simon, Möbitz, Henrik, Ntaganda, Rukundo, Smith, Troy, Visser, Michael, Hill, Susan E, Hurtado, Felipe Kellermann, Chenail, Gregg, Bhang, Hyo-Eun C, Bric, Anka, Xiang, Kay, Bushold, Geoffrey, Gilbert, Tamara, Vattay, Anthony, Dooley, Julie, Costa, Emily A, Park, Isabel, Li, Ailing, Farley, David, Lounkine, Eugen, Yue, Q. Kimberley, Xie, Xiaoling, Zhu, Xiaoping, Kulathila, Raviraj, King, Daniel, Hu, Tiancen, Vulic, Katarina, Cantwell, John, Luu, Catherine, Jagani, Zainab

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Discovery of Darovasertib (NVP-LXS196), a Pan-PKC Inhibitor for the Treatment of Metastatic Uveal Melanoma von Visser, Michael, Papillon, Julien P. N., Luzzio, Michael, LaMarche, Matthew J., Fan, Jianmei, Michael, Walter, Wang, David, Zhang, Alan, Straub, Christopher, Mathieu, Simon, Kato, Mitsunori, Palermo, Mark, Chen, Christine, Ramsey, Timothy, Joud, Carol, Barrett, Rosemary, Vattay, Anthony, Guo, Ribo, Bric, Anka, Chung, Franklin, Liang, Guiqing, Romanowski, Michael J., Lam, Joni, Thohan, Sanjeev, Atassi, Faraj, Wylie, Andrew, Cooke, Vesselina G.

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Structure–Activity Relationships, Pharmacokinetics, and in Vivo Activity of CYP11B2 and CYP11B1 Inhibitors von Papillon, Julien P. N, Adams, Christopher M, Hu, Qi-Ying, Lou, Changgang, Singh, Alok K, Zhang, Chun, Carvalho, Jose, Rajan, Srinivan, Amaral, Adam, Beil, Michael E, Fu, Fumin, Gangl, Eric, Hu, Chii-Whei, Jeng, Arco Y, LaSala, Daniel, Liang, Guiqing, Logman, Michael, Maniara, Wieslawa M, Rigel, Dean F, Smith, Sherri A, Ksander, Gary M

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Discovery of a novel indole pharmacophore for the irreversible inhibition of myeloperoxidase (MPO) von Patnaik, Anup, Axford, Laura, Deng, Lin, Cohick, Evan, Ren, Xianglin, Loi, Sally, Kecman, Sam, Hollis-Symynkywicz, Micah, Harrison, Tyler J., Papillon, Julien P.N., Dales, Natalie, Hamann, Lawrence G., Lee, Lac, Regard, Jean B., Marcinkeviciene, Jovita, Marro, Martin L., Patterson, Andrew W.

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The Discovery of SWI/SNF Chromatin Remodeling Activity as a Novel and Targetable Dependency in Uveal Melanoma von Rago, Florencia, Elliott, GiNell, Li, Ailing, Sprouffske, Kathleen, Kerr, Grainne, Desplat, Aurore, Abramowski, Dorothee, Chen, Julie T., Farsidjani, Ali, Xiang, Kay X., Bushold, Geoffrey, Feng, Yun, Shirley, Matthew D., Bric, Anka, Vattay, Anthony, Möbitz, Henrik, Nakajima, Katsumasa, Adair, Christopher D., Mathieu, Simon, Ntaganda, Rukundo, Smith, Troy, Papillon, Julien P.N., Kauffmann, Audrey, Ruddy, David A., Bhang, Hyo-eun C., Castelletti, Deborah, Jagani, Zainab

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Discovery of N‑[5-(6-Chloro-3-cyano-1-methyl‑1H‑indol-2-yl)-pyridin-3-ylmethyl]-ethanesulfonamide, a Cortisol-Sparing CYP11B2 Inhibitor that Lowers Aldosterone in Human Subjects... von Papillon, Julien P. N, Lou, Changgang, Singh, Alok K, Adams, Christopher M, Ksander, Gary M, Beil, Michael E, Chen, Wei, Leung-Chu, Jennifer, Fu, Fumin, Gan, Lu, Hu, Chii-Whei, Jeng, Arco Y, LaSala, Daniel, Liang, Guiqing, Rigel, Dean F, Russell, Kerry S, Vest, John A, Watson, Catherine

