Structural basis of CX-4945 binding to human protein kinase CK2 von Ferguson, Andrew D., Sheth, Payal R., Basso, Andrea D., Paliwal, Sunil, Gray, Kimberly, Fischmann, Thierry O., Le, Hung V.

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Asymmetric Synthesis of 4,4-Disubstituted-2-Imidazoli-dinones:  Potent NK1 Antagonists von Reichard, Gregory A, Stengone, Carmine, Paliwal, Sunil, Mergelsberg, Ingrid, Majmundar, Sapna, Wang, Cheng, Tiberi, Robert, McPhail, Andrew T, Piwinski, John J, Shih, Neng-Yang

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Design and biological characterization of a series of dual mechanism ERK1/2 inhibitors with a Triazolopyridinone core von Lotfaliansaremi, Sajedeh, Cornwell, Stephen, Casillas, Candice, Sabio, Michael, Tolias, Peter, Windsor, William, Paliwal, Sunil

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Discovery of ZN-c3, a Highly Potent and Selective Wee1 Inhibitor Undergoing Evaluation in Clinical Trials for the Treatment of Cancer von Huang, Peter Q, Boren, Brant C, Hegde, Sayee G, Liu, Hui, Unni, Aditya K, Abraham, Sunny, Hopkins, Chad D, Paliwal, Sunil, Samatar, Ahmed A, Li, Jiali, Bunker, Kevin D

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Discovery of a novel ERK inhibitor with activity in models of acquired resistance to BRAF and MEK inhibitors von Morris, Erick J, Jha, Sharda, Restaino, Clifford R, Dayananth, Priya, Zhu, Hugh, Cooper, Alan, Carr, Donna, Deng, Yongi, Jin, Weihong, Black, Stuart, Long, Brian, Liu, Jenny, Dinunzio, Edward, Windsor, William, Zhang, Rumin, Zhao, Shuxia, Angagaw, Minilik H, Pinheiro, Elaine M, Desai, Jagdish, Xiao, Li, Shipps, Gerald, Hruza, Alan, Wang, James, Kelly, Joe, Paliwal, Sunil, Gao, Xiaolei, Babu, Boga Sobhana, Zhu, Liang, Daublain, Pierre, Zhang, Ling, Lutterbach, Bart A, Pelletier, Marc R, Philippar, Ulrike, Siliphaivanh, Phieng, Witter, David, Kirschmeier, Paul, Bishop, W Robert, Hicklin, Daniel, Gilliland, D Gary, Jayaraman, Lata, Zawel, Leigh, Fawell, Stephen, Samatar, Ahmed A

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Cyclic urea derivatives as potent NK1 selective antagonists. Part II: Effects of fluoro and benzylic methyl substitutions von Shue, Ho-Jane, Chen, Xiao, Schwerdt, John H, Paliwal, Sunil, Blythin, David J, Lin, Ling, Gu, Danlin, Wang, Cheng, Reichard, Gregory A, Wang, Hongwu, Piwinski, John J, Duffy, Ruth A, Lachowicz, Jean E, Coffin, Vicki L, Nomeir, Amin A, Morgan, Cynthia A, Varty, Geoffrey B, Shih, Neng-Yang

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Measurements of Molecular Electrostatic Field Effects in Edge-to-Face Aromatic Interactions and CH-π Interactions with Implications for Protein Folding and Molecular Recognition von Kim, Eun-il, Paliwal, Sunil, Wilcox, Craig S

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Discovery of 3(S)-thiomethyl pyrrolidine ERK inhibitors for oncology von Boga, Sobhana Babu, Alhassan, Abdul-Basit, Cooper, Alan B., Doll, Ronald, Shih, Neng-Yang, Shipps, Gerald, Deng, Yongqi, Zhu, Hugh, Nan, Yang, Sun, Robert, Zhu, Liang, Desai, Jagdish, Patel, Mehul, Muppalla, Kiran, Gao, Xiaolei, Wang, James, Yao, Xin, Kelly, Joseph, Gudipati, Subrahmanyam, Paliwal, Sunil, Tsui, Hon-Chung, Wang, Tong, Sherborne, Bradley, Xiao, Li, Hruza, Alan, Buevich, Alexei, Zhang, Li-Kang, Hesk, David, Samatar, Ahmed A., Carr, Donna, Long, Brian, Black, Stuart, Dayananth, Priya, Windsor, William, Kirschmeier, Paul, Bishop, Robert

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MK-8353: Discovery of an Orally Bioavailable Dual Mechanism ERK Inhibitor for Oncology von Boga, Sobhana Babu, Deng, Yongqi, Zhu, Liang, Nan, Yang, Cooper, Alan B., Shipps, Gerald W., Doll, Ronald, Shih, Neng-Yang, Zhu, Hugh, Sun, Robert, Wang, Tong, Paliwal, Sunil, Tsui, Hon-Chung, Gao, Xiaolei, Yao, Xin, Desai, Jagdish, Wang, James, Alhassan, Abdul Basit, Kelly, Joseph, Patel, Mehul, Muppalla, Kiran, Gudipati, Subrahmanyam, Zhang, Li-Kang, Buevich, Alexei, Hesk, David, Carr, Donna, Dayananth, Priya, Black, Stuart, Mei, Hong, Cox, Kathleen, Sherborne, Bradley, Hruza, Alan W., Xiao, Li, Jin, Weihong, Long, Brian, Liu, Gongjie, Taylor, Stacey A., Kirschmeier, Paul, Windsor, William T., Bishop, Robert, Samatar, Ahmed A.

