Strategies at the Interface of Drug Discovery and Development: Early Optimization of the Solid State Phase and Preclinical Toxicology Formulation for Potential Drug Candidates von Palucki, Michael, Higgins, John D, Kwong, Elizabeth, Templeton, Allen C

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The Mechanistic Basis for Electronic Effects on Enantioselectivity in the (salen)Mn(III)-Catalyzed Epoxidation Reaction von Palucki, Michael, Finney, Nathaniel S, Pospisil, Paul J, Güler, Mehmet L, Ishida, Toyohisa, Jacobsen, Eric N

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First Generation Process for the Preparation of the DPP-IV Inhibitor Sitagliptin von Hansen, Karl B, Balsells, Jaume, Dreher, Spencer, Hsiao, Yi, Kubryk, Michele, Palucki, Michael, Rivera, Nelo, Steinhuebel, Dietrich, Armstrong, Joseph D, Askin, David, Grabowski, Edward J. J

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Synthesis of Oxygen Heterocycles via a Palladium-Catalyzed C−O Bond-Forming Reaction von Palucki, Michael, Wolfe, John P., Buchwald, Stephen L.

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A Practical Synthesis of 5-Lipoxygenase Inhibitor MK-0633 von Gosselin, Francis, Britton, Robert A, Davies, Ian W, Dolman, Sarah J, Gauvreau, Danny, Hoerrner, R. Scott, Hughes, Gregory, Janey, Jacob, Lau, Stephen, Molinaro, Carmela, Nadeau, Christian, O’Shea, Paul D, Palucki, Michael, Sidler, Rick

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Palladium-Catalyzed Intermolecular Carbon−Oxygen Bond Formation:  A New Synthesis of Aryl Ethers von Palucki, Michael, Wolfe, John P, Buchwald, Stephen L

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Highly Enantioselective, Low-Temperature Epoxidation of Styrene von Palucki, Michael, Pospisil, Paul J, Zhang, Wei, Jacobsen, Eric N

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Efficient Access to Azaindoles and Indoles von McLaughlin, Mark, Palucki, Michael, Davies, Ian W

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Solvent-Dependent Dynamic Kinetic Asymmetric Transformation/Kinetic Resolution in Molybdenum-catalyzed Asymmetric Allylic Alkylations von Hughes, David L, Palucki, Michael, Yasuda, Nobuyoshi, Reamer, Robert A, Reider, Paul J

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Palladium-Catalyzed α-Arylation of Ketones von Palucki, Michael, Buchwald, Stephen L

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Efficient Access to Cyclic Ureas via Pd-Catalyzed Cyclization von McLaughlin, Mark, Palucki, Michael, Davies, Ian W

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Development of a New and Practical Route to Chiral 3,4-Disubstituted Cyclopentanones:  Asymmetric Alkylation and Intramolecular Cyclopropanation as Key C−C Bond-Forming Steps von Palucki, Michael, Um, Joann M, Yasuda, Nobuyoshi, Conlon, David A, Tsay, Fuh-Rong, Hartner, Frederick W, Hsiao, Yi, Marcune, Benjamin, Karady, Sandor, Hughes, David L, Dormer, Peter G, Reider, Paul J

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Stereoselective Enol Tosylation:  Preparation of Trisubstituted α,β-Unsaturated Esters von Baxter, Jenny M, Steinhuebel, Dietrich, Palucki, Michael, Davies, Ian W

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On the Viability of Oxametallacyclic Intermediates in the (salen)Mn-Catalyzed Asymmetric Epoxidation von Finney, Nathaniel S., Pospisil, Paul J., Chang, Sukbok, Palucki, Michael, Konsler, Reed G., Hansen, Karl B., Jacobsen, Eric N.

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Asymmetric Arylation of Ketone Enolates von Åhman, Jens, Wolfe, John P, Troutman, Malisa V, Palucki, Michael, Buchwald, Stephen L

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Synthesis of N-arylated sultams: palladium- and copper-catalyzed cross coupling of aryl halides with 1,4-butane and 1,3-propanesultams von Steinhuebel, Dietrich, Palucki, Michael, Askin, David, Dolling, Ulf

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Low Temperature Asymmetric Epoxidation of Unfunctionalized Olefins Catalyzed by (Salen)Mn(III) Complexes von Palucki, M

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A highly efficient enantioselective synthesis of 2-methyl chromans via four sequential palladium-catalyzed reactions von Palucki, Michael, Yasuda, Nobuyoshi

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Asymmetric Hydrogenation of Protected Allylic Amines von Steinhuebel, Dietrich P, Krska, Shane W, Alorati, Anthony, Baxter, Jenny M, Belyk, Kevin, Bishop, Brian, Palucki, Michael, Sun, Yongkui, Davies, Ian W

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Designed Ligands as Probes for the Catalytic Binding Mode in Mo-Catalyzed Asymmetric Allylic Alkylation von Trost, Barry M., Dogra, Kalindi, Hachiya, Iwao, Emura, Takashi, Hughes, David L., Krska, Shane, Reamer, Robert A., Palucki, Michael, Yasuda, Nobuyoshi, Reider, Paul J.

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