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Dinuclear Asymmetric Zn Aldol Additions:  Formal Asymmetric Synthesis of Fostriecin von Trost, Barry M, Frederiksen, Mathias U, Papillon, Julien P. N, Harrington, Paul E, Shin, Seunghoon, Shireman, Brock T

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Ocular Pharmacology and Toxicology of TRPV1 Antagonist SAF312 (Libvatrep) von Mogi, Muneto, Mendonza, Anisha E., Chastain, James, Demirs, John T., Medley, Quintus G., Zhang, Qin, Papillon, Julien P. N., Yang, Junzheng, Gao, Yan, Xu, YongYao, Stasi, Kalliopi

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Discovery and in Vivo Evaluation of Potent Dual CYP11B2 (Aldosterone Synthase) and CYP11B1 Inhibitors von Meredith, Erik L, Ksander, Gary, Monovich, Lauren G, Papillon, Julien P. N, Liu, Qian, Miranda, Karl, Morris, Patrick, Rao, Chang, Burgis, Robin, Capparelli, Michael, Hu, Qi-Ying, Singh, Alok, Rigel, Dean F, Jeng, Arco Y, Beil, Michael, Fu, Fumin, Hu, Chii-Whei, LaSala, Daniel

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Synthetic phospholipids as specific substrates for plasma endothelial lipase von Papillon, Julien P.N., Pan, Meihui, Brousseau, Margaret E., Gilchrist, Mark A., Lou, Changgang, Singh, Alok K., Stawicki, Todd, Thompson, James E.

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Formal synthesis of (+)-neooxazolomycin via a Stille cross-coupling/deconjugation route von Bastin, Reyhan, Dale, James W., Edwards, Michael G., Papillon, Julien P.N., Webb, Michael R., Taylor, Richard J.K.

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Discovery of 1-((6-Aminopyridin-3-yl)Methyl)-3-(4-Bromophenyl)Urea as a Potent, Irreversible Myeloperoxidase Inhibitor von Marro, Martin L, Patterson, Andrew W, Lee, Lac, Deng, Lin, Reynolds, Aimee, Ren, Xianglin, Axford, Laura, Patnaik, Anup, Hollis-Symynkywicz, Micah, Casson, Nigel, Custeau, Dominique, Ames, Lisa, Loi, Sally, Zhang, Lihe, Honda, Toshiyuki, Blank, Jutta, Harrison, Tyler J, Papillon, Julien P N, Hamann, Lawrence G, Marcinkeviciene, Jovita, Regard, Jean B

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Ru-Catalyzed Alkene−Alkyne Coupling. Total Synthesis of Amphidinolide P von Trost, Barry M, Papillon, Julien P. N, Nussbaumer, Thomas

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Recent Developments for the Treatment of Glaucoma von Adams, Christopher M., Papillon, Julien P. N.

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The Preparation of Nonracemic Secondary α-(Carbamoyloxy)alkylzinc and Copper Reagents. A Versatile Approach to Enantioenriched Alcohols von Papillon, Julien P. N, Taylor, Richard J. K

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New synthetic method for the polymerization of alkylthiophenes von Se´vignon, Marc, Papillon, Julien, Schulz, Emmanuelle, Lemaire, Marc

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Alkene−Alkyne Coupling as a Linchpin:  An Efficient and Convergent Synthesis of Amphidinolide P von Trost, Barry M, Papillon, Julien P. N

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The First Syntheses of the 1-Oxo-2-oxa-5-azaspiro[3.4]octane Ring System Found in Oxazolomycin von Papillon, Julien P. N, Taylor, Richard J. K

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Towards the preparation of modified chiral electrodes for heterogeneous asymmetric catalysis: synthesis and electrochemical properties of ( S,S)-5,5′-bis-[3-(3-methyl-pentyl)-thiop... von Papillon, Julien, Schulz, Emmanuelle, Gélinas, Stéphane, Lessard, Jean, Lemaire, Marc

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UREA COMPOUNDS AND COMPOSITIONS AS SMARCA2/BRM-ATPASE INHIBITORS von ADAIR, Christopher, PAPILLON, Julien

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