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Potent and Selective Amidopyrazole Inhibitors of IRAK4 That Are Efficacious in a Rodent Model of Inflammation von McElroy, William T., Tan, Zheng, Ho, Ginny, Paliwal, Sunil, Li, Guoqing, Seganish, W. Michael, Tulshian, Deen, Tata, James, Fischmann, Thierry O., Sondey, Christopher, Bian, Hong, Bober, Loretta, Jackson, James, Garlisi, Charles G., Devito, Kristine, Fossetta, James, Lundell, Daniel, Niu, Xiaoda

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Structure-based drug design of clinical compound MK-8353, a novel inhibitor of ERK von Hruza, Alan, Boga, Sobhana Babu, Alhassan, Abdul-Basit, Cooper, Alan B., Doll, Ronald, Shih, Neng-Yang, Shipps, Gerald, Deng, Yongqi, Zhu, Hugh, Nan, Yang, Sun, Robert, Zhu, Liang, Desai, Jagdish, Patel, Mehul, Muppalla, Kiran, Gao, Xiaolei, Wang, James, Kelly, Joseph, Gudipati, Subrahmanyam, Paliwal, Sunil, Tsui, Hon-Chung, Wang, Tong, Sherborne, Bradley, Xiao, Li, Buevich, Alexei, Hesk, David, Samatar, Ahmed A., Carr, Donna, Long, Brian, Black, Stuart, Dayananth, Priya, Windsor, William, Kirschmeier, Paul, Bishop, Robert

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Thermally stimulated current and electrical conduction in metal (1)-ethyl cellulose-metal (1)/(2) systems von Khare, P K, Verma, Ashish, Paliwal, Sunil K

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Discovery of a series of potent, orally active α,α-disubstituted piperidine NK1 antagonists von DONG XIAO, CHENG WANG, VARTY, Geoffrey, MORGAN, Cynthia, FEI LIU, NOMEIR, Amin, PALANI, Anandan, TSUI, Hon-Chung, REICHARD, Gregory, PALIWAL, Sunil, SHIH, Neng-Yang, ASLANIAN, Robert, DUFFY, Ruth, LACHOWICZ, Jean

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Discovery of a series of potent, orally active alpha , alpha -disubstituted piperidine NK sub(1 antagonists) von Xiao, Dong, Wang, Cheng, Palani, Anandan, Tsui, Hon-Chung, Reichard, Gregory, Paliwal, Sunil, Shih, Neng-Yang, Aslanian, Robert, Duffy, Ruth, Lachowicz, Jean, Varty, Geoffrey, Morgan, Cynthia, Liu, Fei, Nomeir, Amin

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Cyclobutane derivatives as potent NK1 selective antagonists von WROBLESKI, Michelle Laci, REICHARD, Gregory A, PALIWAL, Sunil, SHAH, Sapna, TSUI, Hon-Chung, DUFFY, Ruth A, LACHOWICZ, Jean E, MORGAN, Cynthia A, VARTY, Geoffrey B, SHIH, Neng-Yang

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MULTICYCLIC COMPOUNDS von CRIPE, Lawrence, PALIWAL, Sunil, SAMATAR, Ahmed Abdi

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Cyclic urea derivatives as potent NK1 selective antagonists von SHUE, Ho-Jane, XIAO CHEN, PIWINSKI, John J, DUFFY, Ruth A, LACHOWICZ, Jean E, COFFIN, Vicki L, FEI LIU, NOMEIR, Amin A, MORGAN, Cynthia A, VARTY, Geoffrey B, SHIH, Neng-Yang, BLYTHIN, David J, PALIWAL, Sunil, LING LIN, DANLIN GU, SCHWERDT, John H, SHAH, Sapna, REICHARD, Gregory A

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Discovery of a series of potent, orally active α,α-disubstituted piperidine NK 1 antagonists von Xiao, Dong, Wang, Cheng, Palani, Anandan, Tsui, Hon-Chung, Reichard, Gregory, Paliwal, Sunil, Shih, Neng-Yang, Aslanian, Robert, Duffy, Ruth, Lachowicz, Jean, Varty, Geoffrey, Morgan, Cynthia, Liu, Fei, Nomeir, Amin

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MULTICYCLIC COMPOUNDS von PALIWAL, Sunil, SAMATAR, Ahmed Abdi, CRIPE, Lawrence Saunders

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MULTICYCLIC COMPOUNDS von Cripe, Lawrence Saunders, Paliwal, Sunil, Samatar, Ahmed Abdi

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