Donated chemical probes for open science von Müller, Susanne, Ackloo, Suzanne, Arrowsmith, Cheryl H, Bauser, Marcus, Baryza, Jeremy L, Blagg, Julian, Böttcher, Jark, Bountra, Chas, Brown, Peter J, Bunnage, Mark E, Carter, Adrian J, Damerell, David, Dötsch, Volker, Drewry, David H, Edwards, Aled M, Edwards, James, Elkins, Jon M, Fischer, Christian, Frye, Stephen V, Gollner, Andreas, Grimshaw, Charles E, IJzerman, Adriaan, Hanke, Thomas, Hartung, Ingo V, Hitchcock, Steve, Howe, Trevor, Hughes, Terry V, Laufer, Stefan, Li, Volkhart Mj, Liras, Spiros, Marsden, Brian D, Matsui, Hisanori, Mathias, John, O'Hagan, Ronan C, Owen, Dafydd R, Pande, Vineet, Rauh, Daniel, Rosenberg, Saul H, Roth, Bryan L, Schneider, Natalie S, Scholten, Cora, Singh Saikatendu, Kumar, Simeonov, Anton, Takizawa, Masayuki, Tse, Chris, Thompson, Paul R, Treiber, Daniel K, Viana, Amélia Yi, Wells, Carrow I, Willson, Timothy M, Zuercher, William J, Knapp, Stefan, Mueller-Fahrnow, Anke

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Understanding the Complexity of Epigenetic Target Space von Pande, Vineet

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Understanding the Complexity of Epigenetic Target Space: Miniperspective von Pande, Vineet

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Identification of Two Non-Peptidergic Small Molecule Inhibitors of CBX2 Binding to K27 Trimethylated Oligonucleosomes von Lercher, Lukas, Simon, Nina, Bergmann, Andreas, Tauchert, Marcel, Bochmann, David, Bashir, Tarig, Neuefeind, Torsten, Riley, Daniel, Danna, Ben, Krawczuk, Paul, Pande, Vineet, Patrick, Aaron, Steele, Ruth, Wang, Weixue, Rupnow, Brent, Tummino, Peter, Sharma, Sujata, Finley, Michael

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Structure–Function Defects of the TWINKLE Linker Region in Progressive External Ophthalmoplegia von Korhonen, Jenny A., Pande, Vineet, Holmlund, Teresa, Farge, Géraldine, Pham, Xuan Hoi, Nilsson, Lennart, Falkenberg, Maria

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Structure–function defects of the twinkle amino-terminal region in progressive external ophthalmoplegia von Holmlund, Teresa, Farge, Géraldine, Pande, Vineet, Korhonen, Jenny, Nilsson, Lennart, Falkenberg, Maria

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Exploring the Application of SiteMap and Site Finder for Focused Cryptic Pocket Identification von Ge, Yunhui, Pande, Vineet, Seierstad, Mark J., Damm-Ganamet, Kelly L.

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Application of A lpha F old models in evaluating ligandable cysteines across E 3 ligases von Koldenhof, Patrick, Bemelmans, Martijn P., Ghosh, Brahma, Damm‐Ganamet, Kelly L., van Vlijmen, Herman W. T., Pande, Vineet

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Synthesis and Reactivity of Spirocarbocycles as Scaffolds for Nucleoside Analogues von Verhoeven, Jonas, Deraet, Xavier, Pande, Vineet, Sun, Weimei, Alonso, Mercedes, De Proft, Frank, Meerpoel, Lieven, Thuring, Jan Willem, Verniest, Guido

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Alchemical Free Energy Calculations on Membrane-Associated Proteins von Papadourakis, Michail, Sinenka, Hryhory, Matricon, Pierre, Hénin, Jérôme, Brannigan, Grace, Pérez-Benito, Laura, Pande, Vineet, van Vlijmen, Herman, de Graaf, Chris, Deflorian, Francesca, Tresadern, Gary, Cecchini, Marco, Cournia, Zoe

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Discovery and Pharmacological Characterization of JNJ-64619178, a Novel Small-Molecule Inhibitor of PRMT5 with Potent Antitumor Activity von Brehmer, Dirk, Beke, Lijs, Wu, Tongfei, Millar, Hillary J., Moy, Christopher, Sun, Weimei, Mannens, Geert, Pande, Vineet, Boeckx, An, van Heerde, Erika, Nys, Thomas, Gustin, Emmanuel M., Verbist, Bie, Zhou, Longen, Fan, Yue, Bhargava, Vipul, Safabakhsh, Pegah, Vinken, Petra, Verhulst, Tinne, Gilbert, Angelique, Rai, Sumit, Graubert, Timothy A., Pastore, Friederike, Fiore, Danilo, Gu, Junchen, Johnson, Amy, Philippar, Ulrike, Morschhauser, Barbara, Walker, David, De Lange, Desiree, Keersmaekers, Vikki, Viellevoye, Marcel, Diels, Gaston, Schepens, Wim, Thuring, Jan Willem, Meerpoel, Lieven, Packman, Kathryn, Lorenzi, Matthew, Laquerre, Sylvie

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Application of AlphaFold models in evaluating ligandable cysteines across E3 ligases von Koldenhof, Patrick, Bemelmans, Martijn P., Ghosh, Brahma, Damm‐Ganamet, Kelly L., Vlijmen, Herman W. T., Pande, Vineet

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Insights into structure, dynamics and hydration of locked nucleic acid (LNA) strand-based duplexes from molecular dynamics simulations von Pande, Vineet, Nilsson, Lennart

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Discovery of JNJ-63576253: A Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC) von Zhang, Zhuming, Connolly, Peter J, Lim, Heng Keang, Pande, Vineet, Meerpoel, Lieven, Teleha, Christopher, Branch, Jonathan R, Ondrus, Janine, Hickson, Ian, Bush, Tammy, Luistro, Leopoldo, Packman, Kathryn, Bischoff, James R, Ibrahim, Salam, Parrett, Christopher, Chong, Yolanda, Gottardis, Marco M, Bignan, Gilles

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Gut-Restricted Selective Cyclooxygenase‑2 (COX-2) Inhibitors for Chemoprevention of Colorectal Cancer von Zhang, Zhuming, Ghosh, Avijit, Connolly, Peter J, King, Peter, Wilde, Thomas, Wang, Jianyao, Dong, Yawei, Li, Xueliang, Liao, Daohong, Chen, Hao, Tian, Gaochao, Suarez, Javier, Bonnette, William G, Pande, Vineet, Diloreto, Karen A, Shi, Yifan, Patel, Shefali, Pietrak, Beth, Szewczuk, Lawrence, Sensenhauser, Carlo, Dallas, Shannon, Edwards, James P, Bachman, Kurtis E, Evans, David C

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Preparation of 4′‐Spirocyclobutyl Nucleoside Analogues as Novel and Versatile Adenosine Scaffolds von Verhoeven, Jonas, De Vleeschouwer, Freija, Kong, Hanchu, Van Hecke, Kristof, Pande, Vineet, Sun, Weimei, Vos, Ann, Wu, Tongfei, Meerpoel, Lieven, Thuring, Jan Willem, Verniest, Guido

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Structural diversity of the epigenetics pocketome von Cabaye, Alexandre, Nguyen, Kong T, Liu, Lihua, Pande, Vineet, Schapira, Matthieu

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Pharmacological Characterization of JNJ-75276617, a Menin-KMT2A Inhibitor, As Targeted Treatment for KMT2A-Altered and NPM1-Mutant Acute Leukemia von Kwon, Min Chul, Querolle, Olivier, Dai, Xuedong, Thuring, Jan Willem, Verhulst, Tinne, Marien, Ann, Goffin, Dries, Cai, Wei, Keersmaekers, Vikki, Eyassu, Filmon, Verstraeten, Karin, El Ashkar, Sara, Hogeling, Shanna M, Jacob, Frank, Vinken, Petra, Darville, Nicolas, Pande, Vineet, Krosky, Daniel, Urbanietz, Gregor, Verbist, Bie, Ferrante, Lucille A., Drenberg, Christina Diane, Wilson, David, Attar, Ricardo M., Schuringa, Jan Jacob, Daskalakis, Nikki, Packman, Kathryn, Pietsch, Christine, Elsayed, Yusri, Philippar, Ulrike

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2,4-Diaminoquinazolines as Dual Toll-like Receptor (TLR) 7/8 Modulators for the Treatment of Hepatitis B Virus von Embrechts, Werner, Herschke, Florence, Pauwels, Frederik, Stoops, Bart, Last, Stefaan, Pieters, Serge, Pande, Vineet, Pille, Geert, Amssoms, Katie, Smyej, Ilham, Dhuyvetter, Deborah, Scholliers, Annick, Mostmans, Wendy, Van Dijck, Kris, Van Schoubroeck, Bertrand, Thone, Tine, De Pooter, Dorien, Fanning, Gregory, Jonckers, Tim H. M, Horton, Helen, Raboisson, Pierre, McGowan, David

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Evans Blue is an inhibitor of nuclear factor-kappa B (NF-κB)-DNA binding von Sharma, Rakesh K., Otsuka, Masami, Pande, Vineet, Inoue, Jun-ichiro, João Ramos, Maria

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